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A Study to Test a Medicine (Fitusiran) Injected Under the Skin for Preventing Bleeding Episodes in Male Adolescent or Adult Participants With Severe Hemophilia

Phase 3
Active, not recruiting
Conditions
Hemophilia
Interventions
Drug: Clotting factor concentrates (CFC) or bypassing agents (BPA)
Drug: Antithrombin concentrate (ATIIIC)
Registration Number
NCT05662319
Lead Sponsor
Sanofi
Brief Summary

This is a multicenter, multinational, open-label, one-way cross-over, Phase 3, single-arm study for treatment of hemophilia.

The purpose of this study is to measure the frequency of treated bleeding episodes with fitusiran in male adult and adolescent (≥12 years old) participants with hemophilia A or B, with or without inhibitory antibodies to factor VIII or IX who have switched from their prior standard of care treatment.

The total study duration will be up to approximately 50 months (200 weeks, 1 study month is equivalent to 4 weeks) and will include:

* A screening period up to approximately 60 days,

* A standard of care (SOC) period of approximately 6 study months (24 weeks),

* A fitusiran treatment period of approximately 36 study months (144 weeks),

* An antithrombin (AT) follow-up period of approximately 6 study months (24 weeks) but may be shorter or longer depending on individual participants AT recovery.

The frequency for telephone visits will be approximately every 2 weeks. For site visits the frequency will be approximately every 8 weeks during the SOC period and approximately every 4 weeks during the fitusiran treatment period. If applicable and if allowed by local regulation, home and/or remote visits may be conducted during the study

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
Male
Target Recruitment
79
Inclusion Criteria
  • Diagnosis of severe congenital hemophilia A or B (FVIII <1% or FIX level ≤2%) as evidenced by a central laboratory measurement at screening or documented medical record evidence.
  • For participants currently not on prophylaxis (CFC or BPA on-demand): A minimum of 4 bleeding episodes requiring BPA (inhibitor participants) or CFC (non-inhibitor participants) treatment within the last 6 months prior to screening.
  • Willing and able to comply with the study requirements and to provide written informed consent and assent in the case of participants under the age of legal consent, per local and national requirements
Exclusion Criteria
  • Known co-existing bleeding disorders other than congenital hemophilia A or B
  • History of arterial or venous thromboembolism, not associated with an indwelling venous access
  • History of intolerance to SC injection(s).
  • Current participation in immune tolerance induction therapy (ITI)
  • Prior gene therapy
  • Current or prior participation in a fitusiran trial
  • Current or prior participation in a gene therapy trial
  • Received an investigational drug or device within 30 days prior to the screening visit or within 5 half-lives of the investigational drug (or device) prior to the screening visit, whichever is longer
  • Presence of clinically significant liver disease AT activity <60% at Screening
  • Co-existing thrombophilic disorder
  • Hepatitis C virus antibody positive, except participants who have negative Hepatitis C viral load and no evidence of cirrhosis
  • Presence of acute hepatitis, ie, hepatitis A, hepatitis E.
  • Presence of acute or chronic hepatitis B infection
  • Known to be HIV positive with CD4 count <200 cells/μL.
  • Reduced renal function The above information is not intended to contain all considerations relevant to a patient's potential participation in a clinical trial.

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
All participantsAntithrombin concentrate (ATIIIC)In standard of care (SOC) period, participants will receive on-demand or prophylactic treatment with clotting factor concentrates (CFCs) or bypassing agents (BPAs) for 6 months (from Day -168 to Day -1). In fitusiran treatment period, participants will receive subcutaneous fitusiran prophylaxis once every other month (Q2M) or once monthly (QM) for 36 months (from Day 1 to Day 1009). In case of bleeding events participants will receive IV CFCs or BPAs. Participants may receive Antithrombin concentrate (ATIIIC) as rescue medicine. .
All participantsClotting factor concentrates (CFC) or bypassing agents (BPA)In standard of care (SOC) period, participants will receive on-demand or prophylactic treatment with clotting factor concentrates (CFCs) or bypassing agents (BPAs) for 6 months (from Day -168 to Day -1). In fitusiran treatment period, participants will receive subcutaneous fitusiran prophylaxis once every other month (Q2M) or once monthly (QM) for 36 months (from Day 1 to Day 1009). In case of bleeding events participants will receive IV CFCs or BPAs. Participants may receive Antithrombin concentrate (ATIIIC) as rescue medicine. .
All participantsFitusiranIn standard of care (SOC) period, participants will receive on-demand or prophylactic treatment with clotting factor concentrates (CFCs) or bypassing agents (BPAs) for 6 months (from Day -168 to Day -1). In fitusiran treatment period, participants will receive subcutaneous fitusiran prophylaxis once every other month (Q2M) or once monthly (QM) for 36 months (from Day 1 to Day 1009). In case of bleeding events participants will receive IV CFCs or BPAs. Participants may receive Antithrombin concentrate (ATIIIC) as rescue medicine. .
Primary Outcome Measures
NameTimeMethod
Annualized bleeding rate (ABR) in the fitusiran primary efficacy periodDay 169 to Day 505 (since the first dose of fitusiran)

A bleeding episode is defined as any occurrence of hemorrhage that requires administration of CFCs or BPAs, e.g., hemarthrosis, muscle, or mucosal bleeding.

