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Trastuzumab Deruxtecan (T-DXd) in Patients Who Have Hormone Receptor-negative and Hormone Receptor-positive HER2-low or HER2 IHC 0 Metastatic Breast Cancer

Phase 3
Recruiting
Conditions
Breast Cancer
Interventions
Registration Number
NCT05950945
Lead Sponsor
Daiichi Sankyo
Brief Summary

This study will evaluate the safety and efficacy of trastuzumab deruxtecan (T-DXd) in participants with human epidermal growth factor receptor 2 (HER2)-low or HER2 immunohistochemistry (IHC) 0 (who are both hormone receptor \[HR\]-negative and HR-positive) unresectable and/or metastatic breast cancer.

Detailed Description

The primary endpoint of interest in this study is time to next treatment (TTNT), a measure that will determine how long T-DXd allows patients to derive clinical benefit from the study drug.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
250
Inclusion Criteria
  • Sign and date the main informed consent form

  • Must agree to provide a newly obtained or archival baseline biopsy from primary and/or metastatic lesion.

  • Pathologically documented Breast Cancer (BC) tumor

    • Is unresectable and/or metastatic.

    • Is hormone receptor-negative or hormone receptor-positive.

      • Must include percentage of positively stained cells to characterize if hormone receptor-positive or -negative.
    • Has confirmed HER2 IHC 1+ or IHC 2+/ISH- (HER2-low) status or HER2 IHC 0 status as determined according to ASCO CAP 2018 guidelines1 based on sample collected during Tissue Screening as described above.

    • Was never previously HER2-positive (IHC 3+ or IHC 2+/ISH+) on prior pathology testing (per ASCO CAP guidelines).

    • Was never previously treated with anti-HER2 therapy in the metastatic setting.

  • Has had at least one and up to two prior lines of therapy in the metastatic setting.

    • In participants with hormone receptor-positive HER2-low metastatic BC (Cohort 3):

      • Has recurrent disease <2 years from the initiation of adjuvant ET OR
      • Has disease progression on CDK4/6 inhibitor-based regimen within 12 months of completion of adjuvant therapy with a CDK4/6 inhibitor OR
      • Has disease progression within the first 12 months of CDK4/6 in the first line metastatic setting
  • Presence of at least one measurable lesion based on computed tomography or magnetic resonance imaging.

  • Participants with brain metastases are allowed in the study. The brain lesion(s) should be small (<2 cm), untreated, asymptomatic, not requiring urgent medical intervention, and are asymptomatic and clinically stable.

  • Has an Eastern Cooperative Oncology Group performance status of 0 or 1.

  • Has a minimum life expectancy of 12 weeks at Screening.

  • Has a left ventricular ejection fraction ≥50% within 28 days before enrollment.

  • Has adequate organ and bone marrow function within 28 days before enrollment.

  • Has adequate treatment washout period before enrollment.

  • Male and female subjects of reproductive/childbearing potential must agree to use a highly effective form of contraception.

Exclusion Criteria
  • Prior treatment with an antibody drug conjugate (ADC).
  • Uncontrolled or significant cardiovascular disease.
  • Has a corrected QT interval prolongation.
  • Has a history of (non-infectious) interstitial lung disease (ILD)/pneumonitis that required steroids, has current ILD/pneumonitis, or where suspected ILD/pneumonitis cannot be ruled out by imaging at Screening.
  • Has spinal cord compression or clinically active central nervous system metastases.
  • Has multiple primary malignancies within 3 years, except adequately resected non-melanoma skin cancer, curatively treated in situ disease, other solid tumors curatively treated, or contralateral BC.
  • Has a history of severe hypersensitivity reactions to either the drug substances or inactive ingredients in the drug product.
  • Has a history of severe hypersensitivity reactions to other monoclonal antibodies.
  • Has an uncontrolled infection requiring intravenous (IV) antibiotics, antivirals, or antifungals.
  • Active primary immunodeficiency, known uncontrolled active human immunodeficiency virus (HIV) infection, or active hepatitis B or C infection.
  • Has history of receiving a live, attenuated vaccine (messenger RNA and replication-deficient adenoviral vaccines are not considered attenuated live vaccines) within 30 days prior to the first exposure to study drug.
  • Has unresolved toxicities from previous anticancer therapy, defined as toxicities (other than alopecia) not yet resolved to Grade ≤1 or baseline.
  • Is pregnant or breastfeeding or planning to become pregnant.
  • Lung-specific intercurrent clinically significant illnesses.
  • Any autoimmune, connective tissue, or inflammatory disorders.
  • Prior complete pneumonectomy.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Cohort 2: HR-negative, HER2 IHC 0Trastuzumab DeruxtecanParticipants with HR-negative HER2 IHC 0 unresectable and/or metastatic breast cancer who have received at least one and at most two prior lines of therapy in the metastatic setting will receive T-DXd.
Cohort 1: HR-negative, HER2-lowTrastuzumab DeruxtecanParticipants with HR-negative HER2-low unresectable and/or metastatic breast cancer who have received at least one and at most two prior lines of therapy in the metastatic setting will receive T-DXd.
Cohort 3: HR-positive, HER2-lowTrastuzumab DeruxtecanParticipants with HR-positive HER2-low unresectable and/or metastatic breast cancer who have received at least one and at most two prior lines of therapy in the metastatic setting will receive T-DXd. Participants must also have recurrent disease \<2 years from the initiation of adjuvant ET or have disease progression on CDK4/6 inhibitor-based regimen within 12 months of completion of adjuvant therapy with a CDK4/6 inhibitor or have disease progression within the first 12 months of CDK4/6 in the first line metastatic setting.
Cohort 4: HR-positive, HER2 IHC 0Trastuzumab DeruxtecanParticipants with HR-positive HER2 IHC 0 unresectable and/or metastatic breast cancer who have received at least one and at most two prior lines of therapy in the metastatic setting will receive T-DXd.
Primary Outcome Measures
NameTimeMethod
Time From the Start of T-DXd to Initiation of Subsequent Anticancer Treatment (TTNT)Until subsequent therapy or death, assessed up to 24 months

