MedPath

A Study of Insulin Efsitora Alfa (LY3209590) Compared With Insulin Degludec in Participants With Type 2 Diabetes Currently Treated With Basal Insulin

Phase 3
Completed
Conditions
Type 2 Diabetes
Interventions
Registration Number
NCT05275400
Lead Sponsor
Eli Lilly and Company
Brief Summary

The reason for this study is to see if the study drug insulin efsitora alfa (LY3209590) is safe and effective in participants with Type 2 diabetes that have already been treated with basal insulin. The study consists of a 3-week screening/lead-in period, a 78-week treatment period and a 5-week safety follow-up period. The study will last up to 86 weeks.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
986
Inclusion Criteria
  • Have been diagnosed with Type 2 diabetes according to the World Health Organization (WHO) criteria treated with basal insulin

  • Are receiving ≥10 units of basal insulin per day and ≤110 units per day at screening

  • Have HbA1c value of 6.5% - 10% inclusive, at screening

  • Have a Body mass index (BMI) less than or equal to 45 kilogram/square meter (kg/m²)

  • Have been treated with one of the following stable insulin regimens at least 90 days prior to screening:

    • once daily U100 or U200 of insulin degludec
    • once daily U100 or U300 of insulin glargine
    • once or twice daily U100 of insulin detemir, or
    • once or twice daily human insulin NPH
  • acceptable non insulin glucose lowering therapies may include 0 to up to 3 of the following:

    • dipeptidyl peptidase (DPP-4) IV inhibitors
    • SGLT2 inhibitors
    • metformin
    • alphaglucosidase inhibitors or,
    • Glucagon-Like Peptide-1 (GLP-1) receptor agonists
    • Participants must be willing to stay on stable dose throughout the study
Exclusion Criteria
  • Have Type 1 diabetes mellitus

  • Have acute or chronic hepatitis, cirrhosis, or obvious clinical signs or symptoms of any other liver disease, except Nonalcoholic Fatty Liver Disease (NAFLD)

  • Estimated glomerular filtration rate (eGFR) <20 milliliters/minute/1.73 square meter (m²)

  • Have active or untreated malignancy

  • Are pregnant

  • Have a significant weight gain or loss the past 3 months

  • Have received anytime in the past 6 months, any of the following insulin therapies:

    • prandial insulin
    • insulin mixtures
    • inhaled insulin
    • U-500 insulin, or
    • continuous subcutaneous insulin infusion therapy
  • Have had any of New York Heart Association Class IV heart failure or any of the following CV conditions in the past 3 months:

    • acute myocardial infarctions
    • cerebrovascular accident (stroke), or
    • coronary bypass surgery
  • Gastrointestinal: have undergone gastric bypass (bariatric) surgery, restrictive bariatric surgery (Lap-Band) or sleeve gastrectomy within 1 year prior to screening

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Insulin DegludecInsulin DegludecParticipants with be given insulin degludec SC.
Insulin Efsitora AlfaInsulin Efsitora AlfaParticipants will be given insulin efsitora alfa subcutaneously (SC).
Primary Outcome Measures
NameTimeMethod
Change from Baseline in Hemoglobin A1c (HbA1c)Baseline, Week 26

Change from Baseline in HbA1c of insulin efsitora alfa compared to insulin degludec on glycemic control in participants with type 2 diabetes currently on basal insulin.

Secondary Outcome Measures
NameTimeMethod
Weekly Insulin doseWeek 26

The weekly insulin dose calculated based on participant entry of daily or weekly insulin dose in an electronic diary.

Change from Baseline in Fasting GlucoseBaseline, Week 26

Fasting glucose measured by Self-Monitoring of Blood Glucose (SMBG).

Time in Hypoglycemia RangeWeek 22 to Week 26

Time in hypoglycemia range defined as time in hypoglycemia with glucose \<54 mg/dL measured during the CGM session.

Change from Baseline in Treatment-Related Impact Measure - Diabetes (TRIM-D)Baseline, Week 26

TRIM-D assesses the impact of diabetes treatment on participants' functioning and well-being across available diabetes treatment.

Time in RangeWeek 22 to Week 26

Time in glucose range between 70 and 180 mg/dL inclusive measured by continued glucose monitoring (CGM) during a 4-week CGM session.

Level 2 or Level 3 Nocturnal Hypoglycemia Event RateBaseline to Week 78

The event rate of participant-reported clinically significant nocturnal hypoglycemia (\<54 milligram/deciliter (mg/dL) or severe) measured during treatment phase.

