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First Tacrolimus Dose Trough Level is Better Than CYP3A5 Genotyping in Tacrolimus Dose Prediction

Conditions
Kidney Transplantation Recipients
Interventions
Registration Number
NCT02356146
Lead Sponsor
Chulalongkorn University
Brief Summary

Tacrolimus dose highly varies among Asian kidney transplant recipients. This can be explained by variety of CYP3A5 expression. CYP3A5 genotyping is highly recommended for patients receiving tacrolimus. Here, we assessed the tacrolimus dose prediction by comparing CYP3A5 expression and tacrolimus dosage using tacrolimus concentration after single dose administration prior to kidney transplantation.

Plasma tacrolimus trough level was measured at 12 hours after first dose of 0.1 mg/kg of tacrolimus (TacC12), orally administered in 51 new kidney transplant recipients. Patients with CYP3A5 inhibitor/inducer co-medications were excluded. Genotyping for CYP3A5 expression were carried out by RT-PCR. The dosages of tacrolimus at post-operative day 7 and dosage which provided stable therapeutic levels in post-operative month 1 to 3 (C0 5-8 ng/mL) were recorded.

The genotyping, TacC12, and target tacrolimus dosage have good correlations.

Detailed Description

Not available

Recruitment & Eligibility

Status
UNKNOWN
Sex
All
Target Recruitment
60
Inclusion Criteria
  • All KT recipients
Exclusion Criteria
  • Recipient who not receiving tacrolimus

Study & Design

Study Type
OBSERVATIONAL
Study Design
Not specified
Arm && Interventions
GroupInterventionDescription
All KT recipientTacrolimus C12-
Primary Outcome Measures
NameTimeMethod
target tacrolimus dose at 3 months3 months
Secondary Outcome Measures
NameTimeMethod
rate of rejection3-12 months
rate of CNI toxicity2-12 months

Trial Locations

Locations (1)

Chulalongkorn University and King Chulalongkorn Memorial Hospital

🇹🇭

Bangkok, Thailand

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