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An Efficacy and Safety Study in Children 6 to Less Than 18 Years of Age With Hypertension

Phase 3
Completed
Conditions
Hypertension
Interventions
Drug: Azilsartan Medoxomil High-dose (40 mg)
Drug: Azilsartan Medoxomil Medium-dose (20 mg)
Registration Number
NCT02235909
Lead Sponsor
Arbor Pharmaceuticals, Inc.
Brief Summary

The purpose of the study is to evaluate the efficacy and safety of the study drug relative to an active comparator losartan which is in the same class of drug and is approved for use in the pediatric population aged 6 years and older. Approximately 260 subjects will participate in a 6-week, double-blind, randomized, treatment phase, followed by a 2-week, double-blind, randomized, placebo-controlled withdrawal phase. A 44-week, open-label extension in which all subjects will receive azilsartan and other antihypertensive medications (if needed). Blood pressure will be assessed throughout the study.

Detailed Description

The purpose of the study is to evaluate the efficacy and safety of the study drug relative to an active comparator losartan which the same class of drug and is approved for use in the pediatric population aged 6 years and older. Approximately 260 subjects will participate in a 6-week, double-blind, randomized, treatment phase, followed by a 2-week, double-blind, randomized, placebo-controlled withdrawal phase. This study also includes a 44-week, open-label extension Phase in which all subjects will receive azilsartan and other antihypertensive medications (if needed) in order to reach an optimal blood pressure. Blood pressure will be assessed in the clinic throughout the study, and subjects may also participate in a 24-hour ambulatory blood pressure monitoring procedure at baseline, at the end of the double-blind Phase and at the end of the open-label Phase.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
377
Inclusion Criteria
  • The subject has hypertension (primary or secondary) defined as clinic Seated Diastolic BP ≥95th percentile (by age, gender, and height) or ≥90th percentile (by age, gender, height) if chronic renal disease, diabetes, heart failure or hypertensive target organ damage is present

    1. If currently treated: The subject has a documented historical diagnosis of hypertension AND a post-washout clinic Seated Diastolic BP meeting the above criteria on Day -1 (or Day 1 for subjects not participating in Ambulatory Blood Pressure Monitoring)
    2. If currently untreated: The subject has elevated Seated Diastolic BP meeting the above criteria on 3 separate occasions before Randomization, including on Day -1 (or Day 1 for subjects not participating in Ambulatory Blood Pressure Monitoring)
  • The subject is male or female and aged 6 to <18 years at Baseline and weighs at least 25 kg

  • The subject agrees to continue their previously implemented nonpharmacological life style modifications if begun prior to Screening. Note: For subjects participating in a weight loss program, the weight maintenance

Exclusion Criteria
  • The subject has a clinic Seated Diastolic BP greater than 15 mm Hg and/or Seated Diastolic BP greater than 10 mm Hg above the 99th percentile for age, gender, and height as confirmed by the average (arithmetic mean) of 3 serial clinic seated BP measurements at Screening/Visit 1
  • The subject has a diagnosis of malignant or accelerated hypertension
  • The subject is currently treated with more than 2 antihypertensive agents
  • The subject or parent/legal guardian is not willing for the subject's previous antihypertensive medications to be stopped
  • The subject has participated in the intensive, active weight-loss phase of a weight-loss program within 30 days prior to Screening/Visit 1
  • The subject has any of the following: severe renal impairment (eGFR <30 mL/min/1.73 m2 by the Schwartz formula); is currently undergoing dialysis treatment; renovascular disease affecting both kidneys or a solitary kidney; severe nephrotic syndrome not in remission; or serum albumin <2.5 g/dL
  • The subject has a history or clinical manifestations of severe cardiovascular, hepato-biliary, gastrointestinal, endocrine-metabolic (e.g., hyperthyroidism, Cushing's syndrome), hematologic, immunologic, genito-urinary, or psychiatric disease, cancer, and/or any conditions that would interfere with the health status of the subject through study participation, or would jeopardize study integrity in the opinion of the investigator
  • The subject is suffering from uncorrected coarctation of the aorta, or hemodynamically significant left ventricular outflow tract obstruction due to eg, aortic valvular disease, or is likely to undergo a procedure known to affect blood pressure (eg, repair of arterial anomalies) during the course of the study
  • The subject is poorly controlled diabetic defined as having a glycosylated hemoglobin value >8.5% at Screening/Visit 1
  • The subject has hyperkalemia as defined by the central laboratory's normal reference range or any pertinent electrolyte disorders at Screening/Visit

