MedPath

Safety and Efficacy of Nalmefene in Patients With Alcohol Dependence

Phase 3
Completed
Conditions
Alcohol Dependence
Interventions
Drug: Placebo
Registration Number
NCT00811941
Lead Sponsor
H. Lundbeck A/S
Brief Summary

The purpose of the study is long-term safety, tolerability and efficacy of nalmefene in patients with alcohol dependence.

Detailed Description

Alcohol dependence is a maladaptive pattern of alcohol use, leading to clinically significant impairment or distress, as manifested by at least three of a number of criteria such as tolerance, withdrawal symptoms, frequent use of alcohol in larger amounts or over longer periods than was intended, and others. Excessive intake of alcohol reduces the life span by a decade, and alcohol drinking is strongly related to mortality from liver cirrhosis, chronic pancreatitis, certain cancers, hypertension, accidents and violence. This study is planned to evaluate the long-term safety and tolerability as well as to evaluate the efficacy of as needed use of 18.06 mg nalmefene in patients with alcohol dependence.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
665
Inclusion Criteria

In- and outpatients who:

  • had a primary diagnosis of alcohol dependence according to Diagnostic and Statistical Manual of Mental Disorders - text revision (DSM-IV-TR) criteria
  • had had ≥6 Heavy Drinking Days (HDDs) in the 4 weeks preceding the Screening Visit
Exclusion Criteria

The patient:

  • had a severe psychiatric disorder or an antisocial personality disorder
  • had risk of suicide evaluated by the suicidality module of the Mini-International Neuropsychiatric Interview (MINI)
  • had a history of delirium tremens or alcohol withdrawal seizures
  • reported current or recent (within 3 months preceding screening) treatment with disulfiram, acamprosate, topiramate, naltrexone or carbimide, or with any opioid antagonists
  • was pregnant or breast-feeding

Other protocol-defined inclusion and exclusion criteria may apply.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlacebo-
NalmefeneNalmefene-
Primary Outcome Measures
NameTimeMethod
Number of Patients With Adverse Events (AEs)Serious Adverse Events: 52 weeks and a safety follow-up (visit/telephone call) scheduled for 4 weeks after completion of the study or after withdrawal from the study. Other Adverse Events: 52 weeks.

Overview of AEs

Percentage of Patients Who Withdrew Due to Intolerance to TreatmentBaseline to Week 52
Change From Baseline in the Monthly Number of Heavy Drinking Days (HDDs)Baseline and Month 6

Number of HDDs over a month (28 days), where one HDD was defined as a day with alcohol consumption ≥60 grams (g) for men and ≥40 g for women.

Change From Baseline in the Monthly Total Alcohol Consumption (TAC)Baseline and Month 6

TAC was defined as mean daily alcohol consumption in g/day over a month (28 days).

Secondary Outcome Measures
NameTimeMethod
Drinking Risk Level (RSDRL) ResponseMonth 13

RSDRL response was defined as a downward shift from baseline in Drinking Risk Level (DRL); for patients at very high risk at Baseline: a shift to medium risk or below, and for patients at high or medium risk at Baseline: a shift to low risk or below.

Change From Baseline in Clinical Status Using CGI-SBaseline and Week 52

The Clinical Global Impression - Severity of Illness (CGI-S) provides the clinician's impression of the patient's current state of mental illness. The clinician uses his or her clinical experience of this patient population to rate the severity of the patient's current mental illness on a 7-point scale ranging from 1 (Normal - not at all ill) to 7 (among the most extremely ill patients).

Change in Clinical Status Using the CGI-IWeek 52

The Clinical Global Impression - Global Improvement (CGI-I) provides the clinician's impression of the patient's improvement (or worsening). The clinician assesses the patient's condition relative to a baseline on a 7- point scale ranging from 1 (very much improved) to 7 (very much worse).

