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Combination of Rosuvastatin and Ezetimibe to improve Postprandial Triglyceride and Glucose in Patients with Diabetes Mellitus or Metabolic Syndrome

Not Applicable
Completed
Conditions
Endocrine, nutritional and metabolic diseases
Registration Number
KCT0003198
Lead Sponsor
Seoul National University Hospital
Brief Summary

Combination therapy with ezetimibe plus rosuvastatin significantly lowered post-prandial TG and LDL cholesterol compared with rosuvastatin monotherapy in patients with type 2 diabetes mellitus. Addition of ezetimibe may have effects beyond lowering LDL cholesterol. In conclusion, 12-week treatment with ezetimibe 10mg plus rosuvastatin 10mg was more effective in lowering postprandial TG and LDL cholesterol than was rosuvastatin 10mg in patients with type 2 diabetes. Combination therapy was also associated with favorable results in insulin resistance. The results of the current study could help better understand the mechanism behind beneficial effects of ezetimibe.

Detailed Description

Not available

Recruitment & Eligibility

Status
Completed
Sex
All
Target Recruitment
150
Inclusion Criteria

1) Patients over age of 20 and with a LDL-cholesterol = 100mg/dL, who are not taking medication for dyslipidmeia in the 4 weeks prior to randomization.
2) Patient with either type 2 diabetes mellitus or metabolic syndrome
(1) Type 2 diabetes mellitus
- on oral hypoglycemic agents
- newly diagnosed patients (HbA1c =6.5%, fasting bloos glucose =126mg/dL, PP2 =200mg/dL on post-prandial testing, or random glucose = 200mg/dL with specific symptoms of diabetes)

(2) Metabolic syndrome
- meeting 3 of the below criteria, accoring to NCEP ATP III guidelines modified to Korean standards
? Waist circumference >90 cm in men, >85 cm in women
? Triglycerides 150 mg/dL or greater
? HDL-cholesterol <40 mg/dL in men and <50 mg/dL in women
? BP 130/85 mmHg or greater, or on treatment for hypertension
? Fasting glucose 110 mg/dL or greater, or on treatment for diabetes

Exclusion Criteria

(1) Hypersensitivity to the study drug or its substance
(2) Active liver disease, or AST/ALT levels over 5 times the upper limit of normal
(3) Myopathy or serum CK levels over 5 times the upper limit of normal
(4) Cyclosporine use
(5) Moderate+ kidney dysfunction (creatinine clearance, CLcr <30mL/min)
(6) Pregnancy or breasfeeeding
(7) Alcoholic
(8) Medications that may influence the lipid profile:
- fibrate, bile acid sequestrants, niacin, drugs for management of obesity, systemic steroids, fish oil, fiber-based laxatives, phytosterol margarines, etc.
- medications that influence thyroid function (medications for thyroid replacement therapies are allowed)
(9) Other reasons that the investigator deems to be unfit for enrollment

Study & Design

Study Type
Interventional Study
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
The change(%) in post-prandial TG
Secondary Outcome Measures
NameTimeMethod
Absolute change in post-prandial TG;Absolute change and percentage change in post-prandial glucose;Absolute change and percentage change in TG/HDL ratio;Absolute change and percentage change in post-prandial Apo-B;Change in insulin sensitivity;Absolute change and percentage change in C-reactive protein;Percentage of patients reaching LDL-C target goal according to NCEP ATP III risk
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