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Phase 3 Study of Intranasal Carbetocin (LV-101) in Patients With Prader-Willi Syndrome

Phase 3
Completed
Conditions
Prader-Willi Syndrome
Interventions
Drug: placebo
Drug: 3.2 mg intranasal carbetocin
Drug: 9.6 mg intranasal carbetocin
Registration Number
NCT03649477
Lead Sponsor
Levo Therapeutics, Inc.
Brief Summary

This Phase 3 study is designed to test the effectiveness of intranasal carbetocin (LV-101) in participants with Prader-Willi syndrome (PWS). Carbetocin is an oxytocin analog (a man-made chemical that is like oxytocin). This study will also evaluate the safety and tolerability of LV-101.

Detailed Description

This is a Phase 3 randomized, double-blind study with an 8-week, placebo-controlled period designed to test the effectiveness, safety, and tolerability of LV-101 in participants with PWS.

Effectiveness will be measured using both caregiver-reported and clinician-reported measures of hyperphagia (extreme hunger), obsessive and compulsive behaviors, and anxiety. Safety and tolerability will be measured by adverse events, laboratory tests, and physical exams.

After the 8-week placebo-controlled period, there will be a long-term follow-up period of 56 weeks and an optional extension period after study week 64 during which all participants will receive active treatment with LV-101. At Week 8, participants who were randomized to placebo in the placebo-controlled period will be randomized to one of the two LV-101 doses, administered three times per day before meals.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
130
Inclusion Criteria
  • Genetically-confirmed Prader-Willi syndrome
  • Provide voluntary, written informed consent (parent(s) / legal guardian(s) of participant); provide voluntary, written assent (participants, as appropriate)
  • PWS Nutritional Phase 3 (hyperphagic, rarely feels full)
Exclusion Criteria
  • Living in a group home
  • Genetically diagnosed Schaaf-Yang syndrome or other genetic, hormonal, or chromosomal cognitive impairment
  • New food-related interventions, including environment or dietary restrictions, within 1 month of screening
  • Dose of any allowed chronic concomitant medications or supplements that have not been stable for ≥3 months prior to the study or is not expected to remain stable while participating in the study; adjustments in growth hormone dose ≤10% are not exclusionary
  • Presence of cardiovascular disorders, epilepsy, frequent migraines, or severe asthma
  • More than 3 episodes of sinusitis in the 12 months prior to Screening Visit or presence of nasal diseases that may affect deposition of intranasal medication
  • Unwilling to abstain from nasal saline, other nasal irrigation, or other intranasal medications for 2 weeks prior to the Baseline visit and during the 8-week, placebo-controlled period of the study
  • Use of weight loss medication, oxytocin, carbetocin, or vasopressin in the 6 months prior to screening
  • Participation in an interventional research study involving another investigational medication or device in the 6 months prior to screening or during the study
  • Based on the judgment of the Investigator, is unsuitable for the study for any reason, including but not limited to unstable medical condition, inability to comply with the protocol, or other risk to subject or to the integrity of the study

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Placeboplacebomatched placebo during first 8-weeks; prospectively randomized 1:1 to either one of the two doses of carbetocin during 56-week follow-up and optional extension periods
3.2 mg of LV-1013.2 mg intranasal carbetocin3.2 mg of LV-101 during first 8-weeks; remain on same dose during 56-week follow-up and optional extension periods
9.6 mg of LV-1019.6 mg intranasal carbetocin9.6 mg of LV-101 during first 8-weeks; remain on same dose during 56-week follow-up and optional extension periods
Primary Outcome Measures
NameTimeMethod
Hyperphagia BehaviorBaseline to Week 8

Change in hyperphagia (extreme hunger) as measured by the Hyperphagia Questionnaire for Clinical Trials (HQ-CT) Total Score versus placebo.

Score range: 0-36; higher scores mean a worse outcome. Reduction in score indicates improvement.

Obsessive and Compulsive Behaviorsbaseline to Week 8

Change in obsessive and compulsive behaviors as measured by the Children's Yale-Brown Obsessive-Compulsive Scale (CY-BOCS) Total Score versus placebo.

Score range: 0-40; higher scores mean a worse outcome. Reduction in score indicates improvement.

Secondary Outcome Measures
NameTimeMethod
AnxietyBaseline to Week 8

Change in participant anxiety as measured by the PWS Anxiety and Distress Questionnaire (PADQ) Total Score versus placebo.

Score range: 0-56; higher scores mean a worse outcome. Reduction in score indicates improvement.

Hyperphagia Behavior (Subset)Baseline to Week 8

Change in hyperphagia as measured by the change in specified subsets of HQ-CT questions versus placebo.

Score range: 0-24; higher scores mean a worse outcome. Reduction in score indicates improvement.

Global ImpressionWeek 8

Clinical Global Impression of Change (CGI-C) score versus placebo. Score range: 1-7; higher scores mean a worse outcome. Reduction in score indicates improvement.

Trial Locations

Locations (24)

Ann & Robert H. Lurie Children's Hospital of Chicago

🇺🇸

Chicago, Illinois, United States

University of Harvard Boston Children's Hospital

🇺🇸

Boston, Massachusetts, United States

Vanderbilt University School of Medicine

🇺🇸

Nashville, Tennessee, United States

Children's Hospital of San Antonio

🇺🇸

San Antonio, Texas, United States

Cardinal Glennon Children's Medical Center

🇺🇸

Saint Louis, Missouri, United States

Children's Hospital of Los Angeles (USC)

🇺🇸

Los Angeles, California, United States

Nationwide Children's Hospital

🇺🇸

Columbus, Ohio, United States

British Columbia Children's Hospital

🇨🇦

Vancouver, British Columbia, Canada

Kansas University Medical Center

🇺🇸

Kansas City, Kansas, United States

Children's Hospitals and Clinics of Minnesota

🇺🇸

Saint Paul, Minnesota, United States

University of Oklahoma Health Sciences Center

🇺🇸

Tulsa, Oklahoma, United States

Children's Hospital of Philadelphia

🇺🇸

Philadelphia, Pennsylvania, United States

Texas Children's Hospital

🇺🇸

Houston, Texas, United States

Queensland Children's Hospital

🇦🇺

South Brisbane, Queensland, Australia

University of Alberta

🇨🇦

Edmonton, Alberta, Canada

Toronto Hospital for Sick Kids

🇨🇦

Toronto, Ontario, Canada

CHU Ste Justine

🇨🇦

Montréal, Quebec, Canada

Children's National

🇺🇸

Washington, District of Columbia, United States

Rady Children's Hospital San Diego

🇺🇸

San Diego, California, United States

University of Utah

🇺🇸

Salt Lake City, Utah, United States

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

Phoenix Children's Hospital

🇺🇸

Phoenix, Arizona, United States

University of Florida

🇺🇸

Gainesville, Florida, United States

Children's Hospital Colorado

🇺🇸

Aurora, Colorado, United States

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