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LSALT Peptide for Prevention or Attenuation of Acute Kidney Injury (AKI) in Patients Undergoing On-Pump Cardiac Surgery

Phase 2
Recruiting
Conditions
Acute Kidney Injury
Cardiac Surgery
Interventions
Drug: Placebo
Registration Number
NCT05879432
Lead Sponsor
Arch Biopartners Inc.
Brief Summary

To evaluate the percentage of subjects with AKI within 7 days following on-pump cardiac surgery defined by the KDIGO (Kidney Disease: Improving Global Outcomes) criteria:

1. Increase in baseline (pre-surgery) serum creatinine (SCr) by ≥26.5 μmol/L (≥0.3 mg/dL) within 7 days; OR

2. Increase in baseline SCr to ≥1.5 times baseline, which is known or presumed to have occurred within the first 7 days following surgery; OR

3. Urine output \< 0.5 mL/kg/h for \>6 hours.

Detailed Description

This study is a randomized, double-blind, multicenter interventional study to assess safety and efficacy of LSALT peptide versus placebo (matching drug-free saline) in patients undergoing on-pump cardiac surgery. Patients will be followed for safety and efficacy up to Day 28 (EOS), with Day 1 being the day of randomization of study drug administered at least 1 hour prior to induction of anesthesia.

A total of 240 patients will be included in the study, 120 patients each will be randomized to LSALT peptide or placebo. This study will be double-blinded with only the pharmacist at the site unblinded for the purpose of preparing drug/placebo for injection.

All subjects will undergo tests during the Screening period (window days -14 to Day 1). After satisfying all inclusion and exclusion criteria, the patient will be randomized equally to the following study arms:

* LSALT peptide 10 mg IV administered over 1 hour twice daily, every 12 ± 1hour, for 5 days

* Placebo IV administered over 1 hour twice daily, every 12 ± 1 hour, for 5 days

Study treatment will be initiated pre-operatively on Day 1 and continued for 5 days. Physical examinations, vital signs and urine output will be recorded daily throughout the treatment period and on days 6 and 7. Adverse events will be recorded daily throughout the treatment period, on Days 6, 7, and 28 EOS (Day 28). Kidney function (serum creatinine, serum cystatin C, and BUN), clinical laboratory tests, and other biomarkers will be assessed at baseline (prior to initiation of study drug) and monitored daily throughout the treatment period, on Days 6, 7, and EOS (Day 28). All patients will be maintained on the standard of care (SOC) as per institutional guidelines. Thus, SOC will be followed in each patient with the addition of LSALT peptide or placebo.

Subjects will be followed until EOS (Day 28 ± 3 days) to assess renal function as discussed above.

An independent Data and Safety Monitoring Board (DSMB) will evaluate patients on a continuing basis for primarily safety assessments. Per the DSMB Charter, the DSMB will meet at least monthly if not more frequently based upon enrollment throughout the study period.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
240
Inclusion Criteria
  1. Male and female ≥ 18 years of age.

  2. Scheduled for a non-emergent coronary and/or valve surgery procedure requiring on-pump cardiopulmonary bypass including but not limited to:

    • Coronary artery bypass graft (CABG) alone
    • CABG with aortic, mitral, tricuspid, or pulmonic valve replacement or repair
    • Aortic valve replacement or repair alone, with or without aortic root repair
    • Mitral, tricuspid, or pulmonic valve replacement or repair alone
    • Simultaneous replacement of several cardiac valves.
  3. Have the following AKI risk factors:

    • CKD Stage 3 (CKD-EPI eGFR ≥ 30 and < 60 mL/min/1.73 m2) and ONE or more of the following additional risk factors OR

    • CKD Stage 2 (CKD-EPI eGFR ≥ 60 and < 90 mL/min/1.73 m2) and ONE or more of the following additional risk factors:

      • Age ≥ 75 years;
      • Combined valve & coronary artery surgery;
      • Left ventricular ejection fraction (LVEF) ≤ 35% by invasive or noninvasive techniques;
      • Urinary (TIMP-2 x IGFBP7) > 0.3
      • Diabetes mellitus
      • Hypertension
      • Hyperlipidemia
  4. Sexually active women of child-bearing potential (WCBP) must be using a medically acceptable method of birth control throughout the study and for at least 1 day following the end of study and have a negative urine pregnancy test at the Screening visit. A WCBP is defined as a female who is biologically capable of becoming pregnant. A medically acceptable method of birth control includes intrauterine devices in place for at least 3 months, surgical sterilization, or the implant. In patients who are not sexually active, abstinence is an acceptable form of birth control and urine will be tested per protocol. Women who are of nonchild-bearing potential, i.e., post-menopause, must have this condition captured in their medical history. Pregnant women and nursing mothers are excluded from this study.

  5. Patient or Legally Authorized Representative (LAR) is available and willing to give written informed consent, after being properly informed of the nature and risks of the study and prior to engaging in any study-related procedures.

