MedPath

Efficacy and Safety of Atacicept in Systemic Lupus Erythematosus

Phase 2
Completed
Conditions
Lupus Erythematosus, Systemic
Interventions
Registration Number
NCT01972568
Lead Sponsor
EMD Serono
Brief Summary

This is a multi-center, double-blind, randomized, Phase 2b trial to evaluate the efficacy of atacicept in subjects with systemic lupus erythematosus (SLE).

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
306
Inclusion Criteria
  • Eligible male and female subjects, aged 18 years or older
  • Must have at least moderately active SLE, as defined as SLE Disease Activity Index-2000 (SLEDAI-2K) score greater than or equal to [>=] 6 at screening visit
  • At least 4 of the 11 American college of rheumatology (ACR) classification criteria for SLE (diagnosed >= 6 months prior to the screening visit)
  • Be seropositive for anti-nuclear antibodies (ANA) and/or anti-double-stranded deoxyribonucleic acid (anti-dsDNA) antibodies
  • Other protocol defined inclusion criteria could apply
Exclusion Criteria
  • Subjects have demyelinating disorder
  • Severe central nervous system SLE
  • Use of cyclophosphamide within 3 months of the screening visit
  • Urine protein:creatinine ratio (UPCr) >= 2 milligram per milligram (mg/mg) per day
  • Other protocol defined exclusion criteria could apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Atacicept 75 mgAtacicept 75 milligram (mg)-
PlaceboPlacebo-
Atacicept 150 mgAtacicept 150 mg-
Primary Outcome Measures
NameTimeMethod
Percentage of Subjects With Systemic Lupus Erythematosus (SLE) Responder Index (SRI) Response at Week 24 Using Screening Visit as BaselineWeek 24

SRI response, a composite measure of reduced SLE disease activity, was defined as a reduction in Systemic Lupus Erythematosus Disease Activity Index 2000 (SLEDAI-2K) disease activity score of greater than or equal to (\>=) 4 points; no significant worsening in Physician's Global Assessment (PGA) score (\<10 % increase, defined as \<0.3 point increase for statistical analyses); no new British Isles Lupus Assessment Group (BILAG) A organ domain scores and \<=1 (defined as no more than one) new BILAG B organ domain score.

Percentage of Subjects With Systemic Lupus Erythematosus (SLE) Responder Index (SRI) Response at Week 24 Using Day 1 as BaselineWeek 24

SRI response, a composite measure of reduced SLE disease activity, was defined as a reduction in Systemic Lupus Erythematosus Disease Activity Index 2000 (SLEDAI-2K) disease activity score of greater than or equal to (\>=) 4 points; no significant worsening in Physician's Global Assessment (PGA) score (\<10 % increase, defined as \<0.3 point increase for statistical analyses); no new British Isles Lupus Assessment Group (BILAG) A organ domain scores and \<=1 (defined as no more than one) new BILAG B organ domain score.

Secondary Outcome Measures
NameTimeMethod
Change From Screening in Prednisolone-Equivalent Corticosteroid (CS) Daily Dose at Week 24Screening and Week 24

Change From screening visit to Week 24 of prednisolone-equivalent CS daily dose was presented.

Percentage of Subjects at Week 24 Whose Prednisone-Equivalent Corticosteroid (CS) Dose Reduced From Screening by >=25% and to a Dose of =<7.5mg/Day, and no British Isles Lupus Assessment Group (BILAG) A or 2B Flare in Disease ActivityWeek 24

BILAG A or 2B flare is defined by 1 new BILAG A organ domain score and/or 2 new BILAG B organ domain scores compared to the Screening Visit. The BILAG disease activity index evaluates systemic lupus erythematosus (SLE) activity in 8 organ systems, using a separate alphabetic score (A to E) assigned to each organ system defined as follows. BILAG A: Disease sufficiently active requiring disease-modifying treatment (prednisone \>20 mg daily or immunosuppressants); BILAG B: moderate disease activity requiring treatment with systemic low-dose oral glucocorticoids, intramuscular or intra-articular or soft tissue CS injection, topical CS or immunosuppressants, or symptomatic therapy such as antimalarials or NSAIDs. BILAG C: mild disease; BILAG D: system previously affected but now inactive and BILAG E: system never involved.

