MedPath

A Study of Cariprazine in the Prevention of Relapse of Symptoms in Participants With Schizophrenia

Phase 3
Completed
Conditions
Schizophrenia
Interventions
Drug: Placebo
Drug: Cariprazine
Registration Number
NCT01412060
Lead Sponsor
Forest Laboratories
Brief Summary

The objective of this study is to evaluate the efficacy and safety of cariprazine relative to placebo in the prevention of relapse of symptoms in participants with schizophrenia.

Detailed Description

There were 3 periods (phases) in the study. The Open-label Phase lasted 20 weeks. In the first 6 weeks, participants received 3, 6, or 9 mg cariprazine orally once a day; the dose could be modified during this time. The cariprazine dose was fixed at 3, 6, or 9 mg for the last 14 weeks of this Open-label Phase. At the end of Week 8, participants had to meet the following criteria to continue in the study.

* Positive and Negative Syndrome Scale (PANSS) total score ≤ 60 at the end of Week 8

* At least 20% decrease in PANSS total score from baseline to the end of Week 8

* Clinical Global Impressions - Severity (CGI-S) score ≤ 4 at the end of Week 8

* Score of ≤ 4 on each of the following 7 PANSS items: P1, P2, P3, P6, P7, G8, and G14 at the end of Week 8

* Stable dose during the previous 2 weeks

* No significant tolerability issues as judged by the Investigator at the end of Week 8

At the end of the Open-label Phase, participants were randomized into 2 treatment groups, cariprazine or placebo, if they met the following criteria:

* PANSS total score ≤ 60 at the end of Week 20

* At least 20% decrease in PANSS total score from baseline to the end of Week 20

* CGI-S score ≤ 4 at the end of Week 20

* Score of ≤ 4 on each of the following 7 PANSS items: P1, P2, P3, P6, P7, G8, and G14 at the end of Week 20

* No significant tolerability issues as judged by the Investigator During this Double-blind Treatment Phase, participants received either placebo or cariprazine at the same dosage (3, 6, or 9 mg) that they received during the last 14 weeks of the Open-label Phase.

All participants entered the 4 week Safety Follow-up Phase. They received a treatment other than the investigational product at the discretion of the Investigator.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
765
Inclusion Criteria
  • Participants who have provided informed consent prior to any study specific procedures.
  • Participants currently meeting the Diagnostic and Statistical Manual of Mental Disorders, Fourth Edition - Text Revision (DSM-IV-TR) criteria for schizophrenia.
  • Participants with normal physical examination, laboratory, vital signs, and/or electrocardiogram (ECG).
  • Diagnosis of schizophrenia for a minimum of 1 year before Visit 1 (Screening).
  • Positive and Negative Syndrome Scale (PANSS) total score ≥ to 70 and ≤ 120 at Visit 1 (Screening) and Visit 2 (beginning of Run-in Phase).
  • Negative serum B-human chorionic gonadotropin (B-hCG) pregnancy test (applies to female participants of childbearing potential only).
  • Body mass index between 18 and 40 kg/m^2, inclusive.
Read More
Exclusion Criteria
  • Participants currently meeting DSM-IV-TR criteria for schizoaffective disorder, schizophreniform disorder, bipolar I and II and known or suspected borderline or antisocial personality disorder. or other DSM-IV-TR axis II disorders.
  • Participants in their first episode of psychosis.
  • Treatment-resistant schizophrenia over the last 2 years.
  • Positive result from the blood alcohol test or from the urine drug screen for any prohibited medication.
  • At imminent risk of injuring self or others or causing significant damage to property.
  • Suicide risk.
Read More

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Placebo - Double-blind Treatment PhasePlaceboParticipants received placebo orally once a day for 26 to 72 weeks.
Cariprazine - Open-label PhaseCariprazineParticipants received 3, 6, or 9 mg cariprazine orally once a day for 6 weeks; the dose could be modified during this time. The cariprazine dose was fixed at 3, 6, or 9 mg for the last 14 weeks of this 20 week Open-label Phase.
Cariprazine - Double-blind Treatment PhaseCariprazineParticipants received 3, 6, or 9 mg cariprazine orally once a day for 26 to 72 weeks
Primary Outcome Measures
NameTimeMethod
Time From Baseline to the First Symptom Relapse During the Double-blind PhaseUp to 34 Weeks and Bi-Weekly thereafter until Week 92

Relapse was defined as meeting ≥1 of the following criteria:1-Hospitalization due to worsening of condition;2-increase in Positive and Negative Syndrome Scale(PANSS) total score by ≥30% for participants,scored ≥50 or a ≥10-point increase for participants,scored \<50 at randomization;3-increase in Clinical Global Impressions-Severity(CGI-S) score by ≥2 points at Week 20;4-deliberate self-injury or aggressive behaviour;5-suicidal/homicidal ideation judged clinically significant by Investigator;6-score of \>4 on 1 or more of following PANSS items:P1,P2,P3,P6,P7,G8 or G14. Second assessment not performed based on Investigator discretion.

PANSS is 30-item rating scale. Each item scored on 7-point scale. Total score ranges from 30 to 210. Lower score indicates fewer schizophrenic symptoms. CGI-S is 7-point scale,measures severity of participant's illness in comparison with others with same diagnosis. Lower score indicates less severe illness. 25th percentile for time to relapse was reported.