Time in Hyperglycemia RangeWeek 22 to Week 26

Time in hyperglycemia range defined as time in hyperglycemia with glucose \>180 mg/dL measured during the CGM session.

Nocturnal Hypoglycemia Event RateBaseline to Week 78

The event rate of participant-reported clinically significant nocturnal hypoglycemia (\<54 milligram/deciliter (mg/dL) or severe) measured during treatment phase up to Week 78.

Change from Baseline in Body WeightBaseline, Week 78

Change from baseline in body weight

Change from Baseline in Diabetes Treatment Satisfaction Questionnaire-Status Version (DTSQ)Baseline, Week 78

DTSQ assesses the overall treatment satisfaction and perceived frequency of hyperglycemia and hypoglycemia.

Trial Locations

Locations (127)

Diabetes Associates Medical Group

🇺🇸

Orange, California, United States

Rocky Mountain Clinical Research

🇺🇸

Idaho Falls, Idaho, United States

SKY Clinical Research Network Group - Hall

🇺🇸

Fayette, Mississippi, United States

Clinvest Research LLC

🇺🇸

Springfield, Missouri, United States

Lillestol Research

🇺🇸

Fargo, North Dakota, United States

NYC Research

🇺🇸

New York, New York, United States

Centro Medico Privado CEMAIC

🇦🇷

Capital, Córdoba, Argentina

Centro Diabetológico Dr. Waitman

🇦🇷

Córdoba, Argentina

CENUDIAB

🇦🇷

Ciudad Autónoma de Buenos Aire, Argentina

Tokuyama Clinic

🇯🇵

Mihama-ku,Chiba City, Chiba, Japan

Strazsahegy Medicina Bt.

🇭🇺

Budapest, Hungary

Nakamoto Internal Medicine Clinic

🇯🇵

Mito, Ibaraki, Japan

The Institute of Medical Science, Asahi Life Foundation

🇯🇵

Chuo-ku, Tokyo, Japan

Inje University Sanggye Paik Hospital

🇰🇷

Seoul, Seoul-teukbyeolsi [Seoul], Korea, Republic of

Severance Hospital, Yonsei University Health System

🇰🇷

Seoul, Seoul-teuk, Korea, Republic of

Centrum Badan Klinicznych PI-House sp. z o.o.

🇵🇱

Gdansk, Pomorskie, Poland

Centrum Terapii Wspolczesnej J. M. Jasnorzewska Spolka Komandytowo-Akcyjna

🇵🇱

Lodz, Łódzkie, Poland

MediVet s.r.o.

🇸🇰

Malacky, Bratislavský Kraj, Slovakia

MEDI-DIA s.r.o.

🇸🇰

Sabinov, Prešovský Kraj, Slovakia

CHUAC-Complejo Hospitalario Universitario A Coruña

🇪🇸

A Coruña, A Coruña [La Coruña], Spain

ENDIAMED s.r.o

🇸🇰

Dolny Kubin, Žilinský Kraj, Slovakia

Hospital Universitario Virgen de la Victoria

🇪🇸

Malaga, Andalucía, Spain

Clínica Juaneda

🇪🇸

Palma de Mallorca, Balears [Baleares], Spain

Hospital Quiron Infanta Luisa

🇪🇸

Sevilla, Andalucía, Spain

Centro Periférico de Especialidades Bola Azul

🇪🇸

Almeria, Almería, Spain

Hospital Universitari Vall d'Hebron

🇪🇸

Barcelona, Barcelona [Barcelona], Spain

Hospital Universitario de La Ribera

🇪🇸

Alzira, Valenciana, Comunitat, Spain

Hospital Universitario Marqués de Valdecilla

🇪🇸

Santander, Cantabria, Spain

Hospital General Universitario de Valencia

🇪🇸

Valencia, Valenciana, Comunitat, Spain

Taichung Veterans General Hospital

🇨🇳

Taichung City, Taichung, Taiwan

Centro de Investigaciones Metabólicas (CINME)

🇦🇷

Ciudad Autónoma de Buenos Aire, Buenos Aires, Argentina

Go Centro Medico San Nicolás

🇦🇷

San Nicolas, Buenos Aires, Argentina

Consultorio de Investigación Clínica EMO SRL

🇦🇷

Ciudad Autonoma de Buenos Aire, Buenos Air, Argentina

Stat Research S.A.

