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MPC-004 for the Treatment of an Acute Gout Flare

Phase 3
Completed
Conditions
Gout
Interventions
Drug: High Dose Colchicine (4.8 mg total dose)
Drug: Low Dose Colchicine (1.8mg total dose)
Other: Placebo Control
Registration Number
NCT00506883
Lead Sponsor
Takeda
Brief Summary

This study is a multicenter, randomized, double-blind, placebo-controlled, parallel group, dose-comparison to determine the efficacy and safety of a standard-dose of colchicine (4.8 mg) versus low-dose colchicine (1.8 mg) or placebo for acute gout flares.

Detailed Description

This study is a multi-center, randomized, double-blind, placebo-controlled, parallel group trial to compare the efficacy and safety of standard-dose colchicine (STD)(total dose = 4.8 mg) versus low-dose colchicine (total dose 1.8 mg) or placebo for the treatment of acute gout flares. Eight hundred and thirteen patients with a confirmed diagnosis of gout were screened. 238 of the screened patients failed screening; 235(98.7%) failed because they did not meet inclusion/exclusion criteria. The 575 eligible patients were randomly assigned (1:1:1) to one of three treatment groups . At the randomization visit the investigator dispensed a blister card containing eight identical looking capsules (in a combination of active drug and placebo capsules) in a double blind fashion for use during their next gout flare. Patients were instructed to self-initiate treatment with the study medication within 12 hours of a gout flare onset. Gout flares were determined by calling a Gout Flare Call Center established for this purpose. At Investigator discretion, rescue medication could also be provided, but patients were encouraged not to use rescue medication within the first 24 hours after starting treatment with study drug. Of the 575 study participants, 185 had a qualifying gout flare and 390 did not. Patients used a diary to record study drug administration, pain score, the presence or absence of gastrointestinal adverse events (nausea, vomiting, diarrhea, and abdominal pain) and the timing of any rescue medication use prior to beginning treatment and 1, 2, 3, 4, 5, 6, 7, 8, 16, 24, 32, 40, 48, 56, 64, and 72 hours after the start of dosing.

The pain score was based on a scale of 1 - 10 where 1 was no pain and 10 was the worst pain imaginable. Efficacy was defined as a 50% reduction in pain score in the target joint at 24 hours in patients who did not use rescue medicine. The primary efficacy analysis was to be based on an Intent-to-Treat (ITT) population, defined as all patients who were randomized, contacted the Call Center, and were instructed to begin taking study drug. An otherwise qualified patient was excluded from the ITT population only if the patient returned a study drug blister pack completely unused.

Secondary outcome measures compared the efficacy of STD dose colchicine to a low dose regimen and placebo using the same criteria for efficacy as for the primary outcome measure.

Additional secondary outcome measures were time to 50% and 90% reduction in pain in the target joint analyzed by treatment group using Kaplan-Meier methods, and the change in mean pain intensity from 0 to 72 hours plotted by time point for each treatment group.

All safety analyses were carried out using the safety population defined as all patients who received at least one dose of study medication regardless of authorization by the Call Center To determine the safety of colchicine when administered via two different dose regimens all patients who had a gout flare were seen by the investigator as soon as possible after onset and evaluated until the flare and any adverse events resolved. All adverse effects, whether recorded by the patient in the diary or obtained by systematic evaluation by the investigator were recorded and reported in tabular form. Treatment-emergent adverse events (TEAE) were summarized by MedDRA System Organ Class and preferred terms and tabulated according treatment arm, overall incidence, severity and relationship to study medication. Multiple events within a patient were counted once and at greatest severity and closest relationship to study medication.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
185
Inclusion Criteria
  1. Patients of either gender and of any race ≥18 years of age.
  2. If female, patients must be postmenopausal as evidenced by lack of menses for ≥12 consecutive months.
  3. Patients must present with a confirmed diagnosis of gout.
  4. Patients must have experienced ≥2 acute gouty arthritic attacks in the 12 months prior to randomization.
  5. Patients on urate lowering therapy must be on a stable dose and schedule with no changes in therapy for 4 weeks prior to randomization and expected to remain on a stable regimen during study participation.
  6. Patients must be willing to adhere to the study schedule and the protocol requirements.
  7. Patients must be willing and able to give written informed consent. A HIPAA and/or state privacy consent must also be signed.
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Exclusion Criteria
  1. Patients with acute polyarticular gout (>4 joints).
  2. Patients who have experienced >2 acute gouty arthritic attacks per month, or >12 attacks overall, in the 6 months prior to randomization.
  3. Patients with arthritis due to any cause other than gout that may confound any study assessments per Investigator discretion.
  4. Patients with a history of myocardial infarction, unstable angina, cerebrovascular events, or coronary artery bypass grafting within the previous 6 months prior to screening.
  5. Patients with active myeloid leukemia, obstructive gastrointestinal cancer, or metastatic cancer.
  6. Patients with chronic renal dysfunction (creatinine clearance <60 mL/min as estimated with the Cockcroft Gault formula).
  7. Patients with chronic hepatic dysfunction.
  8. Patients with a history of alcohol or substance abuse within the 12 months prior to randomization.
  9. Patients who have any concomitant illness or other finding that, in the opinion of the Investigator, would confound the study data or place the patient at unacceptable risk if the patient were to participate in the study, or that would require frequent adjustments in concomitant medications during the course of the study.
  10. Patients using systemic corticosteroid, cyclosporine, adalimumab, etanercept, infliximab, anakinra, abatacept, mycophenolate, azathioprine, anticoagulants (warfarin, heparin, low molecular weight heparin [LMWH], antithrombin agents, thrombin inhibitors, or selective Factor Xa inhibitors [note, use of aspirin ≤325 mg/day is allowed]), or chronic use of non steroidal anti inflammatory drugs (NSAIDs), acetaminophen, tramadol, and other analgesics such as opiates at screening
  11. Use of any investigational drug within 30 days prior to randomization.
  12. Patients currently participating in another research study or anticipated to enroll in such during participation in this study.
  13. Patients for whom informed consent cannot be obtained.
  14. Patients who have previously been randomized into this study and begun ingestion of study drug.
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Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
High Dose ColchicineHigh Dose Colchicine (4.8 mg total dose)After confirmation of a gout flare, patients were to begin standard dosing of colchicine 4.8mg (two capsules (1.8mg) initially followed by additional one capsule doses (0.6mg) every hour for an additional 6 doses).
Low Dose ColchicineLow Dose Colchicine (1.8mg total dose)Within 12 hours of a confirmed gout flare, patients were to begin the low dose colchicine regimen consisting of a total dose of 1.8 mg - two colchicine capsules initially (1.2 mg)followed an hour later by a single additional capsule of active drug(0.6 mg)then by 5 additional hourly doses of an identical looking placebo capsules
PlaceboPlacebo Control-
Primary Outcome Measures
NameTimeMethod
Responders24 hours after baseline

