MedPath

A Study of TAK-994 in Adults With Narcolepsy

Phase 2
Terminated
Conditions
Narcolepsy Type 1 (NT 1)
Interventions
Drug: TAK-994
Drug: Placebo
Registration Number
NCT04820842
Lead Sponsor
Takeda
Brief Summary

Adults with narcolepsy who have completed the TAK-994-1501 study will be able to take part in this study.

The main aim of this study is to check if participants have side effects from TAK-994.

Participants will take one of 3 different TAK-994 dose for 8 weeks.

Then, half the participants will continue with their dose of TAK-994 and half will take a placebo. In this study, a placebo will look like a TAK-994 tablet but will not have any medicine in it. Participants will take TAK-994 or placebo for 4 weeks.

Participants will visit the clinic for a final check-up 2 weeks after their last dose of TAK-994 or placebo.

The study doctors will check for side effects from TAK-994 and placebo throughout the study.

Participants will continue to record any narcolepsy symptoms as they did in Part B of the TAK 994-1501 study.

Detailed Description

The drug being tested in the study is called TAK-994. TAK-994, is being tested to treat participants with NT1. Participants who completed Part B of TAK-994-1501(NCT04096560) will be eligible for enrollment in this study.

This study will enroll approximately 112 patients to receive one of three different TAK 994 dose for 8 weeks (active drug extension period). Participants will be randomly assigned to one of these different TAK 994 doses which will remain undisclosed to the participant and study doctor during the study (unless there is an urgent medical need).

Following the 8-week Active Drug Extension Period, participants will continue into a 4-week Double-blind Randomized Withdrawal Period and will receive TAK-994 or Placebo.

Participants randomized to TAK-994 will continue to receive the same dose as before.

This multi-center trial will be conducted worldwide. The duration of treatment in this study is 12 weeks plus a 2 week safety follow up period. Participants will visit the clinic 10 times after the first dosing.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
26
Inclusion Criteria
  1. Participant with a diagnosis of Narcolepsy Type 1 (NT1) who has completed TAK-994-1501 Part B before enrollment (which will occur immediately following the final TAK-994-1501 assessments), and for whom the investigator has no clinical objection they be enrolled.
Read More
Exclusion Criteria
  1. Participant has a clinically significant moderate or severe ongoing AE related to the study drug from the prior study.
Read More

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Active Drug Extension Period: TAK-994 30 mgTAK-994TAK-994 30 mg, twice daily (BID) tablets, orally, from Day 1 (Day 57 of previous study) to Day 56 in the Active Drug Extension Period.
Active Drug Extension Period: TAK-994 90 mgTAK-994TAK-994 90 mg, BID, tablets, orally, from Day 1 (Day 57 of previous study) to Day 56 in the Active Drug Extension Period.
Active Drug Extension Period: TAK-994 180 mgTAK-994TAK-994 180 mg, BID, tablets, orally, from Day 1 (Day 57 of previous study) to Day 56 in the Active Drug Extension Period.
Double-blind Randomized Withdrawal Period: TAK-994 30 mgTAK-994Following the Active Drug Extension Period, participants randomized to active treatment 30 mg, BID, meeting eligibility specification and continued to receive same dose (TAK-994, 30 mg, BID, tablets, orally) from Day 57 to Day 84 in the Double-blind Randomized Withdrawal Period.
Double-blind Randomized Withdrawal Period: TAK-994 90 mgTAK-994Following the Active Drug Extension Period, participants randomized to active treatment 90 mg, BID, meeting eligibility specification and continued to receive same dose (TAK-994, 90 mg, BID, tablets, orally) from Day 57 to Day 84 in the Double-blind Randomized Withdrawal Period.
Double-blind Randomized Withdrawal Period: TAK-994 180 mgTAK-994Following the Active Drug Extension Period, participants randomized to active treatment 180 mg, BID, meeting eligibility specification and continued to receive same dose (TAK-994, 180 mg, BID, tablets, orally) from Day 57 to Day 84 in the Double-blind Randomized Withdrawal Period.
Double-blind Randomized Withdrawal Period: PlaceboPlaceboFollowing the Active Drug Extension Period participants meeting eligibility specification and received placebo-matching tablets for 4 weeks (from Day 57 to Day 84) in the Double-blind Randomized Withdrawal Period.
Primary Outcome Measures
NameTimeMethod
Number of Participants With at Least One Treatment Emergent Adverse Event (TEAE) During the Active Drug Extension PeriodUp to 8 weeks in the Active Drug Extension Period (Weeks 1 to 8)

An adverse event (AE) is defined as any untoward medical occurrence in a clinical investigation participants administered a drug; it does not necessarily have to have a causal relationship with this treatment. An AE can therefore be any unfavorable and unintended sign (example, a clinically significant abnormal laboratory finding), symptom, or disease temporally associated with the use of a drug whether or not it is considered related to the drug. A TEAE is defined as an AE with an onset that occurs after receiving study drug.