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (73)

Forest Investigative Site 002

🇺🇸

Oceanside, California, United States

Forest Investigative Site 008

🇺🇸

Long Beach, California, United States

Forest Investigative Site 011

🇺🇸

Little Rock, Arkansas, United States

Forest Investigative Site 026

🇺🇸

Culver City, California, United States

Forest Investigative Site 018

🇺🇸

Cerritos, California, United States

Forest Investigative Site 305

🇮🇳

Vijayawada, Andhra Pradesh, India

Forest Investigative Site 001

🇺🇸

Paramount, California, United States

Forest Investigative Site 605

🇺🇦

Kharkiv, Ukraine

Forest Investigative Site 607

🇺🇦

Kherson, Ukraine

Forest Investigative Site 602

🇺🇦

Kyiv, Ukraine

Forest Investigative Site 314

🇮🇳

Manipal, Karnataka, India

Forest Investigative Site 404

🇷🇴

Targoviste, Romania

Forest Investigative Site 507

🇸🇰

Bratislava, Slovakia

Forest Investigative Site 408

🇷🇴

Bucuresti, Romania

Forest Investigative Site 410

🇷🇴

Bucuresti, Romania

Forest Investigative Site 412

🇷🇴

Campulung, Romania

Forest Investigative Site 504

🇸🇰

Liptovsky Mikulas, Slovakia

Forest Investigative Site 409

🇷🇴

Iasi, Romania

Forest Investigative Site 604

🇺🇦

Kharkiv, Ukraine

Forest Investigative Site 608

🇺🇦

Vinnytsia, Ukraine

Forest Investigative Site 503

🇸🇰

Roznava, Slovakia

Forest Investigative Site 007

🇺🇸

Costa Mesa, California, United States

Forest Investigative Site 023

🇺🇸

Baltimore, Maryland, United States

Forest Investigative Site 020

🇺🇸

San Diego, California, United States

Forest Investigative Site 017

🇺🇸

Atlanta, Georgia, United States

Forest Investigative Site 013

🇺🇸

Houston, Texas, United States

Forest Investigative Site 009

🇺🇸

Houston, Texas, United States

Forest Investigative Site 302

🇮🇳

Jaipur, Rajasthan, India

Forest Investigative Site 303

🇮🇳

Ahmedabad, Gujarat, India

Forest Investigative Site 304

🇮🇳

Lucknow, Uttar Pradesh, India

Forest Investigative Site 401

🇷🇴

Iasi, Romania

Forest Investigative Site 508

🇸🇰

Bratislava, Slovakia

Forest Investigative Site 311

🇮🇳

Nashik, Maharashtra, India

Forest Investigative Site 309

🇮🇳

Kanpur, Uttar Pradesh, India

Forest Investigative Site 317

🇮🇳

Jaipur, Rajasthan, India

Forest Investigative Site 003

🇺🇸

Flowood, Mississippi, United States

Forest Investigative Site 021

🇺🇸

Chicago, Illinois, United States

Forest Investigative Site 027

🇺🇸

Austin, Texas, United States

Forest Investigative Site 019

🇺🇸

Orange, California, United States

Forest Investigative Site 005

🇺🇸

Washington, District of Columbia, United States

Forest Investigative Site 024

🇺🇸

Leesburg, Florida, United States

Forest Investigative Site 012

🇺🇸

Cedarhurst, New York, United States

Forest Investigative Site 006

🇺🇸

Creve Coeur, Missouri, United States

Forest Investigative Site 010

🇺🇸

Rockville, Maryland, United States

Forest Investigative Site 014

🇺🇸

Saint Louis, Missouri, United States

Forest Investigative Site 022

🇺🇸

Dayton, Ohio, United States

Forest Investigative Site 025

🇺🇸

Dallas, Texas, United States

Forest Investigative Site 015

🇺🇸

Austin, Texas, United States

Forest Investigative Site 308

🇮🇳

Ahmedabad, Gujarat, India

Forest Investigative Site 310

🇮🇳

Ahmedabad, Gujarat, India

Forest Investigative Site 313

🇮🇳

Mangalore, Karnataka, India

Forest Investigative Site 306

🇮🇳

Kalyan, Maharashtra, India

Forest Investigative Site 312

🇮🇳

Madurai, Tamilnadu, India

Forest Investigative Site 405

🇷🇴

Bucuresti, Romania

Forest Investigative Site 403

🇷🇴

Bucuresti, Romania

Forest Investigative Site 406

🇷🇴

Bucuresti, Romania

Forest Investigative Site 411

🇷🇴

Focsani, Romania

Forest Investigative Site 407

🇷🇴

Campulung, Romania

Forest Investigative Site 402

🇷🇴

Constanta, Romania

Forest Investigative Site 506

🇸🇰

Trnava, Slovakia

Forest Investigative Site 613

🇺🇦

Donetsk, Ukraine

Forest Investigative Site 609

🇺🇦

Kerch, AR Crimea, Ukraine

Forest Investigative Site 610

🇺🇦

Dnipropetrovsk, Ukraine

Forest Investigative Site 616

🇺🇦

Ivano-Frankivsk, Ukraine

Forest Investigative Site 606

🇺🇦

Kharkiv, Ukraine

Forest Investigative Site 601

🇺🇦

Kyiv, Ukraine

Forest Investigative Site 603

🇺🇦

Lviv, Ukraine

Forest Investigative Site 615

🇺🇦

Odesa, Ukraine

Forest Investigative Site 611

🇺🇦

Simferopol, Ukraine

Forest Investigative Site 505

🇸🇰

Rimavska Sobota, Slovakia

Forest Investigative Site 612

🇺🇦

Kyiv, Ukraine

Forest Investigative Site 307

🇮🇳

Varanasi, Uttar Pradesh, India

Forest Investigative Site 301

🇮🇳

Aurangabad, Maharashtra, India

© Copyright 2025. All Rights Reserved by MedPath