Percentage of Subjects With Patient Global Impression of Change (PGIC) Categories at Week 24Week 24

The PGIC is self-rated scale that asks the subject to describe the change in activity limitations, symptoms, emotions, and overall Quality of life (QoL) related to the subject's painful condition on the following scale: 1 (very much improved), 2 (much improved), 3 (minimally improved), 4 (no change), 5 (minimally worse), 6 (much worse) and 7 (very much worse). Percentage of subjects in the PGIC categories of very much or much improved (1 or 2), minimally improved or no change or minimally worse (3 or 4 or 5) and much or very much worse (6 or 7) at Week 24 were presented.

Percentage of Subjects With Treatment-Emergent Adverse Events (TEAEs) and Serious TEAEsBaseline up to 24 weeks after last dose of study drug (assessed up to maximum of 48 weeks)

An AE was defined as any unfavourable and unintended sign (including an abnormal laboratory finding), symptom, or disease temporally associated with the use of study drug, whether or not considered related to the study drug. A serious AE was an AE that resulted in any of the following outcomes: death; life threatening; persistent/significant disability/incapacity; initial or prolonged inpatient hospitalization; congenital anomaly/birth defect or was otherwise considered medically important. Treatment-emergent are events between first dose of study drug and up to 48 weeks. TEAEs include both Serious TEAEs and non-serious TEAEs.

Time From Randomization to First SRI Response During Treatment PeriodBaseline up to 24 Weeks

SRI response, a composite measure of reduced SLE disease activity, was defined as a reduction in Systemic Lupus Erythematosus Disease Activity Index 2000 (SLEDAI-2K) disease activity score of greater than or equal to (\>=) 4 points; no significant worsening in Physician's Global Assessment (PGA) score (\<10 % increase, defined as \<0.3 point increase for statistical analyses); no new British Isles Lupus Assessment Group (BILAG) A organ domain scores and \<=1 (defined as no more than one) new BILAG B organ domain score. Time to first SRI response during treatment period was presented.

Percentage of Subjects With British Isles Lupus Assessment Group (BILAG)-Based Combined Lupus Assessment (BICLA) Response at Week 24Week 24

The BICLA response is defined as BILAG-2004 improvement (all screening visit BILAG A improving to B/C/D, all screening visit BILAG B to C/D, and \<=1 new BILAG B and no new BILAG A); no deterioration in SLEDAI total score; PGA increase by \<10% (defined as \<0.3 point increase for the statistical analyses) and no nonpermitted medication/treatment.

Change From Week 0 (Day 1) in SF-36 Components at Week 24Week 0 (Day 1) and Week 24

The 36-Item Short-Form Health Survey (SF-36) is a standardized survey evaluating 8 aspects of functional health and well being: physical and social functioning, physical and emotional role limitations, bodily pain, general health, vitality, mental health. These 8 aspects can also be summarized as physical and mental component summary scores. Total of 10 variables were analyzed (8 aspects, 2 component summary scores). The score for each of the 8 aspects and 2 component summary scores was scaled from 0 to 100, where 0 = lowest level of functioning and 100 = highest level of functioning.

Trial Locations

Locations (137)

Mayo Clinic

🇺🇸

Rochester, Minnesota, United States

Atencion Integral en Reumatologia (AIR)

🇦🇷

Ciudad Autonoma Buenos Aires, Argentina

Organizacion Medica de Investigacion (OMI)

🇦🇷

Ciudad Autonoma Buenos Aires, Argentina

Cordis S.A.