Number of Participants With at Least One Post-dose Markedly Abnormal Value (MAV) in Laboratory Test During the Active Drug Extension PeriodUp to 8 weeks in the Active Drug Extension Period (Weeks 1 to 8)

Clinical laboratory tests included hematology, serum chemistry, and urinalysis. MAV criteria: Hemoglobin \<0.8×lower limit of normal (LLN), \>1.2×upper limit of normal (ULN); Hematocrit \<0.8×LLN, \>1.2×ULN; Red blood cells (RBC) count \<0.8×LLN, \>1.2×ULN; White blood cells (WBC) count \<0.5xLLN, \>1.5xULN; Platelet count \<75x10\^9/liter (L), \>600x10\^9/L; alanine aminotransferase (ALT) \>3xULN; aspartate aminotransferase (AST) \>3xULN; gamma-glutamyl transferase (GGT) \>3xULN; Alkaline phosphatase \>3xULN; Total bilirubin \>1.5xULN; Albumin \<25 grams per liter (g/L); Total protein \<0.8xLLN, \>1.2xULN; Creatinine \>1.5xULN; Blood urea nitrogen \>40 milligrams per deciliters (mg/dL); Sodium \<130 milliequivalents per liter (mEq/L), \>150 mEq/L; Potassium \<3.0 millimoles per liter (mmol/L), \>5.3 mmol/L; creatine phosphokinase (CPK) \>3xULN; Glucose \<50 mg/dL, \>300 mg/dL; Calcium \<7.7 mg/dL, \>11.1 mg/dL. Only categories with at least one participant with event are reported.

Number of Participants With at Least One Post-dose MAV for Vital Signs During the Active Drug Extension PeriodUp to 8 weeks in the Active Drug Extension Period (Weeks 1 to 8)

MAV criteria for vital signs were: Pulse \<40 beats per minute (bpm), \>115 bpm; Systolic blood pressure \<90 millimeters of mercury (mmHg), ≥160 mmHg; Diastolic blood pressure \<50 mmHg, ≥100 mmHg, Systolic or Diastolic blood pressure change of \>20, \>30 mmHg from Baseline, Body temperature \>38.5 degree Celsius, Respiratory Rate \>21 breath/minute. Only categories with at least one participant with event are reported. Baseline for this outcome measure is Day 1 of the Active Drug Extension Period.

Number of Participants With at Least One Post-dose MAV for Electrocardiogram (ECG) Parameters During the Active Drug Extension PeriodUp to 8 weeks in the Active Drug Extension Period (Weeks 1 to 8)

MAV criteria for ECG were: Heart rate \<40 bpm, \>115 bpm; PR interval ≤80 milliseconds (msec), ≥200 msec; QT interval with Fridericia correction method (QTcF) Interval ≤300 msec, \>500 msec or ≥30 msec change from baseline and \>450 msec; QRS duration ≤80 msec, ≥180 msec. Only categories with at least one participant with event are reported.

Secondary Outcome Measures
NameTimeMethod
Number of Participants With at Least One Post-dose MAV for Vital Signs During the Double-blind Randomized Withdrawal PeriodUp to 4 weeks in the Double-blind Randomized Withdrawal Period (Weeks 9 to 12)

MAV criteria for vital signs were: Pulse \<40 bpm, \>115 bpm; Systolic blood pressure \<90 mmHg, ≥160 mmHg; Diastolic blood pressure \<50 mmHg, ≥100 mmHg, Systolic or Diastolic blood pressure change of \>20, \>30 mmHg from Baseline, Body temperature \>38.5 degree Celsius, Respiratory Rate \>21 breath/minute. Only categories with at least one participant with event are reported. Baseline for this outcome measure is Day 1 of the Double-blind Randomized Withdrawal Period (Day 57 of this study).

Number of Participants With at Least One Post-dose MAV for ECG Parameters During the Double-blind Randomized Withdrawal PeriodUp to 4 weeks in the Double-blind Randomized Withdrawal Period (Weeks 9 to 12)

MAV criteria for ECG were: Heart rate \<40 bpm, \>115 bpm; PR interval ≤80 msec, ≥200 msec; QTcF Interval ≤300 msec, \>500 msec or ≥30 msec change from baseline and \>450 msec; QRS duration ≤80 msec, ≥180 msec. Only categories with at least one participant with event are reported.

