MedPath

Safety and Efficacy Study of GRT6005 in Patients With Osteoarthritis (OA) Knee Pain

Phase 2
Completed
Conditions
Moderate to Severe Chronic Pain Due to Osteoarthritis of the Knee
Interventions
Registration Number
NCT01709214
Lead Sponsor
Tris Pharma, Inc.
Brief Summary

The purpose of this study is to evaluate the safety and efficacy of GRT6005 compared to placebo in patients with moderate to severe chronic pain due to osteoarthritis (OA) of the knee. This study includes a maximum 21 day Screening Period followed by a 15-week Double-blind Treatment Period and a 4-7 day Safety Follow-up period. Patients who are eligible for the Double-blind Treatment Period will be randomized to one of following treatment groups: GRT6005 high-dose range (400, 600 or 800 mcg), GRT6005 low-dose range (200, 300 or 400 mcg), oxycodone controlled release (CR) dose range (10, 20, 30, 40 or 50 mg) or placebo.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
619
Inclusion Criteria
  • Diagnosis of osteoarthritis (OA) of the knee
  • OA knee pain present for at least 3 months
  • OA knee pain is the predominant (ie, most painful) pain condition
  • Patients require medication on at least 4 of 7 days per week to treat OA knee pain for at least 1 month.
  • Dissatisfaction with current OA knee pain treatment and willingness to stop taking all pain medications except for the study drug and allowed rescue medication
  • Average daily pain rating of at least 5 on a 0 to 10 point numerical rating scale during the 1 week prior to randomization
  • Female patients either postmenopausal, surgically sterile or practicing a medically acceptable method of contraception
  • Male patients either status post-bilateral vasectomy or using barrier contraception
Exclusion Criteria
  • Knee pain due to a disorder other than OA
  • Other pain that can confound the assessment of, or contribute to, pain at the reference knee
  • Surgery at the reference knee within 6 months of Screening or a history of joint replacement surgery at the reference knee
  • Trauma to the reference knee within 6 months of Screening with active symptoms
  • Steroid injections in the reference knee within 3 months of Screening
  • Hyaluronic acid injections in the reference knee within 6 months of Screening
  • Body Mass Index > 40 kg/m2
  • Patient with any protocol-excluded or clinically significant medical, surgical, or medication history that would limit the patient's ability to complete or participate in this clinical trial or could confound the study assessments

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Cebranopadol (GRT6005) Low-Dose RangePlaceboOnce daily GRT6005, flexible dosing 200, 300 or 400 micrograms, and once daily Placebo; oral administration for 15 weeks
Cebranopadol (GRT6005) High-Dose RangePlaceboOnce daily GRT6005, flexible dosing 400, 600 or 800 micrograms, and once daily Placebo; oral administration for 15 weeks
PlaceboPlaceboTwice daily Placebo, oral administration for 15 weeks
Oxycodone CROxycodone CRTwice daily Oxycodone CR, flexible dosing 10, 20, 30, 40 or 50 milligrams; oral administration for 15 weeks
Cebranopadol (GRT6005) Low-Dose RangeCebranopadol (GRT6005) Low-Dose RangeOnce daily GRT6005, flexible dosing 200, 300 or 400 micrograms, and once daily Placebo; oral administration for 15 weeks
Cebranopadol (GRT6005) High-Dose RangeCebranopadol (GRT6005) High-Dose RangeOnce daily GRT6005, flexible dosing 400, 600 or 800 micrograms, and once daily Placebo; oral administration for 15 weeks
Primary Outcome Measures
NameTimeMethod
Change from baseline in the weekly average of the daily average pain ratingBaseline to end of treatment (Week 15)
Secondary Outcome Measures
NameTimeMethod
Change from baseline in the physical function subscale of the Western Ontario and McMaster University Index of Osteoarthritis Questionnaire (WOMAC)Baseline to end of treatment (Week 15)

Trial Locations

Locations (83)

Site 011

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Bradenton, Florida, United States

Site 061

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Fresno, California, United States