🇦🇷

Salta, Argentina

Hospital Italiano

🇦🇷

Ciudad Autonoma Buenos Aires, Argentina

Centro Polivalente de Asistencia e Inv. Clinica CER

🇦🇷

San Juan, Argentina

Investigaciones Clinicas Tucuman

🇦🇷

San Miguel de Tucuman, Argentina

Centro Integral de Reumatologia

🇦🇷

San Miguel de Tucumán, Argentina

Policlìnica Red Omip S.A - Ensayos Clinicos GC

🇦🇷

Mar De Plata, Argentina

Centro de Investigacion Pergamino SA

🇦🇷

Pergamino, Argentina

MHAT "Eurohospital" - Plovdiv, OOD

🇧🇬

Plovdiv, Bulgaria

Medical Center "Teodora", EOOD

🇧🇬

Ruse, Bulgaria

Biomedica

🇨🇱

Santiago, Chile

DCC "Sveta Anna", EOOD

🇧🇬

Sofia, Bulgaria

Medical Center "Nov Rehabilitatsionen Tsentar", EOOD

🇧🇬

Stara Zagora, Bulgaria

National Center for Global Health and Medicine Hospital

🇯🇵

Shinjuku, Japan

Investigacion y Biomedicina de Chihuahua, S.C.

🇲🇽

Chihuahua, Mexico

Accelerium S. de R.L. de C.V.

🇲🇽

Monterrey, Mexico

Tohoku University Hospital

🇯🇵

Sendai-shi, Japan

Yuaikai Tomishiro Chuo Hospital

🇯🇵

Tomigusuku-shi, Japan

Morales Vargas Centro de Investigacion, S.C.

🇲🇽

Leon, Mexico

Clinica Vesalio

🇵🇪

Lima, Peru

HMA - Hospital Maria Auxiliadora

🇵🇪

Lima, Peru

Mary Mediatrix Medical Center

🇵🇭

Batangas, Philippines

Southern California Permanente Medical Group

🇺🇸

Anaheim, California, United States

Center for Rheumatology, Immunology & Arthritis

🇺🇸

Fort Lauderdale, Florida, United States

The Feinstein Institute for Medical Research

🇺🇸

Manhasset, New York, United States

Rutgers New Jersey Medical School

🇺🇸

Newark, New Jersey, United States

Charite Universitaetsmedizin Berlin - Campus Charite Mitte

🇩🇪

Berlin, Germany

Clínica de Neoplasias Litoral Ltda.

🇧🇷

Santa Catarina, Brazil

Box Arthritis & Rheumatology of the Carolinas PLLC

🇺🇸

Charlotte, North Carolina, United States

Clinical Research of West Florida - Corporate

🇺🇸

Dunedin, Florida, United States

APRILLUS

🇦🇷

Ciudad Autonoma Buenos aires, Argentina

UMHAT "Sv. Ivan Rilski", EAD

🇧🇬

Sofia, Bulgaria

STAT Research, Inc.

🇺🇸

Dayton, Ohio, United States

Danville Orthopedic Clinic, Inc.

🇺🇸

Danville, Virginia, United States

Fundação Faculdade Regional de Medicina de São José do Rio Preto

🇧🇷

São José do Rio Preto, Brazil

CPD - Centro de Pesquisas em Diabetes

🇧🇷

Porto Alegre, Brazil

Washington University School of Medicine

🇺🇸

Saint Louis, Missouri, United States

A-Shine, s.r.o.

🇨🇿

Plzen, Czechia

Revmatologicky Ustav

🇨🇿

Praha 2, Czechia

Rheumazentrum Ruhrgebiet

🇩🇪

Herne, Germany

Royal Sussex County Hospital

🇬🇧

Brighton, United Kingdom

Royal National Hospital for Rheumatic Diseases

🇬🇧

Bath, United Kingdom

Azienda Ospedaliero-Universitaria Consorziale Pol. di Bari

🇮🇹

Bari, Italy

Kyung Hee University Hospital

🇰🇷

Seoul, Korea, Republic of

University Hospital Coventry

🇬🇧

Coventry, United Kingdom

University College London Hospitals

🇬🇧

London, United Kingdom

Wrightington Hospital

🇬🇧

Wigan, United Kingdom

Hospital Clínico Universitario de Valladolid

🇪🇸

Valladolid, Spain

East Bay Rheumatology Medical Group, Inc.

