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PCI Treatment/Gemcitabine & Chemotherapy vs Chemotherapy Alone in Patients With Inoperable Extrahepatic Bile Duct Cancer

Phase 2
Terminated
Conditions
Cholangiocarcinoma
Interventions
Drug: Gemcitabine/Cisplatin chemotherapy
Registration Number
NCT04099888
Lead Sponsor
PCI Biotech AS
Brief Summary

This study will assess the safety and effectiveness of fimaporfin-induced photochemical internalisation (PCI) of gemcitabine complemented by systemic gemcitabine/cisplatin chemotherapy compared to gemcitabine/cisplatin alone, in patients with inoperable cholangiocarcinoma (CCA). Participants will be randomly assigned to one of the treatment groups and will receive study treatment for 6 months, followed by assessments every 3 months, as applicable.

Detailed Description

Cholangiocarcinoma (CCA) is an uncommon adenocarcinoma arising from cells lining the bile ducts. Standard treatment options for CCA include surgery, radiotherapy and chemotherapy, dependent upon if the CCA is intra- or extra-hepatic. Surgical removal of the tumor is the only potential cure, and CCA is very resistant to standard pharmaceutical drug treatment, though chemotherapy has some effect. Current chemotherapy uses cisplatin plus gemcitabine. Photochemical internalisation (PCI) is a novel technology, where photochemical reactions are used to enhance the effect of drugs by increasing their ability cross cell membranes to interact with their intended target. This study will assess the safety and effectiveness of fimaporfin-induced PCI of gemcitabine complemented by systemic gemcitabine/cisplatin chemotherapy compared to gemcitabine/cisplatin alone, in patients with inoperable CCA.

NOTE: Participants are no longer being recruited to this study.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
41
Inclusion Criteria
  1. Each patient must provide signed and witnessed written informed consent and agree to comply with study protocol requirements.
  2. Histopathologically/cytologically verified adenocarcinoma consistent with cholangiocarcinoma (CCA). Must have biliary lesion causing bile obstruction that requires stenting and is accessible for PCI light treatment (ie, extrahepatic CCA [perihilar or distal] only).
  3. CCA must be considered inoperable with respect to radical resection.
  4. At least 1 radiologically evaluable lesion (measurable and/or non-measurable) that can be assessed at baseline and is suitable for repeated radiological evaluation.
  5. If metastatic, metastases must be limited tissues other than bone or the central nervous system.
  6. Must have adequate biliary drainage (at least 50% of the liver volume or at least 2 sectors) with no evidence of active uncontrolled infection (patients on antibiotics are eligible).
  7. Must have Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.
  8. Estimated life expectancy of at least 12 weeks.
Exclusion Criteria
  1. Patients who have previously received any anti-tumor (either local or systemic) treatment for CCA, except for previous treatment of up to 2 cycles of gemcitabine/cisplatin.
  2. Patients with severe visceral disease other than CCA.
  3. A history of frequently recurring septic biliary events.
  4. Patients with porphyria or hypersensitivity to porphyrins.
  5. Patients with a second primary cancer with a disease-free interval of <5 years. A second primary cancer that has been treated with intent to cure may be allowed after consultation with the study Medical Monitor. Adequately treated basal cell carcinoma, squamous cell carcinoma or other non-melanomatous skin cancer, in-situ carcinoma of the uterine cervix, or prostate cancer that is controlled by hormone therapy (patients may continue hormone therapy while on study) are allowed.
  6. Patients not able to undergo contrast-enhanced CT or MRI.
  7. Patients currently participating in any other interventional clinical trial.
  8. Planned surgery, endoscopic examination or dental treatment in the first 30 days after PCI treatment.
  9. Co-existing ophthalmic disease likely to require slit-lamp examination within the first 90 days after PCI treatment.
  10. Clinically significant and uncontrolled cardiac disease except for extra systoles or minor conduction abnormalities and controlled and well-treated chronic atrial fibrillation.
  11. Known allergy or sensitivity to photosensitisers (active substance and/or any of the excipients); or chronic use of other photosensitising therapies; treatment with amiodarone during the last 12 months.
  12. Known hypersensitivity to or contraindication to the use of gemcitabine (active substance and/or any of the excipients).
  13. Known hypersensitivity to or contraindication to the use of cisplatin (active substance and/or any of the excipients).
  14. Patients with ataxia telangiectasia.
  15. Upon the Investigator's discretion, evidence of any other medical conditions (such as psychiatric illness, physical examination or laboratory findings) that may interfere with the planned PCI treatment, affect patient compliance or place the patient at high risk from treatment-related complications.
  16. Patients planning to have or who have recently had vaccination with a live vaccine.
  17. Patients concurrently receiving treatment with phenytoin.
  18. Male patients unwilling to use highly effective contraception or female patients of childbearing potential unwilling to use highly effective form of contraception. Patients must continue the use of contraception during PCI treatment and subsequent chemotherapy for at least 6 months thereafter.
  19. Women who are breastfeeding or who have a positive pregnancy test at baseline.
  20. Patients with inadequate bone marrow function (absolute neutrophil count <1.5 x 10^9/L; platelet count <100 x 10^9/L; haemoglobin <6 mmol/L [transfusion allowed]).
  21. Inadequate liver function despite satisfactory drainage (serum bilirubin persisting at >5 x upper limit of normal for the institution; aspartate aminotransferase or alanine aminotransferase >3.0 x upper limit of normal or >5 x upper limit of normal if liver metastases are present; alkaline phosphatase levels >5.0 x upper limit of normal).
  22. Inadequate renal function, as determined by local practice for patients on fractionated platinum-based chemotherapy. Patients with creatinine clearance <45 mL/min (in France: <60 mL/min) must not be included.