Site 043

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Tustin, California, United States

Site 071

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Clearwater, Florida, United States

Site 058

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Pembroke Pines, Florida, United States

Site 086

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Chicago, Illinois, United States

Site 052

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Marietta, Georgia, United States

Site 001

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Columbus, Ohio, United States

Site 042

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Traverse City, Michigan, United States

Site 069

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Cleveland, Ohio, United States

Site 038

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Dallas, Texas, United States

Site 065

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Seattle, Washington, United States

Site 013

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Miami, Florida, United States

Site 041

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Indianapolis, Indiana, United States

Site 024

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Las Vegas, Nevada, United States

Site 079

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Cincinnati, Ohio, United States

Site 072

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Las Vegas, Nevada, United States

Site 008

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Cincinnati, Ohio, United States

Site 070

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Phoenix, Arizona, United States

Site 040

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San Antonio, Texas, United States

Site 075

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Oklahoma City, Oklahoma, United States

Site 022

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Birmingham, Alabama, United States

Site 035

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Portland, Oregon, United States

Site 018

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Phoenix, Arizona, United States

Site 051

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Birmingham, Alabama, United States

Site 064

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Ogden, Utah, United States

Site 074

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Omaha, Nebraska, United States

Site 023

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Saint Louis, Missouri, United States

Site 031

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Huntsville, Alabama, United States

Site 068

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Albany, New York, United States

Site 005

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Phoenix, Arizona, United States

Site 030

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El Cajon, California, United States

Site 028

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Tucson, Arizona, United States

Site 081

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Chino, California, United States

Site 039

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Fair Oaks, California, United States

Site 080

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Roseville, California, United States

Site 084

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North Hollywood, California, United States

Site 004

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Sacramento, California, United States

Site 044

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San Diego, California, United States

Site 010

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Walnut Creek, California, United States

Site 027

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Westlake Village, California, United States

Site 090

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Edgewater, Florida, United States

Site 060

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Jacksonville, Florida, United States

Site 015

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Jupiter, Florida, United States

Site 003

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New Port Richey, Florida, United States

Site 012

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Ocala, Florida, United States

Site 032

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Orlando, Florida, United States

Site 025

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Ormond Beach, Florida, United States

Site 091

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Pinellas Park, Florida, United States

Site 007

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Sarasota, Florida, United States

Site 033

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Perry, Georgia, United States

Site 073

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Stockbridge, Georgia, United States

Site 077

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Wheaton, Maryland, United States

Site 088

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Towson, Maryland, United States

Site 083

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New Bedford, Massachusetts, United States

Site 021

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North Dartmouth, Massachusetts, United States

Site 016

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Bingham Farms, Michigan, United States

Site 087

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Grand Island, Nebraska, United States

Site 006

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High Point, North Carolina, United States

Site 078

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Wilmington, North Carolina, United States

Site 048

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Toledo, Ohio, United States

Site 029

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Bend, Oregon, United States

Site 034

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Anderson, South Carolina, United States

Site 067

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Medford, Oregon, United States

Site 002

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Duncansville, Pennsylvania, United States

Site 076

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Charleston, South Carolina, United States

Site 009

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Albuquerque, New Mexico, United States

Site 017

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Hartsdale, New York, United States

Site 055

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Austin, Texas, United States

Site 049

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Bryan, Texas, United States

Site 093

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Bristol, Tennessee, United States

Site 089

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San Antonio, Texas, United States

Site 082

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Wichita Falls, Texas, United States

Site 019

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Draper, Utah, United States

Site 059

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Salt Lake City, Utah, United States

Site 092

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Norfolk, Virginia, United States

Site 026

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Virginia Beach, Virginia, United States

Site 066

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Bellevue, Washington, United States

Site 057

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Renton, Washington, United States

Site 085

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Valparaiso, Indiana, United States

Site 020

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Worcester, Massachusetts, United States

Site 045

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Altoona, Pennsylvania, United States

Site 056

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Greensboro, North Carolina, United States

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