Responders were defined as patients who achieved a ≥ 50% reduction in target joint pain score from baseline at 24 hours without using rescue drug, using an 11 point scale from 0 to 10, with 10 being the worst pain imaginable after beginning therapy.

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (45)

Medical Research Trust

🇺🇸

Lake Worth, Florida, United States

Bond Clinic

🇺🇸

Winter Haven, Florida, United States

Jacksonville Center for Clinical Research

🇺🇸

Jacksonville, Florida, United States

North Georgia Rheumatology Group, PC

🇺🇸

Lawrenceville, Georgia, United States

Lake County Research Associates

🇺🇸

Libertyville, Illinois, United States

Arthritis & Osteoporosis Center of South Georgia

🇺🇸

Tifton, Georgia, United States

Health Awareness, Inc.

🇺🇸

Jupiter, Florida, United States

Idaho Arthritis & Osteoporosis Center

🇺🇸

Meridian, Idaho, United States

Physicians Clinic of Iowa

🇺🇸

Cedar Rapids, Iowa, United States

Tomac, Inc.

🇺🇸

Columbiana, Alabama, United States

Innovative Clinical Trials

🇺🇸

Birmingham, Alabama, United States

Rheumatology Associates of North Alabama

🇺🇸

Huntsville, Alabama, United States

Arkansas Primary Care Clinic

🇺🇸

Little Rock, Arkansas, United States

Genova Clinical Research

🇺🇸

Tucson, Arizona, United States

Irvine Center for Clinical Research

🇺🇸

Irvine, California, United States

Rancho Cucamonga Clinical Trials

🇺🇸

Rancho Cucamonga, California, United States

Florida Medical Center

🇺🇸

Clearwater, Florida, United States

Nature Coast Clinical Research

🇺🇸

Crystal River, Florida, United States

George E. Platt, MD

🇺🇸

Green Cove Springs, Florida, United States

Hillcrest Medical Center

🇺🇸

Orange City, Florida, United States

Farmer MD, PA

🇺🇸

Ormond Beach, Florida, United States

Geodessey Research, LLC

🇺🇸

Vero Beach, Florida, United States

Global Research Partners & Consultants, Inc.

🇺🇸

Calhoun, Georgia, United States

The Center for Arthritis & Osteoporosis

🇺🇸

Elizabethtown, Kentucky, United States

Future Care Studies

🇺🇸

Springfield, Massachusetts, United States

Gulf Coast Research

🇺🇸

Baton Rouge, Louisiana, United States

The Center for Rheumatology & Bone Research

🇺🇸

Wheaton, Maryland, United States

Arthritis Associates

🇺🇸

Hattiesburg, Mississippi, United States

Clinical Pharmacology Study Group

🇺🇸

Worcester, Massachusetts, United States

Justus Fiechtner, MD, MPH

🇺🇸

Lansing, Michigan, United States

Medical Center Healthcare Research

🇺🇸

Florissant, Missouri, United States

Medex Healthcare

🇺🇸

Saint Louis, Missouri, United States

Arthritis Center of Reno

🇺🇸

Reno, Nevada, United States

Arthritis & Osteoporisis Associates

🇺🇸

Manalapan, New Jersey, United States

Rheumatology and Arthritis Associates

🇺🇸

Medford, New Jersey, United States

Arthritis Consultants of the Carolinas

🇺🇸

Belmont, North Carolina, United States

Concorde medical Group

🇺🇸

New York, New York, United States

Arthritis & Osteoporosis Consultants of the Carolinas

🇺🇸

Charlotte, North Carolina, United States

Southwest Medical Associates

🇺🇸

Brewster, New York, United States

NEA Clinic

🇺🇸

Jonesboro, Arkansas, United States

Coastal Medical Research, Inc.

🇺🇸

Port Orange, Florida, United States

Southeastern Integrated Medical

🇺🇸

Gainesville, Florida, United States

Southwest Florida Clinical Research Center

🇺🇸

Tampa, Florida, United States

David H. Neustadt PSCq

🇺🇸

Louisville, Kentucky, United States

Arthritis and Osteoporosis Center of Maryland

🇺🇸

Frederick, Maryland, United States

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