Other protocol-defined criteria may apply.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PCI treatment in conjunction with Standard of Care (SoC)Fimaporfin and GemcitabineArm A: Fimaporfin-induced photochemical internalisation (PCI) of gemcitabine complemented by gemcitabine/cisplatin chemotherapy
PCI treatment in conjunction with Standard of Care (SoC)Gemcitabine/Cisplatin chemotherapyArm A: Fimaporfin-induced photochemical internalisation (PCI) of gemcitabine complemented by gemcitabine/cisplatin chemotherapy
Standard of Care (SoC)Gemcitabine/Cisplatin chemotherapyArm B: Gemcitabine/cisplatin chemotherapy
Primary Outcome Measures
NameTimeMethod
Progression-free Survival (PFS)Up to 18 months

From date of randomisation to date of objective disease progression or death, whichever comes first (in months)

Secondary Outcome Measures
NameTimeMethod
Overall Survival (OS)Up to 24 months

From date of randomisation to date of death from any cause (in months)

Change in Tumor SizeUp to 18 months

Best overall percentage change in tumour size from baseline

Best Overall Response (BOR)Up to 18 months

Best response recorded from start of treatment until disease progression/recurrence (according to RECIST 1.1)

Objective Response Rate (ORR)Up to 18 months

Proportion of patients with measurable disease at baseline who have at least one visit response with a complete response (CR) or partial response (PR) noted (according to RECIST 1.1)

Duration of Response (DoR)Up to 24 months

From first documented tumour response until first documented disease progression, or death in the absence of disease progression (in months)

Adverse Events (AEs)/Serious Adverse Events (SAEs)Up to 12 months

Number and proportion of patients with AEs/SAEs

Time to Cmax (Tmax) Was Performed for Patients in Arm A.Timepoints for PK sampling: Day -4 (before, 30 min and 4 hours after Amphinex), C1-D1, C1-D8, C2-D8, C3-D8, C4-D8, C4-D18 (before, 30 min and 4 hours after Amphinex) , C5-D1, and C5-D8

A non-compartmental analysis (NCA) was applied on the data as described by Gabrielsson \& Weiner (Methods in molecular biology, 929:161-180, 2012).

Health-related Quality of Life (QoL)Up to 18 months

QoL assessment. Patients select one of four answers to 22 questions ranging from 1 (not at all) to 4 (very much). Lower total scores indicate a more favorable QoL perception than a higher score.

Overall Disease Control Rate (DCR)6 months and 12 months

Proportion of patients with BOR of CR, PR or stable disease (SD) (according to RECIST 1.1) at or after the first follow-up scan, partial response or complete response

Loco-regional Tumour-related Events and Biliary ComplicationsUp to 12 months

Frequency and severity of loco-regional tumour related events and biliary complications

Area Under the Plasma Concentration Curve (AUC) Was Performed for Patients in Arm A.Time Frame AUC calculated from time zero to C5-D8 (3 months from the first PCI treatment)

A non-compartmental analysis (NCA) was applied on the data. AUC from time zero to the last measured concentration (AUC 0-t) was initially estimated by the linear trapezoidal method.

Maximum Observed Concentration (Cmax) Was Performed for Patients in Arm A.Timepoints for pharmacokinetic (PK) sampling: Day -4 (before, 30m and 4hrs after Amphinex), C1-D1, C1-D8, C2-D8, C3-D8, C4-D8, C4-D18 (before, 30m and 4hrs after Amphinex), C5-D1, and C5-D8

A non-compartmental analysis (NCA) was applied on the data.

Trial Locations

Locations (50)

