MedPath

Overnight Switch From Rasagiline To Safinamide

Phase 4
Completed
Conditions
Parkinson Disease
Interventions
Registration Number
NCT03843944
Lead Sponsor
IRCCS San Raffaele Roma
Brief Summary

Rasagiline label report the indication to wait at least 14 days between discontinuation of rasagiline and initiation of another MAO inhibitor. This results in a major inconvenience for Parkinsonian patients (PD) due to their clinical worsening. Safinamide is a reversible MAO-B inhibitor, characterized by a good safety profile. In clinical practice safinamide is often introduced instead of rasagiline following an overnight switch. The aim of this study is to explore the safety and tolerability of the immediate switch from rasagiline (irreversible MAO-B inhibitor) to safinamide, with the expectation that there will be no adverse events or increased risk of hypertensive crisis for patients with PD or signs of serotonin syndrome

Detailed Description

Objective: The aim of this study is to verify safety and tolerability of the immediate switch from rasagiline to safinamide trough monitoring of BP by 24-hour Holter recording. The primary objective of the study will be achieved if the mean BP will not increase by \>10 mmHg in the studied population.

Methods: This is an open-label, single-centre study conducted at IRCCS San Raffaele Pisana. Study population included patients with idiopathic PD in the mid-late stage of the disease, suffering from motor fluctuation, on stable treatment with rasagiline and Levodopa (alone or in combination with other anti-parkinsonian medication). The protocol contemplates five visits during six weeks, with two 24-hour Holter recording (first in rasagiline and second in first-day of safinamide therapy), monitoring typical symptoms of the serotonin syndrome.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
20
Inclusion Criteria
  • Patients able to comprehend and provide consent form
  • Patients with idiopathic Parkinson's disease diagnosed according to the UK Brain Bank criteria
  • Patients in mid-to late stage of the disease (Hoehn & Yahr: between the stage 2 and 4 in on state).
  • Patients suffering from motor fluctuations
  • Patients must have a good response to levodopa in the opinion of the investigators (evaluated as improvement ≥ 30% of the UPDRS scores)
  • Stable dosage of antiparkinsonian medication for at least 4 weeks prior to study enrollment
  • Female patients in post-menopausal state; women of childbearing potential must use an acceptable method of contraception
Exclusion Criteria
  • Atypical Parkinsonism
  • Any significant psychiatric, metabolic and systemic concomitant disease
  • Patients with clinically significant out of range laboratory values
  • Patients participating in a clinical trial in the last 6 weeks
  • Patients with moderate-severe cognitive decline not able to provide consent form
  • Patients currently lactating or pregnant or planning to become pregnant during the duration of the study
  • Patients for whom Xadago is contraindicated according to the current SmPC

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
SafinamideSafinamideOvernight switch from rasagiline 1 mg OD to safinamide 50 mg OD
Primary Outcome Measures
NameTimeMethod
Change From Baseline in Blood Pressure (BP)through study completion, an average of 8 weeks

Monitoring of BP by 24-hour Holter (increase by \>10 mmHg)

Secondary Outcome Measures
NameTimeMethod
Clinical change in UPDRS compared to baselinethrough study completion, an average of 8 weeks

Unified Parkinson's Disease rating scale (UPDRS total score ranges between 0 - normal - to 199 points - severe)

Clinical change in H&Y compared to baselinethrough study completion, an average of 8 weeks

Hoehn and Yahr scale is a system for describing progress of Parkinson's disease (range between 1 -less affect- to 5-more affect)

Clinical change in MoCA compared to baselinethrough study completion, an average of 8 weeks

The Montreal Cognitive Assessment (MoCA) is a widely used screening assessment for detecting cognitive impairment (ranges between 0-more affect- and 30-normal)

Trial Locations

Locations (1)

IRCCS San Raffaele

🇮🇹

Roma, Italy

IRCCS San Raffaele
🇮🇹Roma, Italy

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