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Double-blind: Azilsartan Medoxomil - Low doseAzilsartan Medoxomil Low-dose6-week, double-blind (DB), randomized, treatment phase (DB Phase): Azilsartan medoxomil low-dose (AZM-L), 10 mg once daily.
Double blind phase: LosartanLosartan6-week, double-blind (DB), randomized, treatment phase (DB Phase): Starting at Losartan 25/50 and force titrated to 50/100 mg daily at Week 2.
Withdrawal Phase: Azilsartan medoxomil low-dose (AZM-L)Azilsartan Medoxomil Low-doseExperimental Arm in the Withdrawal Phase, subjects will be randomized (1:1) to continue taking their previously assigned active treatment (AZM-L) that was taken in Double blind OR to be switched to placebo.
Withdrawal Phase: Placebo to match azilsartan medoxomil low dose (AZM-L)LosartanPlacebo Arm in the Withdrawal Phase for subjects who were on AZM-L in double blind then randomized (1:1) to placebo for withdrawal phase
Open Label Phase: Azilsartan MedoxomilAzilsartan Medoxomil Low-doseAzilsartan Medoxomil 10 mg which can be titrated to higher dose(s) (up to 40 mg for subjects \<50 kg or up to 80 mg for subjects ≥50 kg)
Withdrawal Phase: Losartan 50 mgLosartanWithdrawal Phase, subjects will be randomized (1:1) to continue taking their previously assigned active treatment or to be switched to placebo.
Withdrawal Phase: Placebo to LosartanPlacebo for LosartanPlacebo Arm In the Withdrawal Phase, subjects will be randomized (1:1) to continue taking their previously assigned active treatment or to be switched to placebo.
Double-blind: Azilsartan Medoxomil - Medium doseAzilsartan Medoxomil Low-dose6-week, double-blind (DB), randomized, treatment phase (DB Phase), Azilsartan medoxomil Medium-dose (AZM-M), 20 mg once daily at Week 2.
Double-blind: Azilsartan Medoxomil - Medium dosePlacebo for Losartan6-week, double-blind (DB), randomized, treatment phase (DB Phase), Azilsartan medoxomil Medium-dose (AZM-M), 20 mg once daily at Week 2.
Double-blind: Azilsartan Medoxomil - Medium doseAzilsartan Medoxomil Medium-dose (20 mg)6-week, double-blind (DB), randomized, treatment phase (DB Phase), Azilsartan medoxomil Medium-dose (AZM-M), 20 mg once daily at Week 2.
Double-blind: Azilsartan Medoxomil - High dose (AZM-H)Azilsartan Medoxomil High-dose (40 mg)6-week, double-blind (DB), randomized, treatment phase (DB Phase): Azilsartan medoxomil High-dose (AZM-H), 40 mg AZM-M
Withdrawal: Azilsartan Medoxomil - Medium doseAzilsartan Medoxomil Low-doseExperimental Arm in the Withdrawal Phase, subjects will be randomized (1:1) to continue taking their previously assigned active treatment (AZM-M) that was taken in Double blind OR to be switched to placebo.
Withdrawal: Azilsartan Medoxomil - Medium doseAzilsartan Medoxomil Medium-dose (20 mg)Experimental Arm in the Withdrawal Phase, subjects will be randomized (1:1) to continue taking their previously assigned active treatment (AZM-M) that was taken in Double blind OR to be switched to placebo.
Withdrawal: Azilsartan Medoxomil - High doseAzilsartan Medoxomil High-dose (40 mg)Experimental Arm in the Withdrawal Phase, subjects will be randomized (1:1) to continue taking their previously assigned active treatment (AZM-H) that was taken in double blind OR to be switched to placebo.
Withdrawal Phase: Placebo to match azilsartan medoxomil medium dose (AZM-M)Placebo for Azilsartan MedoxomilPlacebo arm in the Withdrawal Phase for subjects who were on AZM-M in double blind then randomized (1:1) to matching placebo for withdrawal phase
Withdrawal Phase: Placebo to match azilsartan medoxomil high dose (AZM-H)Placebo for Azilsartan MedoxomilPlacebo arm in the Withdrawal Phase for subjects who were on AZM-H in Double blind then randomized (1:1) to matching placebo for withdrawal phase
Primary Outcome Measures
NameTimeMethod
Change in Seated Diastolic Blood Pressure Between AZM and PlaceboFrom Week 6/Final Visit of DB Phase to Week 8/Final Visit of Withdrawal Phase

Change in Seated Diastolic Blood Pressure from Week 6/Final visit of DB Phase to Week 8/Final Visit of the Withdrawal Phase, analysis of study subjects randomized to receiving placebo at Week 6 of treatment versus those who remained on treatment

Secondary Outcome Measures
NameTimeMethod
Change in Trough Seated Systolic Blood PressureFrom Week 6/Final Visit of the Double-Blind Phase to Week 8/Final Visit of the Withdrawal Phase

Change in Trough Seated Systolic Blood Pressure from Week 6 of the Double-Blind Phase to Week 8 of the Withdrawal Phase Between AZM and Placebo, analysis of study subjects randomized to receiving placebo at Week 6 of treatment versus those who remained on treatment

Change in Mean Arterial PressureFrom Week 6 of the Double-Blind Phase to Week 8 of the Withdrawal Phase

Change in Mean Arterial Pressure from Week 6 of the Double-Blind Phase to Week 8 of the Withdrawal Phase Between AZM and Placebo, analysis of study subjects randomized to receiving placebo at Week 6 of treatment versus those who remained on treatment

Trial Locations

Locations (69)

Advanced Research Center, INC

🇺🇸

Anaheim, California, United States

Direct Helpers Research Center

🇺🇸

Hialeah, Florida, United States

JDH Medical Group LLC

🇺🇸

Miami, Florida, United States

University of Miami/Jackson Memorial Hospital

🇺🇸

Miami, Florida, United States

Medical Research Center of Miami II, Inc.

🇺🇸

Miami, Florida, United States

Pioneer Clinical Research

🇺🇸

North Miami, Florida, United States

Georgia Clinical Research

🇺🇸

Snellville, Georgia, United States

Zoe Center for Pediatrics

🇺🇸

Thomaston, Georgia, United States

University of Louisville

🇺🇸

Louisville, Kentucky, United States

David M. Headley, MD PA

🇺🇸

Port Gibson, Mississippi, United States

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Advanced Research Center, INC
🇺🇸Anaheim, California, United States

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