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Asparaginase Encapsulated in Erythrocytes for Patients With ALL and Hypersensitivity to PEG-asparaginase

Phase 2
Completed
Conditions
Acute Lymphoblastic Leukemia
Interventions
Registration Number
NCT03267030
Lead Sponsor
Birgitte Klug Albertsen
Brief Summary

Pegylated-asparaginase (PEG-ASP) is an important part of the treatment of childhood acute lymphoblastic leukaemia (ALL). Unfortunately 13% of patients develops allergy and further treatment is impossible. Furthermore, 6% of patients have developed antibodies (silent inactivation) and have no effect of the PEG-ASP treatment. Truncated asparaginase therapy is associated with inferior event-free survival outcomes, in particular relapse in central nervous system (CNS).

Eryaspase is a new formulation of asparaginase encapsulated in erythrocytes. The erythrocyte membrane protects asparaginase against fast degradation and elimination processes. The encapsulation eliminates the direct somatic contact, and it is hypothesized that this provides the potential to prolong the activity of the enzyme and reduce toxicities.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
55
Inclusion Criteria
  1. Male or female aged 1-45 years at diagnosis of ALL.

  2. First line non-high risk ALL patients enrolled in NOPHO ALL2008 or ALLTogether pilot protocols including PEG-ASNase regimen.

  3. Documented hypersensitivity reaction to PEG-ASNase with either:

    Clinical allergy to PEG-ASNase (mild/severe). Serum ASNase activity below the lower level of quantification.

  4. Karnofsky/Lansky score ≥50.

  5. Ability to understand and willingness to sign a written ICF and to comply with the scheduled visits, treatment plans, laboratory tests and other study procedures. For patients under 18 years of age, either both parents or the legally appointed representatives had to provide consent.

Exclusion Criteria
  1. Philadelphia chromosome positive ALL.

  2. Participation in another clinical trial interfering with the study therapy with exception of NOPHO ALL-2008 or ALLTogether pilot protocol. Patients can participate in other clinical trials not interfering with the study drug. In case of doubt this is assessed by the PI.

  3. Uncontrolled intercurrent illness including, but not limited to, patients receiving combination antiretroviral therapy or patients with severe or systemic infection, or psychiatric illness/social situations that would limit compliance with study requirements.

  4. Other severe acute/chronic medical or psychiatric condition or laboratory abnormality that may increase the risk associated with study participation or study drug administration, or may interfere with the interpretation of study results, and in the judgment of the investigator would make the patient inappropriate for entry into this study.

  5. Pregnant or lactating females (serum human chorionic gonadotropin pregnancy test at screening). Use of a highly effective contraceptive measure in women of child-bearing potential and sexually active girls that are of child-bearing potential is required (contraceptive measures are specified in section 6.0).

  6. Inadequate organ functions, which prohibit further asparaginase administration;

    1. History of pancreatitis
    2. History of serious hemorrhage or serious thrombosis with prior asparaginase therapy
    3. Severe hepatic impairment at the time of administration (bilirubin >3 times ULN, transaminases >10 times ULN)
    4. Pre-existing known coagulopathy (e.g. haemophilia)
  7. History of grade 3 or higher transfusion reactions or any contraindication to receive blood transfusion. Presence of specific anti-erythrocytes antibodies (auto-antibodies or anti-public antibodies) preventing from getting a compatible packed Red Blood Cells for the patient.

  8. Patient under concomitant treatment likely to cause hemolysis.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
GRASPAGRASPAGRASPA will replace remaining PEG-asparaginase doses in case of hypersensitivity.
Primary Outcome Measures
NameTimeMethod
Pharmacokinetics ASNase Activity >100 U/L at 14 Days14 days after first infusion

The primary endpoint was the percentage of patients with ASNase activity \>100 U/L at 14 days following the first infusion (nadir). ASNase activity \>100 U/L is considered adequate for complete asparagine depletion in the blood.

Secondary Outcome Measures
NameTimeMethod
Pharmacokinetic Parameters14 days after fourth infusion

Percentage of patients with ASNase activity \>100 U/L at 14 days following the fourth infusion of the 2-week dosing intervals. ASNase activity \>100 U/L is considered adequate for complete asparagine depletion in the blood.

Trial Locations

Locations (23)

Tallin Childrens Hospital

🇪🇪

Tallin, Estonia

Childrens Hospital, Helsinki. University Central Hospital

🇫🇮

Helsinki, Finland

Tartu University Clinics

🇪🇪

Tartu, Estonia

Turku University Hospital

🇫🇮

Turku, Finland

Aarhus University hospital

🇩🇰

Aarhus, Aarhus N, Denmark

Rigshospitalet, Hematological department

🇩🇰

Copenhagen, Denmark

University Hospital of Oulu

🇫🇮

Oulu, Finland

Tampere University Hospital

🇫🇮

Tampere, Finland

Oslo Universitetssykehus, Rikshospitalet

🇳🇴

Oslo, Norway

Aahus University hospial, hematological department

🇩🇰

Aarhus, Aarhus C, Denmark

Aalborg University Hospital, pediatric department

🇩🇰

Aalborg, Denmark

Odense University hospital, pediatric department

🇩🇰

Odense, Denmark

Rigshospitalet, Child and Adolescent Medicine

🇩🇰

Copenhagen, Denmark

Kuopio University Hospital

🇫🇮

Kuopio, Finland

St Olavs Hospital

🇳🇴

Trondheim, Norway

Vilnius University Children's Hospital

🇱🇹

Vilnius, Lithuania

Helse Bergen

🇳🇴

Bergen, Norway

Drottning Silvias Barn- och ungdomssjukhus

🇸🇪

Göteborg, Sweden

Universitetssjukhuset Linköping

🇸🇪

Linköping, Sweden

Skånes Universitets sjukhus

🇸🇪

Lund, Sweden

Astrid Lindgrens Barnsjukhus Karolinska

🇸🇪

Stockholm, Sweden

arn- och Ungdomscentrum Norrlands Universitetssjukhus

🇸🇪

Umeå, Sweden

Akademiska sjukhuset Uppsala

🇸🇪

Uppsala, Sweden

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