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Clinical Trials to Reduce the Risk of Antimicrobial Resistance

Phase 2
Terminated
Conditions
Bacterial Pneumonia
Interventions
Drug: Parenteral aminoglycoside; tobramycin for injection USP OR gentamicin sulfate injection solution concentrate 5mg.kg IV q24h; amikacin sulfate injection USP 20 mg/kg IV q24h
Device: tobramycin nebulization
Registration Number
NCT01570192
Lead Sponsor
University of Florida
Brief Summary

The primary objective of this study is to demonstrate a low rate of emergence of antibiotic resistance in P. aeruginosa and Acinetobacter spp during the treatment of hospitalized patients with pneumonia requiring mechanical ventilation treated with PD optimized meropenem administered as a prolonged infusion in combination with a parenteral aminoglycoside plus tobramycin by inhalation (Group 1) compared to therapy with meropenem alone (Group 2 - control arm).

Detailed Description

The goal of this clinical study is to demonstrate that the application of pharmacodynamic dosing principles to the antibiotic treatment of hospitalized subjects with culture-documented pneumonia (including HABP, VABP and HCAP) requiring mechanical ventilation can inhibit the emergence of antibiotic-resistant organisms during treatment and therefore may improve the rate of a satisfactory clinical response. Antibiotic resistance is defined as an increase in meropenem or aminoglycoside MIC by two tube dilutions (fourfold) from baseline. In animal models of infection, the pharmacodynamic driver for bactericidal effect by β lactam antibiotics such as meropenem is the proportion of the dosing interval during which plasma drug levels are maintained above the MIC of the causative pathogen. The hypothesis of this study is that prolongation of time above MIC by increasing total meropenem dose and the duration of infusion will counter-select for the emergence of antimicrobial resistance during the treatment of hospitalized subjects with pneumonia (i.e. HABP, VABP and HCAP) caused by P.aeruginosa, Acinetobacter species (spp), or other pathogens with intermediate susceptibility to meropenem, and that the addition of parenteral aminoglycosides (amikacin, tobramycin or gentamicin) and nebulized aminoglycoside (tobramycin) given along optimal pharmacodynamic principles will further reduce the likelihood of resistance emergence, particularly among the non-fermenting Gram-negative bacilli, such as Pseudomonas aeruginosa and Acinetobacter spp. The observed incidence of resistance emergence to meropenem will be compared across therapeutic regimens.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
43
Inclusion Criteria

Not provided

Exclusion Criteria

Subjects with pneumonia caused by pathogens resistant to meropenem (MIC greater than or equal to 16µg/ml) or a prior meropenem therapy failure.

Subjects with contra-indications to ANY study medication, in particular with known or suspected allergy or hypersensitivity.

Women who are pregnant or lactating.

Subjects taking anticonvulsant medications for a known seizure disorder.Patients with a history of seizures, AND who are stabilized on anti-seizure medication, may be enrolled into the study at the discretion of the site investigator.

Subjects with known or suspected community acquired bacterial pneumonia (CABP) or viral pneumonia; or Subjects with acute exacerbation of chronic bronchitis without evidence of pneumonia.

Subjects with primary lung cancer or another malignancy metastatic to the lungs.

Subjects who were previously enrolled in this study.

Subjects who have had an investigational drug or have used an investigational device within 30 days prior to entering the study.

Subjects with another focus of infection requiring concurrent antibiotics that would interfere with evaluation of the response to study drug.

Subjects with cystic fibrosis, AIDS with a CD4 lymphocyte count <200 cells/µl, neutropenia (absolute neutrophil count <500 cells/ml), known or suspected active tuberculosis.

Subjects with little chance of survival for the duration of study therapy.

Subjects with an APACHE II score >35.

Subjects with underlying condition(s) which would make it difficult to interpret response to the study drugs.

Subjects with hypotension or acidosis despite attempts at fluid resuscitation. Subjects requiring ongoing treatment with vasopressors will be eligible for the study if their hypotension is controlled and acidosis has resolved. Subjects with intractable septic shock are not eligible for enrollment.

Subjects who have undergone bone marrow transplantation.