Liver Function Test Gamma-glutamyl Transferase (GGT)Week 52

GGT values

Liver Function Test Alanine Aminotransferase (ALAT)Week 52

ALAT values

Change From Baseline in the Monthly Number of Heavy Drinking Days (HDDs)Baseline and Month 13

Number of HDDs over a month (28 days), where one HDD was defined as a day with alcohol consumption ≥60 g for men and ≥40 g for women.

Change From Baseline in the Monthly Total Alcohol Consumption (TAC)Baseline and Month 13

TAC was defined as mean daily alcohol consumption in g/day over a month (28 days).

Trial Locations

Locations (60)

UA010

🇺🇦

Ternopil, Ukraine

CZ001

🇨🇿

Usti nad Labem, Czech Republic

PL011

🇵🇱

Krakow, Poland

RU006

🇷🇺

St. Petersburg, Russian Federation

SK004

🇸🇰

Nitra, Slovakia

UA009

🇺🇦

Kherson, Ukraine

RU013

🇷🇺

Rostov on Don, Russian Federation

UA007

🇺🇦

Kharkiv, Ukraine

PL015

🇵🇱

Belchatow, Poland

PL010

🇵🇱

Lodz, Poland

PL012

🇵🇱

Swicie n/Wisla, Poland

UA003

🇺🇦

Donetsk, Ukraine

LV004

🇱🇻

Sigulda, Latvia

PL008

🇵🇱

Bydgoszcz, Poland

PL002

🇵🇱

Leszno, Poland

PL003

🇵🇱

Skorzewo, Poland

UA006

🇺🇦

Simferopol, Ukraine

LT003

🇱🇹

Kaunas, Lithuania

PL006

🇵🇱

Gdansk, Poland

PL014

🇵🇱

Lodz, Poland

PL007

🇵🇱

Starogard Gdanski, Poland

RU002

🇷🇺

Leningrad, Russian Federation

RU005

🇷🇺

St. Petersburg, Russian Federation

SK001

🇸🇰

Banska Bysterica, Slovakia

UA004

🇺🇦

Glevakha, Ukraine

CZ007

🇨🇿

Litomerice, Czech Republic

CZ004

🇨🇿

Praha 6, Czech Republic

EE002

🇪🇪

Parnu, Estonia

EE004

🇪🇪

Tallinn, Estonia

EE001

🇪🇪

Voru, Estonia

LV002

🇱🇻

Jelgava, Latvia

LV001

🇱🇻

Riga, Latvia

LT002

🇱🇹

Kaunas, Lithuania

PL009

🇵🇱

Szczecin, Poland

PL001

🇵🇱

Torun, Poland

HU002

🇭🇺

Budapest, Hungary

CZ006

🇨🇿

Lnare, Czech Republic

CZ005

🇨🇿

Prague, Czech Republic

EE005

🇪🇪

Tallinn, Estonia

EE003

🇪🇪

Vorumaa, Estonia

HU004

🇭🇺

Budapest, Hungary

PL004

🇵🇱

Lublin, Poland

PL005

🇵🇱

Lublin, Poland

PL013

🇵🇱

Piekary Slaskie, Poland

RU001

🇷🇺

St. Petersburg, Russian Federation

RU004

🇷🇺

Voronezh, Russian Federation

RU012

🇷🇺

St. Petersburg, Russian Federation

RU003

🇷🇺

St. Petersburg, Russian Federation

SK002

🇸🇰

Krupina, Slovakia

SK005

🇸🇰

Rimavska Sobota, Slovakia

UA001

🇺🇦

Chernihiv, Ukraine

UA008

🇺🇦

Dnipropetrovsk, Ukraine

GB007

🇬🇧

Birmingham, United Kingdom

GB006

🇬🇧

Glasgow, United Kingdom

GB009

🇬🇧

London, United Kingdom

UA002

🇺🇦

Kyiv, Ukraine

UA005

🇺🇦

Odessa, Ukraine

GB008

🇬🇧

Manchester, United Kingdom

LV003

🇱🇻

Daugavpils, Latvia

GB005

🇬🇧

Reading, United Kingdom

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