🇦🇷

Ciudad Autónoma de Buenos Aire, Buenos Air, Argentina

Mautalen Salud e Investigación

🇦🇷

Buenos Aires, Ciudad Aut, Argentina

Medical Investigations

🇺🇸

Little Rock, Arkansas, United States

CIPADI - Centro Integral de Prevencion y Atencion en Diabetes

🇦🇷

Godoy Cruz, Mendoza, Argentina

Zala Megyei Szent Rafael Kórház

🇭🇺

Zalaegerszeg, Zala, Hungary

Noritake Clinic

🇯🇵

Ushiku, Ibaraki, Japan

Matoba Internal Medicine Clinic

🇯🇵

Ebina, Kanagawa, Japan

Medical Corporation Yuga Tsuruma Kaneshiro Diabetes Clinic

🇯🇵

Yamato-shi, Kanagawa, Japan

Yeungnam Univeristy Medical Center

🇰🇷

Gyeongsan-si, Kyǒngsangbuk-do, Korea, Republic of

GCM Medical Group, PSC - Hato Rey Site

🇵🇷

San Juan, Puerto Rico

Human Care s.r.o.

🇸🇰

Kosice, Košický Kraj, Slovakia

Diacrin .s.ro.

🇸🇰

Bratislava, Slovakia

Fu Jen Catholic University Hospital

🇨🇳

New Taipei, Taiwan

West Orange Endocrinology

🇺🇸

Ocoee, Florida, United States

Chase Medical Research, LLC

🇺🇸

Waterbury, Connecticut, United States

Encore Medical Research

🇺🇸

Hollywood, Florida, United States

Instituto de Investigaciones Clínicas Mar del Plata

🇦🇷

Mar del Plata, Buenos Aires, Argentina

Suncoast Clinical Research, Inc.

🇺🇸

New Port Richey, Florida, United States

DRC Gyógyszervizsgáló Központ

🇭🇺

Balatonfüred, Veszprém, Hungary

Kanizsai Dorottya Korhaz

🇭🇺

Nagykanizsa, Zala, Hungary

Takai Internal Medicine Clinic

🇯🇵

Kamakura-shi, Kanagawa, Japan

Shiraiwa Medical Clinic

🇯🇵

Kashiwara, Osaka, Japan

Abe Clinic

🇯🇵

Oita, Japan

Korea University Ansan Hospital

🇰🇷

Ansan-si, Kyǒnggi-do, Korea, Republic of

Seoul National University Hospital

🇰🇷

Seoul, Seoul-teukbyeolsi [Seoul], Korea, Republic of

Hallym University Kangnam Sacred Heart Hospital

🇰🇷

Seoul, Seoul-teukbyeolsi [Seoul], Korea, Republic of

Kyung Hee University Hospital at Gangdong

🇰🇷

Seoul, Seoul-teukbyeolsi [Seoul], Korea, Republic of

NZOZ Przychodnia Specjalistyczna Andrzej Wittek, Henryk Rudzki

🇵🇱

Ruda Slaska, Śląskie, Poland

Areteus s.r.o.

🇸🇰

Trebisov, Košický Kraj, Slovakia

Arcturus Healthcare , PLC, Troy Internal Medicine Research Division

🇺🇸

Troy, Michigan, United States

Instituto Centenario

🇦🇷

Caba, Ciudad Autónoma De Buenos Aire, Argentina

Kozawa Eye Hospital and Diabetes Center

🇯🇵

Mito, Ibaraki, Japan

Oyama East Clinic

🇯🇵

Oyama, Tochigi, Japan

CenterMed Lublin NZOZ

🇵🇱

Lublin, Lubelskie, Poland

OMEDICA Medical Center

🇵🇱

Poznan, Wielkopolskie, Poland

DIA-MED CENTRUM s.r.o.