TTNT is defined as the time interval from the date of first dose of T-DXd to the initiation of the next anticancer treatment or death due to any cause.

Secondary Outcome Measures
NameTimeMethod
Time From Start of T-DXd to Discontinuation of T-DXd or Death (TTD)Until treatment discontinuation or death, up to 24 months

TTD is defined as the time interval from the date of first dose of T-DXd to the date of discontinuation of T-DXd or death due to any cause.

Objective Response Rate (ORR)Until progression, assessed up to 24 months

ORR is defined as the proportion of participants with a best overall response (BOR) of confirmed complete response (CR) or confirmed partial response (PR) according to the investigator and per RECIST version 1.1 criteria.

Time to First and Definitive Deterioration in European Organization for Research and Treatment of Cancer Quality of Life Questionnaires (EORTC-QLQ) ScalesAssessed up to 24 months

Time to first and definitive deterioration in EORTC-QLQ scales. Scale scores range from 0-100. For functioning and global health status/ QoL scales, higher scores indicate better functioning or global health status/QoL. For symptom scales, higher scores indicate greater symptom burden.

Time to First and Definitive Deterioration in EuroQol Questionnaire-5 Dimensions-5 Levels (EQ-5D-5L) Visual Analog Scale (VAS)Assessed up to 24 months

Time to first and definitive deterioration in EQ-5D-5L VAS. The EQ-5D-5L VAS ranging from 0 (worse) to 100 (better) is used to assess an overall rating of participant's current health status. Higher scores indicate better clinical outcomes.

Patient's Global Impression of Change (PGI-C) ResponseAssessed up to 24 months

The PGI-C is a single-item questionnaire asking for the participant's overall impression of changes in clinical condition from baseline (prior to study drug initiation), where 1 is "Normal" and 7 is "Severely ill". Lower scores indicate better clinical outcome.

Mean Change from Baseline in European Organization for Research and Treatment of Cancer Quality of Life Questionnaires (EORTC-QLQ)-BR45 ScoreAssessed up to 24 months

Change from baseline in the EORTC QLQ-BR45 scale scores range from 0-100. For functioning and global health status/ QoL scales, higher scores indicate better functioning or global health status/QoL. For symptom scales, higher scores indicate greater symptom burden.

Real-World Progression Free Survival (PFS)Until progression or death, assessed up to 24 months

Real-world PFS is defined as time from date of first dose of T-DXd to time of disease progression per investigator assessment based on Response Evaluation Criteria in Solid Tumors (RECIST) v1.1 or death due to any cause.

Number of Participants With Treatment-emergent Adverse Events (TEAEs)Up to follow up period, up to 24 months

TEAEs are graded according to National Cancer Institute-Common Terminology Criteria for Adverse Events (NCI-CTCAE) v5.0. A TEAE is defined as an adverse event (AE) that occurs, having been absent before the first dose of study drug, or has worsened in severity or seriousness after initiating the study drug until 47 days after the last dose of the study drug.

Mean Change from Baseline in European Organization for Research and Treatment of Cancer Quality of Life Questionnaires (EORTC-QLQ)-C30 ScoreAssessed up to 24 months

Change from baseline in the EORTC-QLQ-C30 scale scores range from 0-100. For functioning and global health status/ QoL scales, higher scores indicate better functioning or global health status/QoL. For symptom scales, higher scores indicate greater symptom burden.