Secondary Outcome Measures
NameTimeMethod
Annualized bleeding rate (ABR) while on fitusiran prophylaxis in the fitusiran primary efficacy period and ABR while on prophylaxis standard of care (SOC) in the SOC periodDay 169 to Day 505 (primary efficacy period) and Day -168 to Day -1 (SOC period)

A bleeding episode is defined as any occurrence of hemorrhage that requires administration of CFCs or BPAs, e.g., hemarthrosis, muscle, or mucosal bleeding.

Annualized spontaneous bleeding rate in the fitusiran primary efficacy period and in the SOC periodDay 169 to Day 505 (primary efficacy period) and Day -168 to Day -1 (SOC period)

A bleeding episode is defined as any occurrence of hemorrhage that requires administration of CFCs or BPAs, e.g., hemarthrosis, muscle, or mucosal bleeding.

A spontaneous bleeding episode is a bleeding event that occurs for no apparent or known reason, particularly into the joints, muscles, and soft tissues.

Annualized bleeding rate (ABR) while on fitusiran prophylaxis in the fitusiran primary efficacy period and ABR while on on-demand standard of care (SOC) in the SOC periodDay 169 to Day 505 (primary efficacy period) and Day -168 to Day -1 (SOC period)

A bleeding episode is defined as any occurrence of hemorrhage that requires administration of CFCs or BPAs, e.g., hemarthrosis, muscle, or mucosal bleeding.

Annualized joint bleeding rate in the fitusiran primary efficacy period and in the SOC periodDay 169 to Day 505 (primary efficacy period) and Day -168 to Day -1 (SOC period)

A bleeding episode is defined as any occurrence of hemorrhage that requires administration of CFCs or BPAs, e.g., hemarthrosis, muscle, or mucosal bleeding.

A joint bleeding episode is characterized by an unusual sensation in the joint ("aura") in combination with 1) increasing swelling or warmth over the skin over the joint, 2) increasing pain, or 3) progressive loss of range of motion or difficulty in using the limb as compared with baseline.

Change in Haem-A-QOL physical health score and total score during SOC and during fitusiran prophylaxisDay 1 (D1) to Day 505, and from D1 to Day 1009, and during SOC from Day-168 to D-1

The Haem-A-QoL will be provided to participants ≥17 years of age and includes 46 items contributing to 10 QoL domains (physical health, feelings, view of yourself, sports and leisure, work and school, dealing with hemophilia, treatment, future, family planning, partnership, and sexuality). Scoring for each item is based on a 5-point Likert scale (never, rarely, sometimes, often, and all the time), and higher scores represent greater impairment.

Annualized bleeding rate (ABR) in the fitusiran 18-month efficacy periodDay 1 to Day 505

A bleeding episode is defined as any occurrence of hemorrhage that requires administration of CFCs or BPAs, e.g., hemarthrosis, muscle, or mucosal bleeding.

Annualized bleeding rate (ABR) in the fitusiran 36-month treatment periodDay 1 to Day 1009

A bleeding episode is defined as any occurrence of hemorrhage that requires administration of CFCs or BPAs, e.g., hemarthrosis, muscle, or mucosal bleeding.

Number of participants with adverse eventsDate of signed ICF (Day -228 to Day -169) until last visit (approximately 50 months after date of signed ICF)

All AEs (serious or nonserious) will be collected from the signing of the informed consent form (ICF) until last AT follow up visit.

Annualized weight-adjusted consumption of CFC/BPADay -168 until Day 1009

All CFC or BPA doses (including doses per kg body weight) administered during the study treatment will be recorded

Trial Locations

Locations (58)

