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Trial of EXenatide in Acute Ischaemic Stroke

Phase 2
Conditions
Acute Ischemic Stroke
Interventions
Registration Number
NCT03287076
Lead Sponsor
Neuroscience Trials Australia
Brief Summary

A multicentre, randomised controlled Trial of Exenatide versus standard care in Acute Ischemic Stroke

Detailed Description

Overview: Elevated blood glucose levels are common in many acute diseases, resulting in worse clinical outcomes. Hyperglycaemia in acute ischaemic stroke (post-stroke hyperglycaemia \[PSH\]) occurs in up to 50% patients, reduces the efficacy of stroke thrombolysis with increased risk of haemorrhage, increases infarct size, and results in worse clinical outcomes and death. Insulin-based therapies have not proved beneficial in treating PSH: they are difficult to implement and maintain, cause frequent hypoglycaemia, may cause increased infarct size, and do not reduce mortality or improve clinical outcomes. An alternative, simple to use, treatment for PSH may therefore have a significant impact not only for acute stroke care, but in other acute diseases.

Pilot data: Exenatide is a commonly used diabetes drug (a synthetic glucagon- like peptide-1 receptor agonist) that increases insulin secretion. Importantly, this action is glucose dependent - as blood glucose levels decrease, its stimulatory effect on insulin secretion subsides, with a very low risk of hypoglycaemia. A small randomised pilot study of 17 consecutive, unselected patients (ie. regardless of their admission glucose level) with acute ischaemic stroke compared subcutaneous exenatide 5μg for 5 days with routine standard of care. Overall, blood glucose levels remained consistently lower (and less variable) in the exenatide group, and most noticeably in those stroke patients with known diabetes. Exenatide was safe and well tolerated by all patients, with no symptomatic hypoglycaemia.

Trial design: TEXAIS is a 3 year Phase 2, multi centre, prospective, randomised, open label, blinded end-point (PROBE) trial comparing Exenatide to Standard of Care. The sample size is 528 patients (264 in each arm).

Intervention: Treatment arm will receive Exenatide (Byetta) 5μg subcutaneously twice daily for five days, commencing within 9 hours of symptom onset. Stroke onset time for wake-up strokes is taken as mid-point between going to bed, and waking up. Antiemetic therapy (metoclopramide or ondansetron) will be commenced with the first dose of Exenatide. In patients receiving tPA, Exenatide will be given alongside, or as soon as possible, following tPA administration (within 60 minutes). Diabetic patients already on oral agents and/or insulin may continue these (as per standard practice) in addition to Exenatide. Continuous glucose monitors (CGMs) will track the intra-day dynamic variability of glucose in acute stroke.

Translation: TEXAIS is a simple, practical, study that can enrol all patients with ischaemic stroke, regardless of admission blood glucose level, regardless of stroke severity, with no target glucose level, and with low risk of hypoglycaemia.

Recruitment & Eligibility

Status
UNKNOWN
Sex
All
Target Recruitment
350
Inclusion Criteria
  • Males and females 18 years or older
  • Acute Ischaemic Stroke - CT brain exclusion of haemorrhagic stroke
  • Blood glucose level on admission ≥ 4mmol/L
  • First trial treatment possible within 9 hours of stroke onset
  • Pre-morbid /mRS score of 0-2
Exclusion Criteria
  • Haemorrhagic stroke
  • Poor clinical prognosis /palliation (considered unlikely to survive beyond 14 days post stroke).
  • Any known allergy or hypersensitivity to Exenatide
  • Females who are pregnant (known or suspected) or currently breastfeeding
  • Any past history of pancreatitis or evidence of active pancreatitis
  • History of active severe gastrointestinal disease (including but not limited to gastroparesis and dumping syndrome)
  • Current chronic kidney disease stage 4 or 5 (creatinine clearance <30ml/min)
  • Current participation in another interventional clinical trial
  • Inability to provide consent (participant or person responsible as local laws apply)
  • Current use of Exenatide (Byetta®), or other GLP-1 agonist diabetes medication
  • Patients considered unlikely to be able to be followed up at 3 months (including but not limited to geographical location of patient at 3 months)

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
ActiveExenatide InjectionPatients will receive exenatide injections
Primary Outcome Measures
NameTimeMethod
improved neurological outcome7 days

Treatment with short acting Exenatide (Byetta) in patients with acute ischaemic stroke is hypothesised to improve neurological outcome as measured by ≥8 point improvement in the National Institutes of Health Stroke Scale (NIHSS) stroke disability score (or NIHSS 0-1) at 7 days

Secondary Outcome Measures
NameTimeMethod
NIHSS90 days

improve NIHSS at 90 days

post stroke hyperglycaemia90 days

reduce the occurrence of post stroke hyperglycaemia (\>7mmol/l).

Modified Rankin Scale90 days

improve Modified Rankin Scale (mRS) at 90 days

Trial Locations

Locations (15)

Austin Hospital

🇦🇺

Heidelberg, Victoria, Australia

Royal Melbourne Hospital

🇦🇺

Parkville, Victoria, Australia

Helsinki University Hospital

🇫🇮

Helsinki, Finland

St Vincent's Hospital Sydney

🇦🇺

Darlinghurst, New South Wales, Australia

CDHB Christchurch Hospital

🇳🇿

Christchurch, New Zealand

Princess Alexandra Hospital

🇦🇺

Woolloongabba, Queensland, Australia

Alfred Hospital

🇦🇺

Melbourne, Victoria, Australia

Liverpool Hospital

🇦🇺

Liverpool, New South Wales, Australia

Sunshine Coast University Hospital

🇦🇺

Birtinya, Queensland, Australia

Launceston General Hospital

🇦🇺

Launceston, Tasmania, Australia

Royal Brisbane and Women's Hospital

🇦🇺

Herston, Queensland, Australia

St John of God Midland Public & Private Hospital

🇦🇺

Midland, Western Australia, Australia

Fiona Stanley Hospital

🇦🇺

Murdoch, Western Australia, Australia

Box Hill Hospital

🇦🇺

Box Hill, Victoria, Australia

St Vincent's Hospital Melbourne

🇦🇺

Fitzroy, Victoria, Australia

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