🇺🇸

San Leandro, California, United States

Goldpoint Clinical Research, LLC

🇺🇸

Indianapolis, Indiana, United States

Achieve Clinical Research, LLC

🇺🇸

Birmingham, Alabama, United States

Arthritis & Rheumatology Center of Oklahoma

🇺🇸

Oklahoma City, Oklahoma, United States

OMRF

🇺🇸

Oklahoma City, Oklahoma, United States

University of Alabama at Birmingham - (UAB)

🇺🇸

Birmingham, Alabama, United States

Gachon University Gil Medical Center

🇰🇷

Incheon, Korea, Republic of

Konkuk University Medical Center

🇰🇷

Seoul, Korea, Republic of

Ajou University Hospital

🇰🇷

Suwon-si, Korea, Republic of

Wallace Rheumatic Study Center

🇺🇸

Los Angeles, California, United States

Ohio State University Medical Center

🇺🇸

Columbus, Ohio, United States

University of Miami Miller School of Medicine

🇺🇸

Miami, Florida, United States

AA MRC LLC Ahmed Arif Medical Research Center

🇺🇸

Grand Blanc, Michigan, United States

Clinical Research Center of Reading LLC

🇺🇸

Wyomissing, Pennsylvania, United States

UTMB Pathology Clinical Services

🇺🇸

Galveston, Texas, United States

Arthritis & Osteoporosis Clinic

🇺🇸

Waco, Texas, United States

Tsukuba University Hospital

🇯🇵

Tsukuba-shi, Japan

Unidad de Investigacion en Enfermedades Cronico Degenerativas SC

🇲🇽

Guadalajara, Mexico

Pinnacle Research Group LLC

🇺🇸

Anniston, Alabama, United States

Clinical Research of West Florida, Inc.

🇺🇸

Tampa, Florida, United States

North MS Medical Clinics, Inc.

🇺🇸

Tupelo, Mississippi, United States

Hospital for Special Surgery

🇺🇸

New York, New York, United States

MetroHealth System

🇺🇸

Cleveland, Ohio, United States

Lynn Health Science Institute

🇺🇸

Oklahoma City, Oklahoma, United States

Medical University of South Carolina (MUSC)

🇺🇸

Charleston, South Carolina, United States

Centro Medico Privado de Reumatologia

🇦🇷

San Miguel de Tucuman, Argentina

CLION - Clínica de Oncologia da Bahia

🇧🇷

Salvador, Brazil

MHAT-Targovishte, AD

🇧🇬

Targovishte, Bulgaria

Centro de Estudios Reumatologicos

🇨🇱

Santiago, Chile

Centro Medico Prosalud

🇨🇱

Santiago, Chile

SOMEAL

🇨🇱

Santiago, Chile

CINVEC - Centro de Investigacion Clinica V Region

🇨🇱

Vina del Mar, Chile

MEDICAL PLUS s.r.o.

