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A Phase I, Multicenter, Open-label, First-in-Human, Dose Escalation and Expansion Study of AZD9592 as Monotherapy and in Combination With Anti-cancer Agents in Patients With Advanced Solid Tumors

Phase 1
Recruiting
Conditions
Advanced Solid Tumours, Carcinoma Non-small Cell Lung, Head and Neck Neoplasms
Registration Number
JPRN-jRCT2031230002
Lead Sponsor
Hibi Kazushige
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
Recruiting
Sex
All
Target Recruitment
417
Inclusion Criteria

Age 18 years or more

- Eastern Cooperative Oncology Group (ECOG) Performance Status: 0-1

- Life expectancy 12 weeks or more

- Measurable disease per RECIST v1.1

- Adequate organ and marrow function as defined in the protocol

Additional Inclusion Criteria for Module 1:
- Histologically or cytologically confirmed metastatic or locally advanced EGFRmut., NSCLC; metastatic EGFRwt. NSCLC; recurrent or metastatic HNSCC of the oral cavity; metastatic CRC.

Additional Inclusion Criteria for Module 2:
- Histologically or cytologically confirmed metastatic NSCLC EGFRmut.

Additional Inclusion Criteria for Module 3:
- Histologically or cytologically confirmed metastatic CRC.

Exclusion Criteria

- History of (non-infectious) ILD/pneumonitis that required steroids, has current ILD/pneumonitis, or where suspected ILD/pneumonitis cannot be ruled out by imaging at screening.

- Spinal cord compression or a history of leptomeningeal carcinomatosis.

- Active infection including tuberculosis and HBV, HCV or HIV

- Brain metastases unless treated (prior treatment required only for Module 1), asymptomatic, stable, and not requiring continuous corticosteroids at a dose of > 10 mg prednisone/day or equivalent for at least 4 weeks prior to start of study treatment.

- Participants with cardiac comorbidities as defined in the study protocol

Study & Design

Study Type
Interventional
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
Secondary Outcome Measures
NameTimeMethod
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