MedPath

Yttrium Y 90 Anti-CD45 Monoclonal Antibody AHN-12 in Treating Patients With Advanced Leukemia

Phase 1
Terminated
Conditions
Leukemia
Myelodysplastic Syndromes
Interventions
Biological: anti-CD45 monoclonal antibody AHN-12
Radiation: yttrium Y 90 anti-CD45 monoclonal antibody AHN-12
Registration Number
NCT00618696
Lead Sponsor
Masonic Cancer Center, University of Minnesota
Brief Summary

RATIONALE: Monoclonal antibodies can block cancer growth in different ways. Some block the ability of cancer cells to grow and spread. Radioactive monoclonal antibodies, such as yttrium Y 90 monoclonal antibody, can find cancer cells and either kill them or carry cancer-killing substances to them without harming normal cells.

PURPOSE: This phase I trial is studying the side effects and best dose of a yttrium Y 90 monoclonal antibody and how much radiation is taken in by the organs in the body in treating patients with advanced leukemia or other hematologic disorder.

Detailed Description

OBJECTIVES:

Primary

* To establish that a dose of 150 mg/m² of nonradiolabeled anti-CD45 monoclonal antibody AHN-12 results in normal biodistribution, normal-organ estimated radiation-absorbed dose of less than 20 Gy, and estimated radiation-absorbed dose of no more than 13 Gy to the red marrow.

Secondary

* To determine the maximum tolerated dose of yttrium Y 90 anti-CD45 monoclonal antibody AHN-12 (\^90Y-AHN-12).

* To determine the human anti-mouse antibody (HAMA) response.

* To define, preliminarily, the antitumor activity of \^90Y-AHN-12.

OUTLINE: This is a dose-escalation study of yttrium Y 90 anti-CD45 monoclonal antibody AHN-12 (\^90Y-AHN-12).

* Biodistribution: Patients receive nonradiolabeled monoclonal antibody AHN-12 IV and an imaging dose of indium Y 111 monoclonal antibody AHN-12 (\^111In-AHN-12) IV over 10 minutes on day 0. Patients undergo whole-body gamma-camera imaging immediately following infusion, at 4-6 hours, and on days 1, 3, 4, and 7. Blood samples are collected prior to each imaging for dosimetry calculations and pharmacokinetics.

Patients also undergo bone marrow biopsy 16-24 hours after infusion for dosimetry calculations. Patients with the expected biodistribution of \^111In-AHN-12, an estimated radiation-absorbed dose to the normal organ of \< 20 Gy, an estimated radiation-absorbed dose to the red marrow of ≤ 13 Gy, and a negative human anti-mouse antibody at day 7 proceed to the therapy portion.

* Treatment: Patients receive nonradiolabeled anti-CD45 monoclonal antibody AHN-12 IV over 60 minutes and escalating therapy doses of yttrium Y 90 anti-CD45 monoclonal antibody AHN-12 (\^90Y-AHN-12) IV over 10 minutes on day 7 or 8.

After completion of study treatment, patients are followed periodically for 1 year.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
4
Inclusion Criteria
  • Histologically confirmed CD45+ diseases:

    • Acute lymphoblastic leukemia or acute myeloid leukemia (AML), meeting any of the following criteria:

      • Primary refractory disease
      • Relapsed disease, defined as persistent disease following a minimum of 2 different standard chemotherapy induction attempts at time of diagnosis or at relapse
    • Acute myelogenous leukemia (AML), primary refractory or relapsed disease - defined as persistent disease after a minimum of two different standard chemotherapy induction attempts at time of diagnosis or relapse

    • Advanced myelodysplastic syndrome (MDS) defined as > or = 15% bone marrow blasts following a minimum of one standard chemotherapy induction attempt

    • AML arising from preexisting MDS, refractory - defined as persistent disease following a minimum of one standard chemotherapy induction attempt

    • Chronic myelogenous leukemia (CML) following blast crisis (> or = 15% marrow blasts following a minimum of one standard chemotherapy induction attempt

  • Peripheral leukemic blasts (by morphology) must be < 5,000/μL (hydroxyurea to control peripheral blast count allowed)

  • Must have source of allogeneic stem cells (sibling, unrelated cord[s], or donor) identified prior to initiation of protocol therapy

  • Eastern Cooperative Oncology Group (ECOG) performance status (PS) 0-2 or Karnofsky PS 60-100%

  • Life expectancy > 12 weeks

  • Total bilirubin ≤ 2.5 times upper limit of normal (ULN)

  • aspartate aminotransferase (AST) and Alanine transaminase (ALT) ≤ 2.5 times upper limit of normal (ULN)

  • Creatinine ≤ 1.3 mg/dL OR creatinine clearance ≥ 60 mL/min

  • Left ventricular ejection fraction (LVEF) ≥ 45% by Multi Gated Acquisition Scan (MUGA) or echocardiogram (ECHO)

  • Carbon Monoxide Diffusing Capacity (DLCO) (corrected) ≥ 50% of predicted

  • Human anti-mouse antibody (HAMA) must be negative

  • Not pregnant or nursing

  • Fertile patients must use effective contraception

  • Human immunodeficiency virus (HIV) negative

  • Recovered from all prior therapy

  • At least 7 days since prior biologic agents

Exclusion Criteria
  • Bone marrow cellularity < 15%

  • Known brain metastases or active central nervous system (CNS) disease

  • History of allergic reactions attributed to compounds of similar chemical or biologic composition to ^90Y-AHN-12 or other agents used in study

  • Uncontrolled illness, including, but not limited to, any of the following:

    • Ongoing or active infection
    • Symptomatic or congestive heart failure
    • Unstable angina pectoris
    • Cardiac arrhythmia
    • Psychiatric illness or social situations that would limit compliance with study requirements
  • Other concurrent investigational agents

  • Prior allogeneic transplantation

  • Less than 60 days since prior autologous transplantation with relapsed disease

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
AHN-12anti-CD45 monoclonal antibody AHN-122.0, 5.0, 7.5, 10.0 or 12.5 mCi/m\^2 of \^90Y-AHN-12 at Day 7/8
AHN-12yttrium Y 90 anti-CD45 monoclonal antibody AHN-122.0, 5.0, 7.5, 10.0 or 12.5 mCi/m\^2 of \^90Y-AHN-12 at Day 7/8
Primary Outcome Measures
NameTimeMethod
Biodistribution of nonradiolabeled anti-CD45 monoclonal antibody AHN-12Within 1 hour, 4-6 hours, Days 1, 3, 4 and 7 post infusion
Secondary Outcome Measures
NameTimeMethod
Presence of human antibody to murine antibodyat baseline and at 28 days, 90 days, and 6 months after completion of study treatment
Dose-limiting toxicity and responseat days 28 and 90 after completion of study treatment
Maximum tolerated dose of yttrium Y 90 anti-CD45 monoclonal antibody AHN-12Week 8

Trial Locations

Locations (1)

Masonic Cancer Center at University of Minnesota

🇺🇸

Minneapolis, Minnesota, United States

© Copyright 2025. All Rights Reserved by MedPath