Center for Inherited Blood Disorders (CIBD) Site Number : 8400012

🇺🇸

Orange, California, United States

University of California San Diego Site Number : 8400011

🇺🇸

San Diego, California, United States

University of Minnesota Site Number : 8400016

🇺🇸

Minneapolis, Minnesota, United States

Hackensack University Site Number : 8400009

🇺🇸

Hackensack, New Jersey, United States

Northwell Health Hemostasis and Thrombosis Center Site Number : 8400015

🇺🇸

New Hyde Park, New York, United States

University Hospitals of Cleveland Site Number : 8400001

🇺🇸

Cleveland, Ohio, United States

UPMC Children's Hospital of Pittsburgh-4401 Penn Ave Site Number : 8400017

🇺🇸

Pittsburgh, Pennsylvania, United States

Children's Medical Center of Dallas Site Number : 8400018

🇺🇸

Dallas, Texas, United States

The Gulf States Hemophilia and Thrombophilia Center Site Number : 8400002

🇺🇸

Houston, Texas, United States

University Of Utah Health Sciences Center Site Number : 8400006

🇺🇸

Salt Lake City, Utah, United States

Medical College of Wisconsin Site Number : 8400007

🇺🇸

Milwaukee, Wisconsin, United States

Investigational Site Number : 1240001

🇨🇦

Hamilton, Ontario, Canada

Investigational Site Number : 1240002

🇨🇦

Hamilton, Ontario, Canada

Investigational Site Number : 1240004

🇨🇦

Toronto, Ontario, Canada

Investigational Site Number : 1560003

🇨🇳

Beijing, China

Investigational Site Number : 1560001

🇨🇳

Guangzhou, China

Investigational Site Number : 1560002

🇨🇳

Jinan, China

Investigational Site Number : 2500003

🇫🇷

Kremlin Bicetre, France

Investigational Site Number : 2500002

🇫🇷

Lille, France

Investigational Site Number : 2500001

🇫🇷

Paris, France

Investigational Site Number : 2760001

🇩🇪

Berlin, Germany

Investigational Site Number : 2760002

🇩🇪

Hamburg, Germany

Investigational Site Number : 3000001

🇬🇷

Athens, Greece

Investigational Site Number : 3000002

🇬🇷

Athens, Greece

Investigational Site Number : 3000003

🇬🇷

Thessaloniki, Greece

Investigational Site Number : 3560004

🇮🇳

Bangalore, India

Investigational Site Number : 3560007

🇮🇳

Bhubaneswar, India

Investigational Site Number : 3560001

🇮🇳

Pune-411011, India

Investigational Site Number : 3560006

🇮🇳

Punjab, India

Investigational Site Number : 3560003

🇮🇳

Vellore, India

Investigational Site Number : 3800003

🇮🇹

Rozzano, Lombardia, Italy

Investigational Site Number : 3800001

🇮🇹

Milano, Italy

Investigational Site Number : 3800002

🇮🇹

Roma, Italy

Investigational Site Number : 3920001

🇯🇵

Kashihara-shi, Nara, Japan

Investigational Site Number : 3920004

🇯🇵

Shinjuku-ku, Tokyo, Japan

Investigational Site Number : 3920003

🇯🇵

Nagoya, Japan

Investigational Site Number : 3920002

🇯🇵

Saitama-shi, Japan

Investigational Site Number : 4100001

🇰🇷

Seoul, Seoul-teukbyeolsi, Korea, Republic of

Investigational Site Number : 4100002

🇰🇷

Seoul, Seoul-teukbyeolsi, Korea, Republic of

Investigational Site Number : 4840002

🇲🇽

Monterrey, Nuevo León, Mexico

Investigational Site Number : 4840004

🇲🇽

Chihuahua, Mexico

Investigational Site Number : 4840001

🇲🇽

Veracruz, Mexico

Investigational Site Number : 6160004

🇵🇱

Lodz, Lódzkie, Poland

Investigational Site Number : 6160002

🇵🇱

Krakow, Malopolskie, Poland

Investigational Site Number : 6160001

🇵🇱

Warszawa, Mazowieckie, Poland

Investigational Site Number : 6820002

🇸🇦

Jeddah, Saudi Arabia

Investigational Site Number : 7100003

🇿🇦

Benoni, South Africa

Investigational Site Number : 7100001

🇿🇦

Parktown, South Africa

Investigational Site Number : 7240002

🇪🇸

La Coruña, A Coruña [La Coruña], Spain

Investigational Site Number : 7240001

🇪🇸

Madrid, Madrid, Comunidad De, Spain

Investigational Site Number : 7240003

🇪🇸

Zaragoza, Spain

Investigational Site Number : 1580002

🇨🇳

Taichung, Taiwan

Investigational Site Number : 1580001

🇨🇳

Taipei, Taiwan

Investigational Site Number : 1580003

🇨🇳

Taipei, Taiwan

Investigational Site Number : 7920002

🇹🇷

Adana, Turkey

Investigational Site Number : 7920004

🇹🇷

Akdeniz, Turkey

Investigational Site Number : 7920001

🇹🇷

Capa, Turkey

Investigational Site Number : 7920003

🇹🇷

Izmir, Turkey

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