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A Study of the Safety and Pharmacokinetics of SAR245409 Tablets in Patients With Solid Tumors or Lymphoma

Phase 1
Completed
Conditions
Neoplasm Malignant
Interventions
Registration Number
NCT01596270
Lead Sponsor
Sanofi
Brief Summary

Primary Objective:

- To evaluate the safety and tolerability of SAR245409 tablets administered once or twice a day in patients with solid tumors or lymphoma.

Secondary Objectives:

* To evaluate blood levels of SAR245409 after administration of SAR245409 tablets once or twice a day in patients with solid tumors or lymphoma.

* To evaluate the effect of food on blood levels of SAR245409 after administration of SAR245409 tablets in patients with solid tumors or lymphoma.

* To evaluate the effect of SAR245409 on the body after administration of SAR245409 tablets once or twice a day in patients with solid tumors or lymphoma.

* To obtain information on how SAR245409 administered once or twice a day to patients with solid tumors or lymphoma affect disease symptoms and study treatment side effects as reported by the patients on a questionnaire.

* To explore the antitumor activity of SAR245409 tablets administered once or twice a day to patients with solid tumors or lymphoma.

Detailed Description

The total study duration per patient will be 58 to 128 days and will include a screening period (1 to 28 days), a food interaction investigation period (when applicable; 4 to 11 days), two 28-day treatment cycles (56 days), an end-of-treatment visit (within 7 days after the last SAR245409 administration) and a follow-up visit (within 30 ± 3 days after the last SAR245409 administration).

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
49
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Twice daily dosingSAR245409escalating doses, twice daily dosing every day, no eating for 2 hours prior and 1 hour after dose
Once daily dosingSAR245409escalating doses, once daily dosing every day, no eating for 2 hours prior and 1 hour after dose
Primary Outcome Measures
NameTimeMethod
Dose Limiting ToxicitiesUp to Day 28
Secondary Outcome Measures
NameTimeMethod
Maximum SAR245409 plasma concentrationCycle 1 Days 1, 2, 8, 15, and 28, and Cycle 2 Day 1
Number of patients with treatment-emergent adverse eventsFrom first dose of SAR245409 until 30 days after the last dose
Area under the SAR245409 plasma concentration versus time curveCycle 1 Days 1, 2, 8, 15, and 28, and Cycle 2 Day 1
Ratio of maximum SAR245409 plasma concentration between fed and fasted dosingDays 1, 2, 3, and 4 of the food interaction period
Ratio of area under the SAR245409 plasma concentration versus time curve between fed and fasted dosingDays 1, 2, 3, and 4 of the food interaction period

Trial Locations

Locations (3)

Investigational Site Number 840001

🇺🇸

Detroit, Michigan, United States

Investigational Site Number 840002

🇺🇸

New Brunswick, New Jersey, United States

Investigational Site Number 840003

🇺🇸

Dallas, Texas, United States

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