Number of Participants With at Least One TEAE During the Double-blind Randomized Withdrawal PeriodUp to 4 weeks in the Double-blind Randomized Withdrawal Period (Weeks 9 to 12)

An AE is defined as any untoward medical occurrence in a clinical investigation participants administered a drug; it does not necessarily have to have a causal relationship with this treatment. An AE can therefore be any unfavorable and unintended sign (example, a clinically significant abnormal laboratory finding), symptom, or disease temporally associated with the use of a drug whether or not it is considered related to the drug. A TEAE is defined as an AE with an onset that occurs after receiving study drug.

Number of Participants With at Least One Post-dose MAV in Laboratory Test During the Double-blind Randomized Withdrawal PeriodUp to 4 weeks in the Double-blind Randomized Withdrawal Period (Weeks 9 to 12)

Clinical laboratory tests included hematology, serum chemistry, and urinalysis. MAV criteria: Hemoglobin \<0.8×LLN, \>1.2×ULN; Hematocrit \<0.8×LLN, \>1.2×ULN; RBC count \<0.8×LLN, \>1.2×ULN; WBC count \<0.5xLLN, \>1.5xULN; Platelet count \<75x10\^9/L, \>600x10\^9/L; ALT \>3xULN; AST \>3xULN; GGT \>3xULN; Alkaline phosphatase \>3xULN; Total bilirubin \>1.5xULN; Albumin \<25 g/L; Total protein \<0.8x LLN, \>1.2xULN; Creatinine \>1.5xULN; Blood urea nitrogen \>40 mg/dL; Sodium \<130 mEq/L, \>150 mEq/L; Potassium \<3.0 mmol/L, \>5.3 mmol/L; CPK \>3xULN; Glucose \<50 mg/dL, \>300 mg/dL; Calcium \<7.7 mg/dL, \>11.1 mg/dL.

Trial Locations

Locations (70)

Raleigh Neurology Associates,300209729

🇺🇸

Raleigh, North Carolina, United States

Fort Wayne Neurological Center 150711262

🇺🇸

Fort Wayne, Indiana, United States

Turku University Hospital

🇫🇮

Turku, Finland

SomnoCenter Budapest

🇭🇺

Budapest, Hungary

Sleep Medicine Specialists of South Florida

🇺🇸

Miami, Florida, United States

Clinical Site Partners, LLC

🇺🇸

Miami, Florida, United States

NeuroTrials Research, Inc. 300116336

🇺🇸

Atlanta, Georgia, United States

Beth Israel Deaconess Medical Center CardioVascular Institute

🇺🇸

Boston, Massachusetts, United States

The Cleveland Clinic Foundation 100428

🇺🇸

Cleveland, Ohio, United States

Pacific Research Network, Inc 150118105

🇺🇸

San Diego, California, United States

Intrepid Research

🇺🇸

Cincinnati, Ohio, United States

Stanford School of Medicine

🇺🇸

Redwood City, California, United States

Delta Waves Sleep Disorders and Research Center 300148510

🇺🇸

Colorado Springs, Colorado, United States

CITrials - Bellflower

🇺🇸

Bellflower, California, United States

Toronto Sleep Institute

🇨🇦

Toronto, Ontario, Canada

SDS Clinical Trials, Inc.

🇺🇸

Santa Ana, California, United States

Jodha Tishon Inc.