Mean Change from Baseline in EuroQol Questionnaire-5 Dimensions-5 Levels (EQ-5D-5L)Assessed up to 24 months

Change from baseline in EQ-5D-5L. The EQ-5D-5L is a health-related QoL questionnaire based on five dimensions of health: mobility, self-care, usual activities, pain/discomfort, and anxiety/depression. Each dimension contains five levels: no problems, slight, moderate, severe, and extreme problems. The EQ-5D-5L results can be converted into a single utility value. Utility values range from 0 to 1, with 1 corresponding to perfect health and 0 corresponding to a health status equivalent to death. In addition, participants can provide an overall rating of their current health status using a visual analog scale ranging from 0 (worse) to 100 (better).

Mean Change From Baseline in EuroQol Questionnaire-5 Dimensions-5 Levels (EQ-5D-5L) Index ScoreAssessed up to 24 months

Change from baseline in EQ-5D-5L index score. The EQ-5D-5L index score ranges from less than 0 (worse) to 1 (better), with higher scores representing a better health status.

Mean Change From Baseline in EuroQol Questionnaire-5 Dimensions-5 Levels (EQ-5D-5L) Visual Analog Scale (VAS)Assessed up to 24 months

Change from baseline in EQ-5D-5L VAS. The EQ-5D-5L VAS ranging from 0 (worse) to 100 (better) is used to assess an overall rating of participant's current health status. Higher scores indicate better clinical outcomes.

Patient's Global Impression of Treatment Tolerability (PGI-TT) ResponseAssessed up to 24 months

The PGI-TT is a single-item questionnaire asking for the subject's overall impression of treatment tolerability over the past week, where 1 is "Not at all" and 5 is "Very much". Higher scores indicate a worse outcome.

Patient's Global Impression of Severity (PGI-S) ResponseAssessed up to 24 months

The PGI-S is a single-item questionnaire asking for the subject's overall impression of symptoms assessed over the past week, where 1 is "Normal" and 4 is "Severe". Lower scores indicate better clinical outcome.

Trial Locations

Locations (82)

Mount Sinai Medical Center

🇺🇸

Miami Beach, Florida, United States

USF College of Medicine

🇺🇸

Tampa, Florida, United States

Dana-Farber Cancer Institute

🇺🇸

Boston, Massachusetts, United States

Beth Israel Lahey Health

🇺🇸

Burlington, Massachusetts, United States

Overlook Medical Center

🇺🇸

Summit, New Jersey, United States

Mater Hospital Sydney

🇦🇺

North Sydney, New South Wales, Australia

Monash Medical Centre Moorabbin

🇦🇺

East Bentleigh, Victoria, Australia

Institut Jules Bordet

🇧🇪

Anderlecht, Belgium

GZA Ziekenhuizen

🇧🇪

Wilrijk, Belgium

Universitair Ziekenhuis Brussel

🇧🇪

Bruxelles, Belgium

Cliniques Universitaires Saint-Luc

🇧🇪

Bruxelles, Belgium

UZ Leuven

🇧🇪

Leuven, Belgium

Centre Hospitalier Universitaire de Liege Sart-Tilman

🇧🇪

Liege, Belgium

Centro de Oncologia - Unidade Brasília - Hospital Sírio Libanês

🇧🇷

Brasilia, Brazil

CIONC-Centro Integrado de Oncologia de Curitiba

🇧🇷

Curitiba, Brazil

Hospital Erasto Gaertner - Liga Paranaense de Combate ao Câncer

🇧🇷

Curitiba, Brazil

CEPON - Centro de Pesquisas Oncológicas de Santa Catarina

🇧🇷

Florianopolis, Brazil

Oncosite - Centro de Pesquisa Clinica e Oncologia

🇧🇷

Ijuí, Brazil

Fundação Doutor Amaral Carvalho

🇧🇷

Jaú, Brazil

Instituto de Cancer de Londrina

🇧🇷

Londrina, Brazil

Hospital das Clínicas FMRP-USP

🇧🇷

Riberão Preto, Brazil

Hospital Nossa Senhora da Conceicao

🇧🇷

Rio Grande Do Sul, Brazil

Ensino e Terapia de Inovação Clínica AMO-ETICA

🇧🇷

Salvador, Brazil

Catarina Pesquisa Clinica

🇧🇷

Santa Catarina, Brazil

CEPHO - Centro de Estudos e Pesquisas de Hematologia e Oncologia

🇧🇷

Santo André, Brazil

Fundacao Faculdade Regional de Medicina de Sao Jose do Rio Preto

🇧🇷

Sao Jose do Rio Preto, Brazil

ICESP - Instituto do Câncer do Estado de São Paulo Octavio Frias de Oliveira

🇧🇷

São Paulo, Brazil

Clínica de Pesquisas e Centro de Estudos em Oncologia Ginecológica e Mamária Ltda