🇨🇿

Uherske Hradiste, Czechia

Kerckhoff-Klinik gGmbH

🇩🇪

Bad Nauheim, Germany

Vseobecna fakultni nemocnice v Praze

🇨🇿

Praha 2, Czechia

Klinikum der Johann Wolfgang Goethe-Universitaet

🇩🇪

Frankfurt, Germany

Universitaetsklinikum Freiburg

🇩🇪

Freiburg, Germany

Presidio Ospedaliero Vittorio Emanuele

🇮🇹

Catania, Italy

Universitaetsklinikum Schleswig-Holstein - Campus Kiel

🇩🇪

Kiel, Germany

Universitaetsmedizin der Johannes Gutenberg-Universitaet Mainz

🇩🇪

Mainz, Germany

Azienda Ospedaliero Universitaria San Martino

🇮🇹

Genova, Italy

Azienda Ospedaliera Universitaria Careggi

🇮🇹

Firenze, Italy

Fondazione IRCCS Policlinico San Matteo

🇮🇹

Pavia, Italy

Fondazione IRCCS Ca' Granda Ospedale Maggiore Policlinico

🇮🇹

Milano, Italy

St. Luke's International Hospital

🇯🇵

Chuo-ku, Japan

NHO Kyushu Medical Center

🇯🇵

Fukuoka-shi, Japan

Toho University Ohashi Medical Center

🇯🇵

Meguro-ku, Japan

Okayama University Hospital

🇯🇵

Okayama-shi, Japan

Kitasato University Hospital

🇯🇵

Sagamihara-shi, Japan

Hokkaido University Hospital

🇯🇵

Sapporo-shi, Japan

Sapporo City General Hospital

🇯🇵

Sapporo-shi, Japan

Hakujujikai Sasebochuo Hospital

🇯🇵

Sasebo-shi, Japan

Jichi Medical University Hospital

🇯🇵

Shimotsuke-shi, Japan

Icle S.C.

🇲🇽

Guadalajara, Mexico

Investigacion Clinica de Leon S.C.

🇲🇽

Leon, Mexico

Centro de Estudios Clinicos Especializados

🇲🇽

Merida, Mexico

Clinica de Enfermedades Cronicas y de Procedimientos Especiales, S.C.

🇲🇽

Morelia, Mexico

Hospital Universitario de Saltillo "Dr. Gonzalo Valdés Valdés"

🇲🇽

Saltillo, Mexico

ALIVIA Clínica de Alta Especialidad S.A. de C.V.

🇲🇽

Monterrey, Mexico

Clinica El Golf

🇵🇪

Lima, Peru

Clinica Medica Cayetano Heredia

🇵🇪

Lima, Peru

Angeles University Foundation Medical Center

🇵🇭

Angeles City, Philippines

Iloilo Doctors Hospital

🇵🇭

Iloilo City, Philippines

Davao Doctors Hospital

🇵🇭

Davao City, Philippines

St. Luke's Medical Center

🇵🇭

Quezon City, Philippines

Szpital Uniwersytecki nr 2 im.dr J. Biziela

🇵🇱

Bydgoszcz, Poland

Rheuma Medicus Zaklad Opieki Zdrowotnej

🇵🇱

Warsaw, Poland

Niepubliczny Zaklad Opieki Zdrowotnej "Nasz Lekarz" Praktyka Grupowa Lekarzy Rodzinnych z

🇵🇱

Torun, Poland

Wojskowy Instytut Medyczny

🇵🇱

Warszawa, Poland

SBEI HPE Altai State Medical University of MoH and SD

🇷🇺

Barnaul, Russian Federation

SBHI of Kem. "Regional Clinical Hospital for War Veterans"

🇷🇺

Kemerovo, Russian Federation

Municipal City Hospital #2

🇷🇺

Omsk, Russian Federation

First Moscow State Medical University n.a. I.M. Sechenov

🇷🇺

Moscow, Russian Federation

Republican Hospital n.a. V.A. Baranov

🇷🇺

Petrozavodsk, Russian Federation

Regional Clinical Hospital

🇷🇺

Vladimir, Russian Federation

City Clinical Hospital #12

🇷🇺

Saratov, Russian Federation

Clinical Rheumatology Hospital #25

🇷🇺

St. Petersburg, Russian Federation

Out - patient Clinic # 107

🇷🇺

St. Petersburg, Russian Federation

Yaroslavl State Medical University

🇷🇺

Yaroslavl, Russian Federation

Dr CE Spargo and Dr RB Bhorat

🇿🇦

Cape Town, South Africa

Naidoo, A

🇿🇦

Durban, South Africa

Winelands Medical Research Centre

🇿🇦

Stellenbosch, South Africa

Hospital General Universitario Gregorio Marañon

🇪🇸

Madrid, Spain

Hospital Universitario 12 de Octubre

🇪🇸

Madrid, Spain

Hospital de Sagunto

🇪🇸

Sagunto, Spain

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

Guy's Hospital

🇬🇧

London, United Kingdom

© Copyright 2025. All Rights Reserved by MedPath