🇸🇰

Puchov, Slovakia

Endocrine and Metabolic Consultants

🇺🇸

Rockville, Maryland, United States

Instituto Médico Catamarca IMEC

🇦🇷

Rosario, Santa Fe, Argentina

Centro Médico Viamonte

🇦🇷

Buenos Aires, Ciudad Aut, Argentina

CEMEDIC

🇦🇷

Buenos Aires, Argentina

Shimizu Clinic Fusa

🇯🇵

Saitama-shi, Saitama, Japan

Tokyo-Eki Center-building Clinic

🇯🇵

Chuo Ku, Tokyo, Japan

Medical Corporation Chiseikai Tokyo Center Clinic

🇯🇵

Chuo-ku, Tokyo, Japan

Yonsei University-Wonju Severance Christian Hospital

🇰🇷

Wonju, Kang-won-do, Korea, Republic of

Hanyang University Guri Hospital

🇰🇷

Guri-si, Kyǒnggi-do, Korea, Republic of

Szent Margit Rendelointézet

🇭🇺

Budapest, Hungary

Szent János Kórház

🇭🇺

Budapest, Hungary

Taipei Veterans General Hospital

🇨🇳

Taipei, Taiwan

Yuri Ono Clinic

🇯🇵

Sapporo, Hokkaido, Japan

Takatsuki Red Cross Hospital

🇯🇵

Takatsuki, Osaka, Japan

Fukuwa Clinic

🇯🇵

Chuo-ku, Tokyo, Japan

Jinnouchi Hospital

🇯🇵

Kumamoto, Japan

Heiwadai Hospital

🇯🇵

Miyazaki, Japan

AMC Nishiumeda Clinic

🇯🇵

Osaka, Japan

Kangwon National University Hospital

🇰🇷

Chuncheon-si, Kang-won-do, Korea, Republic of

Asan Medical Center

🇰🇷

Seoul, Seoul-teukbyeolsi [Seoul], Korea, Republic of

Ulsan University Hospital

🇰🇷

Ulsan, Ulsan-Kwangyǒkshi, Korea, Republic of

NZOZ Medica

🇵🇱

Lublin, Lubelskie, Poland

NZOZ Diab-Endo-Met

🇵🇱

Krakow, Małopolskie, Poland

Private Practice - Dr. Robert Witek

🇵🇱

Tarnów, Małopolskie, Poland

Gaja Poradnie Lekarskie Maciej Wiza

🇵🇱

Poznan, Wielkopolskie, Poland

IRMED

🇵🇱

Piotrkow Trybunalski, Łódzkie, Poland

Mgcendo Llc

🇵🇷

San Juan, Puerto Rico

Vithas Hospital Sevilla

🇪🇸

Seville, Sevilla, Spain

Chi Mei Medical Center

🇨🇳

Tainan City, Tainan, Taiwan

National Cheng Kung University Hospital

🇨🇳

Tainan, Taiwan

Chung Shan Medical University Hospital

🇨🇳

Taichung City, Taichung, Taiwan

John Muir Physician Network Research Center

🇺🇸

Concord, California, United States

AMCR Institute

🇺🇸

Escondido, California, United States

National Research Institute - Huntington Park

🇺🇸

Huntington Park, California, United States

University Clinical Investigators, Inc.

🇺🇸

Tustin, California, United States

Scripps Whittier Diabetes Institute

🇺🇸

La Jolla, California, United States

Balanced Life Health Care Solutions/SKYCRNG

🇺🇸

Lawrenceville, Georgia, United States

Iowa Diabetes and Endocrinology Research Center

🇺🇸

West Des Moines, Iowa, United States

Albany Medical College, Division of Community Endocrinology

🇺🇸

Albany, New York, United States

Aventiv Research Inc

🇺🇸

Columbus, Ohio, United States

Intend Research, LLC

🇺🇸

Norman, Oklahoma, United States

Heritage Valley Medical Group, Inc.

🇺🇸

Beaver, Pennsylvania, United States

Jefferson Clinical Research Institute (JCRI)

🇺🇸

Philadelphia, Pennsylvania, United States

Preferred Primary Care Physicians

🇺🇸

Uniontown, Pennsylvania, United States

Dallas Diabetes Research Center

🇺🇸

Dallas, Texas, United States

Juno Research

🇺🇸

Houston, Texas, United States

Biopharma Informatic, LLC

🇺🇸

Houston, Texas, United States

Texas Diabetes & Endocrinology, P.A.

🇺🇸

Round Rock, Texas, United States

Southern Endocrinology Associates

🇺🇸

Mesquite, Texas, United States

Consano Clinical Research, LLC

🇺🇸

Shavano Park, Texas, United States

Rainier Clinical Research Center

🇺🇸

Renton, Washington, United States

Gabinety TERPA

🇵🇱

Lublin, Lubelskie, Poland

Clínica nuevas Tecnologías en Diabetes y Endocrinología (NTDE)

🇪🇸

Sevilla, Spain

New Horizon Research Center

🇺🇸

Miami, Florida, United States

L-MARC Research Center

🇺🇸

Louisville, Kentucky, United States

HealthPartners Institute dba International Diabetes Center

🇺🇸

Minneapolis, Minnesota, United States

Palm Research Center Tenaya

🇺🇸

Las Vegas, Nevada, United States

Gadolin Research

🇺🇸

Beaumont, Texas, United States

© Copyright 2025. All Rights Reserved by MedPath