Subjects with profound hypoxia as defined by a PaO2/FiO2 ratio <100.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
IV meropenem; parenteral aminoglycosideLinezolid or Vancomycin (per institutional guidelines) will be available for MRSA coverage.Subjects assigned to this group will receive: * IV meropenem (2 g infused over 3 hrs q 8 hr); * a parenteral aminoglycoside (tobramycin or gentamicin-5mg/kg IV Q24h or amikacin 20 mg/kg IV Q24h) * tobramycin nebulization Linezolid or vancomycin (per institutional guidelines) will be available for MRSA coverage to treat potential Gram-positive pathogens.
IV meropenem; parenteral aminoglycosideIV meropenemSubjects assigned to this group will receive: * IV meropenem (2 g infused over 3 hrs q 8 hr); * a parenteral aminoglycoside (tobramycin or gentamicin-5mg/kg IV Q24h or amikacin 20 mg/kg IV Q24h) * tobramycin nebulization Linezolid or vancomycin (per institutional guidelines) will be available for MRSA coverage to treat potential Gram-positive pathogens.
IV meropenem; parenteral aminoglycosideParenteral aminoglycoside; tobramycin for injection USP OR gentamicin sulfate injection solution concentrate 5mg.kg IV q24h; amikacin sulfate injection USP 20 mg/kg IV q24hSubjects assigned to this group will receive: * IV meropenem (2 g infused over 3 hrs q 8 hr); * a parenteral aminoglycoside (tobramycin or gentamicin-5mg/kg IV Q24h or amikacin 20 mg/kg IV Q24h) * tobramycin nebulization Linezolid or vancomycin (per institutional guidelines) will be available for MRSA coverage to treat potential Gram-positive pathogens.
IV meropenem; parenteral aminoglycosidetobramycin nebulizationSubjects assigned to this group will receive: * IV meropenem (2 g infused over 3 hrs q 8 hr); * a parenteral aminoglycoside (tobramycin or gentamicin-5mg/kg IV Q24h or amikacin 20 mg/kg IV Q24h) * tobramycin nebulization Linezolid or vancomycin (per institutional guidelines) will be available for MRSA coverage to treat potential Gram-positive pathogens.
I.V. MeropenemLinezolid or Vancomycin (per institutional guidelines) will be available for MRSA coverage.Subjects assigned to this group will receive IV meropenem (2 g infused over 3 hrs q 8 hr). Linezolid or vancomycin (per institutional guidelines) will be available for MRSA coverage to treat Gram-positive pathogens. \*\*NOTE: Empiric MRSA coverage is allowed in both arms. This therapy is advised for any subjects with known or suspected MRSA entering the study. Once microbiologic results are available, this coverage may be discontinued at the investigator's discretion.
I.V. MeropenemI.V. MeropenemSubjects assigned to this group will receive IV meropenem (2 g infused over 3 hrs q 8 hr). Linezolid or vancomycin (per institutional guidelines) will be available for MRSA coverage to treat Gram-positive pathogens. \*\*NOTE: Empiric MRSA coverage is allowed in both arms. This therapy is advised for any subjects with known or suspected MRSA entering the study. Once microbiologic results are available, this coverage may be discontinued at the investigator's discretion.
Primary Outcome Measures
NameTimeMethod
Number of Participants With Suppression and Emergence of Resistanceup to 28 days after enrollment

The emergence of resistance is defined as a change of meropenem MIC or aminoglycoside MIC by two tube dilutions (fourfold) from baseline when assessed at the second BAL procedure on day 5/early extubation. Patients are evaluable for this endpoint IF they had baseline BAL and Day 5/early extubation and if they had positive cultures on baseline and Day/EE.

Secondary Outcome Measures
NameTimeMethod
Clinical ResponseEnd of treatment - up to 28 days after enrollment

Percentage of patients with successful responses by efficacy endpoint, treatment group and population (n/N)

Clinical Response in Subjects Who Received Prior AntibioticsEnd of treatment - up to 28 days after enrollment

Percentage of patients with successful responses by efficacy endpoint, treatment group and population (n/N)

Overall Microbiologic ResponseEnd of treatment - up to 28 days after enrollment

Percentage of patients with successful responses by efficacy endpoint, treatment group and population (n/N)

Pretreatment Pathogen ResponseEnd of treatment - up to 28 days after enrollment

Percentage of patients with successful responses by efficacy endpoint, treatment group and population (n/N)

Suppression of the Emergence of Resistance in Other Gram-negative PathogensDay 5/Early Extubation

Percentage of patients with successful responses by efficacy endpoint, treatment group and population (n/N)

Occurrence of Repeat Negative CulturesDay 5/Early Extubation

Percentage of patients with successful responses by efficacy endpoint, treatment group and population (n/N)

Mortality28 days

Percentage of patients who died by efficacy endpoint, treatment group and population (n/N)

Trial Locations

Locations (11)

UFL Department of Medicine: Pulmonary, Critical Care and Sleep Medicine

🇺🇸

Gainesville, Florida, United States

InClin, Inc.

🇺🇸

San Mateo, California, United States

Institut de Cardiologie, Groupe Hospitalier Pitie-Salpetriere

🇫🇷

Paris, France

Hospital Vall d'Hebron

🇪🇸

Barcelona, Spain

Northwestern University

🇺🇸

Chicago, Illinois, United States

Hannover Clinical Trial Center GmbH

🇩🇪

Hannover, Germany

Weill Cornell Medical Center of Cornell University

🇺🇸

New York, New York, United States

JMI Laboratories

🇺🇸

North Liberty, Iowa, United States

Washington University in St. Louis School of Medicine

🇺🇸

Saint Louis, Missouri, United States

Cleveland Clinic Lerner College of Medicine

🇺🇸

Cleveland, Ohio, United States

Emory University

🇺🇸

Atlanta, Georgia, United States

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