🇧🇷

São Paulo, Brazil

Beijing Hospital

🇨🇳

Beijing, China

307 Hospital of PLA

🇨🇳

Beijing, China

Fujian Cancer Hospital

🇨🇳

Fujian, China

Sun Yat sen University Cancer Center

🇨🇳

Guangzhou, China

Zhejiang Cancer Hospital

🇨🇳

Hangzhou, China

Anhui Provincial Cancer Hospital

🇨🇳

Hefei, China

Shandong Cancer Hospital

🇨🇳

Jinan, China

Yunnan Cancer Hospital

🇨🇳

Kunming, China

Nanchang People's Hospital

🇨🇳

Nanchang, China

Jiangxi Cancer Hospital

🇨🇳

Nanchang, China

The Affiliated Hospital of Qingdao University

🇨🇳

Qingdao, China

Fudan University Shanghai Cancer Center

🇨🇳

Shanghai, China

Henan Cancer Hospital

🇨🇳

Zhengzhou, China

Cork University Hospital

🇮🇪

Cork, Ireland

St Vincent's University Hospital

🇮🇪

Dublin, Ireland

St James Hospital

🇮🇪

Dublin, Ireland

Beaumont Hospital

🇮🇪

Dublin, Ireland

Galway University Hospital

🇮🇪

Galway, Ireland

Istituto Tumori Giovanni Paolo II IRCCS Ospedale Oncologico Bari

🇮🇹

Bari, Italy

Azienda Ospedaliera Universitaria Policlinico Sant Orsola Malpighi IRCCS

🇮🇹

Bologna, Italy

Istituto Nazionale per la Ricerca sul Cancro di Genova

🇮🇹

Genova, Italy

Ospedale San Raffaele

🇮🇹

Milano, Italy

Humanitas Istituto Clinico Catanese

🇮🇹

Misterbianco, Italy

Istituto Nazionale Tumori Fondazione G Pascale

🇮🇹

Naples, Italy

IOV - Istituto Oncologico Veneto IRCCS

🇮🇹

Padova, Italy

Nuovo Ospedale di Prato

🇮🇹

Prato, Italy

Azienda Ospedaliera Universitaria Policlinico Umberto I - Università di Roma La Sapienza

🇮🇹

Rome, Italy

Fondazione Policlinico Universitario Agostino Gemelli IRCCS

🇮🇹

Rome, Italy

Ospedale Santa Chiara

🇮🇹

Trento, Italy

Amsterdam UMC, Locatie VUMC

🇳🇱

Amsterdam, Netherlands

Amphia Ziekenhuis Molengracht

🇳🇱

Breda, Netherlands

Haga Ziekenhuis

🇳🇱

Den Haag, Netherlands

Medisch Centrum Leeuwarden

🇳🇱

Leeuwarden, Netherlands

Alrijne Ziekenhuis Leiden

🇳🇱

Leiden, Netherlands

Maastricht University Medical Center

🇳🇱

Maastricht, Netherlands

Elisabeth TweeSteden Ziekenhuis

🇳🇱

Tilburg, Netherlands

Bernhoven Uden

🇳🇱

Uden, Netherlands

Hospital de Braga

🇵🇹

Braga, Portugal

Instituto Português de Oncologia de Lisboa Francisco Gentil, EPE

🇵🇹

Lisboa, Portugal

Centro Hospitalar de Lisboa Norte E P E Hospital de Santa Maria

🇵🇹

Lisboa, Portugal

Hospital de la Santa Creu i Sant Pau

🇪🇸

Barcelona, Spain

ICO l'Hospitalet - Hospital Duran i Reynals

🇪🇸

Barcelona, Spain

Hospital Universitario Virgen de las Nieves

🇪🇸

Granada, Spain

Complejo Hospitalario Universitario Insular Materno-Infantil

🇪🇸

Las Palmas de Gran Canaria, Spain

Hospital Beata Maria Ana

🇪🇸

Madrid, Spain

Hospital Universitario 12 de Octubre

🇪🇸

Madrid, Spain

Hospital Universitario Puerta de Hierro Majadahonda

🇪🇸

Majadahonda, Spain

Hospital General Universitario Morales Meseguer

🇪🇸

Murcia, Spain

Clinica Universidad de Navarra

🇪🇸

Pamplona, Spain

Hospital Universitario Donostia

🇪🇸

San Sebastian, Spain

Complejo Hospitalario Universitario de Santiago

🇪🇸

Santiago de Compostela, Spain

Hospital Universitario Virgen Macarena

🇪🇸

Sevilla, Spain

Hospital Clinico Universitario de Valencia

🇪🇸

Valencia, Spain

Hospital Arnau de Vilanova de Valencia

🇪🇸

Valencia, Spain

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