Baylor College of Medicine

🇺🇸

Houston, Texas, United States

Odense Universitetshospital

🇩🇰

Odense, Denmark

The Mayo Clinic Hospital - Saint Mary's Campus, 1216 Second Street Southwest

🇺🇸

Rochester, Minnesota, United States

Pusan National University Hospital, 179 Gudeok-ro, Seo-gu

🇰🇷

Busan, Korea, Republic of

City of Hope National Medical Center

🇺🇸

Duarte, California, United States

University of Louisville

🇺🇸

Louisville, Kentucky, United States

Emory University Hospital, 1365C Clifton Road NE

🇺🇸

Atlanta, Georgia, United States

University of Chicago Medical Center, 5841 South Maryland Avenue

🇺🇸

Chicago, Illinois, United States

UZ Gent

🇧🇪

Gent, Oost-Vlaanderen, Belgium

Centre Hospitalier Universitaire Grenoble Alpes - Hopital Albert Michallon

🇫🇷

Grenoble, Cedex 09, France

UZ Leuven

🇧🇪

Leuven, Belgium

Tampereen yliopistollinen sairaala, Syöpätautien klinikka

🇫🇮

Tampere, Finland

CHU Angers

🇫🇷

Angers, Cedex 9, France

Klinikum rechts der Isar der Technischen Universität München

🇩🇪

MĂĽnchen, Bayern, Germany

Institut Gustave Roussy, Département de gastro-entérologie

🇫🇷

Villejuif, France

CHU Dupuytren, 2 Avenue Martin Luther King

🇫🇷

Limoges, France

Universitätsklinikum Frankfurt

🇩🇪

Frankfurt am main, Hessen, Germany

Universitätsklinikum Essen

🇩🇪

Essen, Nordrhein-Westfalen, Germany

Universitätsklinikum Bonn

🇩🇪

Bonn, Germany

Klinikum Landshut

🇩🇪

Landshut, Germany

Universität Leipzig KöR

🇩🇪

Leipzig, Germany

LAKUMED Kliniken

🇩🇪

Landshut, Germany

Klinikum Mannheim Universitätsklinikum gGmbH

🇩🇪

Mannheim, Germany

Klinikum der Ludwig-Maximilians-Universität MünchenKlinik

🇩🇪

Muenchen, Germany

Azienda Ospedaliero Universitaria Di Modena Policlinico

🇮🇹

Modena, Emilia-Romagna, Italy

National Cancer Center, 323 Ilsan-ro, Ilsandong-gu

🇰🇷

Goyang-si, Gyeonggido, Korea, Republic of

Klinikum NĂĽrnberg Nord, Medizinische Klinik 6 - (Schwerpunkte Gastroenterologie, Hepatologie, Endokrinologie)

🇩🇪

NĂĽrnberg, Germany

IRCCS Saverio de Bellis, Via Turi, 27

🇮🇹

Castellana Grotte, Italy

Zaklad Opieki Zdrowotnej MSW z Warminsko-Mazurskim Centrum Onkologii

🇵🇱

Olsztyn, Warminsko-mazurskie, Poland

Asan Medical Center, 88 Olympic-ro 43-gil, Songpa-gu

🇰🇷

Seoul, Korea, Republic of

Kyungpook National University Chilgok Hospital, 807 Hoguk-ro, Buk-gu

🇰🇷

Daegu, Korea, Republic of

Clinica Universidad Navarra

🇪🇸

Pamplona, Navarra, Spain

Severance Hospital Yonsei University Health System, 50-1, Yonsei-Ro, Seodaemun-Gu

🇰🇷

Soeul, Korea, Republic of

Hospital Universitario 12 de Octubre

🇪🇸

Madrid, Spain

Hospital del Mar

🇪🇸

Barcelona, Spain

Med-Polonia Sp. z o.o.

🇵🇱

Poznań, Poland

The Catholic University of Korea, Seoul St. Mary's Hospital, 222 Banpo-Daero Seocho-gu

🇰🇷

Soeul, Korea, Republic of

Hospital Universitario HM Sanchinarro - CIOCC

🇪🇸

Madrid, Spain

Hospital Universitario Puerta de Hierro - Majadahonda

🇪🇸

Majadahonda, Spain

Taichung Veterans General Hospital, No. 1650 Taiwan Boulevard, Sec. 4

🇨🇳

Taichung, Taiwan

Corporacio Sanitaria Parc Tauli

🇪🇸

Sabadell, Spain

Karolinska Universitetssjukhuset Solna, P.O Bäckencancer, Karolinska Universitetssjukhuset

🇸🇪

Stockholm, Stockholms Ian, Sweden

Taipei Veterans General Hospital, No. 201, Sction 2, Shi-pai Road

🇨🇳

Taipei, Taiwan

Chang Gung Memorial Hospital, Linkou, Dept. of Medical Oncology, 5 Fuxing Street, Guishan

🇨🇳

Taoyuan, Taiwan

SI "National Institute of Surgery and Transplantology n.a. O.O. Shalimov " of NAMS of Ukraine

🇺🇦

Kyiv, Ukraine

MNPE of Kharkiv Regional Council Regional Clinical Specialized Dispensary of Radiation Protection

🇺🇦

Kharkiv, Ukraine

SI Institute for General and Urgent Surgery n.a. V.T. Zaitseva of NAMS of Uktraine

🇺🇦

Kharkiv, Ukraine

Universitätsklinikum Hamburg Eppendorf, I. Medizinische Klinik und Poliklinik (Gastroenterologie mit Sektionen Infektiologie und Tropenmediz)

🇩🇪

Hamburg, Germany

Municipal Nonprofit Enterprise City Hospital #3 of Zaporizhzhia City Council

🇺🇦

Zaporizhzhya, Ukraine

Oslo Universitetssykehus HF Radiumhospitalet

🇳🇴

Oslo, Norway

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