🇨🇦

Toronto, Ontario, Canada

Kurume University Hospital Dept of Neuropsychiatry

🇯🇵

Kurume-shi, Fukuoka-Ken, Japan

Santa Monica Clinical Trials

🇺🇸

Los Angeles, California, United States

Comprehensive Sleep Medicine Associates

🇺🇸

Sugar Land, Texas, United States

CTI Clinical Research Center

🇺🇸

Cincinnati, Ohio, United States

Koishikawa Tokyo Hospital Dept of Psychiatry

🇯🇵

Bunkyo-ku, Tokyo-To, Japan

The Catholic University of Korea, St. Vincent's Hospital 300187879

🇰🇷

Suwon-si, Gyeonggi-do, Korea, Republic of

West Ottawa Sleep Centre

🇨🇦

Ottawa, Ontario, Canada

Bogan Sleep Consultants, LLC 150711087

🇺🇸

Columbia, South Carolina, United States

Hospital General de Castellon Servicio de Neurofisiologia

🇪🇸

Castellon de la Plana, Castellon, Spain

Hospital Clinic de Barcelona Servicio de Neurologia

🇪🇸

Barcelona, Spain

Hospital Vithas Nuestra Senora de America Neurofisiologia Clinica

🇪🇸

Madrid, Spain

Gokeikai Osaka Kaisei Hospital Dept of Sleep Medicine

🇯🇵

Osaka-shi, Osaka-Fu, Japan

Hospital Universitario Araba Sede Santiago Sleep Unit

🇪🇸

Vitoria, Alava, Spain

Yoyogi Sleep Disorder Center Dept of Psychiatry

🇯🇵

Shibuya-ku, Tokyo-To, Japan

Sumida Hospital Phase I

🇯🇵

Sumida-ku, Tokyo-To, Japan

Jinyukai Kotorii Isahaya Hospital Dept of Psychiatry

🇯🇵

Isahaya-shi, Nagasaki-Ken, Japan

Shunkaikai Inoue Hospital Dept of Respiratory Medicine

🇯🇵

Nagasaki-shi, Nagasaki-Ken, Japan

Mayo Clinic Arizona 300151190

🇺🇸

Phoenix, Arizona, United States

Sleep Therapy & Research Center 300151246

🇺🇸

San Antonio, Texas, United States

JSV Clinical Research Study, Inc

🇺🇸

Tampa, Florida, United States

Wright Clinical Research

🇺🇸

Alabaster, Alabama, United States

Alpine Clinical Research Center 1024762

🇺🇸

Boulder, Colorado, United States

Florida Pulmonary Research Institute, LLC 300127039

🇺🇸

Winter Park, Florida, United States

Clinical Research Institute 300169881

🇺🇸

Stockbridge, Georgia, United States

Sleep Practitioners, LLC Macon

🇺🇸

Macon, Georgia, United States

Clinical Research of Gastonia

🇺🇸

Gastonia, North Carolina, United States

University of Kansas Medical Center Research Institute, Inc. University of Kansas Hospital

🇺🇸

Kansas City, Kansas, United States

Helene A. Emsellem, MD PC trading as "The Center for Sleep & Wake Disorders" 150119420

🇺🇸

Chevy Chase, Maryland, United States

Raleigh Neurology Associates 300209729

🇺🇸

Raleigh, North Carolina, United States

Respiratory Specialists Berks Schuylkill Respiratory Specialists Ltd

🇺🇸

Wyomissing, Pennsylvania, United States

Terveystalo Helsinki Uniklinikka 300186257

🇫🇮

Helsinki, Finland

Fakultni nemocnice Hradec Kralove Dept of Neurologicka klinika

🇨🇿

Hradec Kralove, Czechia

Universita di Bologna-Clinica Neurologica-Dipartimento di Scienze Neurologiche

🇮🇹

Bologna, Italy

Hopital Gui de Chauliac Service de Neurologie

🇫🇷

Montpellier, Herault, France

Vseobecna fakultni nemocnice v Praze Dept of Neurologicka klinika 1.LF UK a VFN v Praze

🇨🇿

Praha 2, Czechia

Azienda Ospedaliera Universitaria Policlinico Tor Vergata U.O.C. Neurologia

🇮🇹

Roma, Italy

Ospedale San Raffaele (San Raffaele Turro) Clinica Neurologica- Div Malattie del Sonno

🇮🇹

Milano, Italy

SOUSEIKAI PS Clinic Dept of Internal Medicine

🇯🇵

Fukuoka-shi, Fukuoka-Ken, Japan

Howakai Kuwamizu Hospital Dept of Internal Medicine

🇯🇵

Kumamoto-shi, Kumamoto-Ken, Japan

You Ariyoshi Sleep Clinic Dept of Psychiatry

🇯🇵

Kitakyushu-shi, Fukuoka-Ken, Japan

Kaiseikai Kita Shin Yokohama Internal Medicine Clinic Dept of Internal Medicine

🇯🇵

Yokohama-shi, Kanagawa-Ken, Japan

Kyowakai Hannan Hospital Dept of Psychiatry

🇯🇵

Sakai-shi, Osaka-Fu, Japan

Nihon University Itabashi Hospital Dept of Neuropsychiatry

🇯🇵

Itabashi-ku, Tokyo-To, Japan

Keimyung University Dongsan Hospital 300144594

🇰🇷

Daegu, Korea, Republic of

Research Carolina Elite

🇺🇸

Denver, North Carolina, United States

St. Francis Medical Institute

🇺🇸

Clearwater, Florida, United States

Hawaii Pacific Neuroscience

🇺🇸

Honolulu, Hawaii, United States

Ohio Sleep Medicine and Neuroscience Institute 186

🇺🇸

Dublin, Ohio, United States

Sleep & Stress Clinic Dept of Psychiatry

🇯🇵

Shinagawa-ku, Tokyo-To, Japan

Sleep Support Clinic Dept of Psychosomatic Medicine/Psychiatry

🇯🇵

Shinagawa-ku, Tokyo-To, Japan

Medical University of South Carolina (MUSC) PARENT

🇺🇸

Charleston, South Carolina, United States

IRCCS Oasi Maria SS 300206751

🇮🇹

Troina, Enna, Italy

Hopital Roger Salengro - CHU Lille service de neurologie D

🇫🇷

Lille Cedex, Nord, France

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