MedPath

Trial of Deforolimus in Combination With Bevacizumab for Patients With Advanced Cancers (8669-010)(COMPLETED)

Phase 1
Completed
Conditions
Solid Tumor
Interventions
Registration Number
NCT00781846
Lead Sponsor
Merck Sharp & Dohme LLC
Brief Summary

The purpose of this study is to assess the safety, tolerability, and recommended phase 2 dose of oral ridaforolimus administered in combination with intravenous bevacizumab in patients with advanced cancers.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
17
Inclusion Criteria
  • 18 years of age or older
  • Advanced or metastatic solid tumor malignancy
  • ECOG performance status of less than or equal to 1
  • Life expectancy of greater than 3 months
  • At least 4 weeks must have elapsed between prior investigational therapy, chemotherapy, or radiotherapy, and the first dose of deforolimus
  • Adequate hematological, hepatic and renal function
  • Serum cholesterol less than or equal to 350 mg/dL and triglycerides less than or equal to 400 mg/dL
  • Signed informed consent
  • Women of childbearing potential must have a negative serum pregnancy test within 7 days of starting therapy and must use an approved contraceptive method from time of screening until 30 days after the last dose of study drug
Exclusion Criteria
  • Tumor location in close proximity to a major blood vessel
  • History of brain metastases, spinal cord compression, or carcinomatous meningitis. Primary brain tumors (for example, glioblastoma) are allowed.
  • New brain metastases, spinal cord compression, or leptomeningeal metastases on screening CT scan or MRI
  • Hemoptysis or hematemesis within 28 days prior to entering the trial
  • Clinical significant unexplained bleeding within 28 days prior to entering the trial
  • Uncontrolled hypertension
  • Proteinuria at screening
  • Clinically significant cardiovascular disease
  • Newly diagnosed or poorly controlled type 1 or 2 diabetes
  • Active infection requiring prescribed intervention
  • Other concurrent illness that, in the Investigator's judgement, would either compromise the patient's safety or interfere with the evaluation of the safety of the study drug
  • Major surgery within 28 days before trial entry, or any incompletely healed surgical incision; minor surgery or procedures within 7 days
  • Pregnant or breastfeeding
  • Known allergy to macrolide antibiotics
  • Known hypersensitivity to any component of bevacizumab
  • Concurrent treatment with medications that strongly induce or inhibit cytochrome P450 (CYP3A)
  • Known history of HIV sero-positivity
  • Any condition in the Investigator's judgement that renders the patient unable to fully understand and provide informed consent and/or comply with the protocol

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
1ridaforolimus30mg QDx5/wk ridaforolimus plus 10mg/kg Q2wks bevacizumab for 4 weeks
1bevacizumab30mg QDx5/wk ridaforolimus plus 10mg/kg Q2wks bevacizumab for 4 weeks
2bevacizumab40mg QDx5/wk ridaforolimus plus 10mg/kg Q2wks bevacizumab for 4 weeks
2ridaforolimus40mg QDx5/wk ridaforolimus plus 10mg/kg Q2wks bevacizumab for 4 weeks
3bevacizumab40mg QDx5/wk ridaforolimus plus 15mg/kg Q3wks bevacizumab for 3 weeks
3ridaforolimus40mg QDx5/wk ridaforolimus plus 15mg/kg Q3wks bevacizumab for 3 weeks
Primary Outcome Measures
NameTimeMethod
Identification of recommended phase 2 dose of ridaforolimus in combination with bevacizumabDuration of the trial
Secondary Outcome Measures
NameTimeMethod
Characterize the overall safety and tolerability of ridaforolimus in combination with bevacizumabDuration of the study
Description of the anti-tumor activity of ridaforolimus in combination with bevacizumabDuration of the study
© Copyright 2025. All Rights Reserved by MedPath