Exclusion Criteria
  1. The presence of AKI (KDIGO criteria) at the time of randomization
  2. Off-pump cardiac surgery
  3. Surgery to be performed under conditions of circulatory arrest or hypothermia with rectal temperature < 28°C (82.4° F)
  4. Severe chronic kidney disease: CKD-eGFR < 30 mL/min/1.73 m2) OR requiring dialysis
  5. Imminent or recent surgery for aortic dissection
  6. Surgery to correct a major congenital heart defect (e.g., Tetralogy of Fallot, transposition of the great vessels, single ventricle, or Ebstein's anomaly. Bicuspid aortic valve is not considered a congenital heart defect)
  7. Known history of active cancer which may interfere with interpretation of the results of this study
  8. Known or suspected sepsis at time of screening
  9. Pregnancy or lactation
  10. Known hypersensitivity to the study drug or any of its excipients
  11. Treatment with an investigational drug or participation in an interventional trial within 30 days prior to the first dose of study drug and throughout the study
  12. Any disease processes or confounding variables that would inappropriately alter the outcome of the study in the opinion of the investigator
  13. Inability to comply with the requirements of the study protocol.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
LSALT PeptideLSALT PeptideLSALT peptide 10 mg IV administered over 1 hour twice daily, every 12 ± 1 hour, for 5 days
PlaceboPlaceboPlacebo IV administered over 1 hour twice daily, every 12 ± 1 hour, for 5 days
Primary Outcome Measures
NameTimeMethod
To evaluate the percentage of subjects with AKI within 7 days following on-pump cardiac surgery defined by the KDIGO (Kidney Disease: Improving Global Outcomes) criteria7 days

1. Increase in baseline (pre-surgery) serum creatinine (SCr) by ≥26.5 μmol/L (≥0.3 mg/dL) within 7 days; OR

2. Increase in baseline SCr to ≥1.5 times baseline, which is known or presumed to have occurred within the first 7 days following surgery; OR

3. Urine output \< 0.5 mL/kg/h for \>6 hours.

Secondary Outcome Measures
NameTimeMethod
Need for RRT within the first 7 days following surgery7 days
Maximum severity of AKI per patient between treatment groups7 days

1. Stage 1: SCr 1.5 - 1.9 times baseline OR ≥26.5 μmol/L (≥0.3 mg/dL) increase OR urine output \<0.5 mL/kg/hr for 6-12 hours

2. Stage 2: SCr 2.0 - 2.9 times baseline OR urine output \<0.5 mL/kg/h for ≥ 12 hours

3. Stage 3: SCr ≥3.0 times baseline OR increase in SCr of ≥26.5 μmol/L (≥0.3 mg/dL) to ≥353.6 μmol/L (≥4.0 mg/dL) OR initiation of renal replacement therapy (RRT) OR urine output \<0.3 mL/kg/h for ≥24 hours OR anuria for ≥12 hours.

Time to mild, moderate, and severe AKI per patient between treatment groups7 days
Need for RRT at any time during the 28-day study28 days
Kidney function (SCr, eGFR) at 28 days (EOS)28 days
28-day all-cause mortality28 days
Composite of death, need for RRT, and/or persistent impaired renal function from baseline (MAKE [major adverse kidney event] criteria) at Day 28 (EOS)28 days
ICU length of stay (in days)28 days
Changes in urinary TIMP-2 and IGFBP7 biomarker and serum NGAL, AGT, and IL-18 biomarker levels7 days

Biomarkers will be measured at baseline and days 1, 3, 5, and 7

Development of serum anti-drug antibodies levels throughout the study28 days

Anti-drug antibodies will be measured at baseline (Day 1 prior to the first dose of study medication) and at days 1, 2, 3, 4, 5 and day 28 (EOS)

Duration of AKI at 28 days (EOS)28 days

Duration of AKI is defined as the number of days from start of AKI per KDIGO criteria to onset of resolution

Hospitalization length of stay (in days)28 days
Incidence of new-onset lung or liver disorders following surgery28 days
Change in baseline serum cystatin C, serum NGAL, serum IP-10, serum IL-1beta, serum IL-6, and serum IL-18 biomarker levels28 days

Trial Locations

Locations (8)

Cumming School of Medicine & Libin Cardiovascular Centre, University of Calgary

🇨🇦

Calgary, Alberta, Canada

Unity Health Toronto, St. Michael's Hospital

🇨🇦

Toronto, Ontario, Canada

University Health Network

🇨🇦

Toronto, Ontario, Canada

Gazi University

🇹🇷

Yenimahalle, Ankara, Turkey

Kosuyolu High Specialization Training and Research Hospital

🇹🇷

Kartal, Istanbul, Turkey

Erciyes University, Faculty of Medicine - Semiha Kibar Organ Transplant & Dialysis Hospital

🇹🇷

Melikgazi, Kayseri, Turkey

Kocaeli University, Faculty of Medicine Practices and Research Hospital

🇹🇷

İzmit, Kocaeli, Turkey

Sütçü İmam University, Faculty of Medicine

🇹🇷

Kahramanmaraş, Onikişubat, Turkey

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