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A Clinical Trial to Evaluate the Pharmacokinetics and Safety of Fimasartan and Amlodipine in Healthy Male Subjects

Phase 1
Completed
Conditions
Hypertension
Interventions
Drug: Fimasartan/Amlodipine
Registration Number
NCT02920047
Lead Sponsor
Boryung Pharmaceutical Co., Ltd
Brief Summary

The purpose of this study is to evaluate the pharmacokinetics and safety when administrated Fimasartan/Amlodipine and when co-administrated Fimasartan and Amlodipine.

Detailed Description

This is an open-label, randomized, 3x3 partial replicated crossover study to evaluate the pharmacokinetics and safety/tolerability. Within each period, randomized subjects will be 2 dosing regimens with a fixed dose combination of Fimasartan/Amlodipine and co-administration of Fimasartan and Amlodipine.

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
60
Inclusion Criteria
  1. Male 19-50 years of age.
  2. Body mass index (BMI) ≥ 18 and ≤ 27 kg/m2 at screening.
  3. Medically healthy with no clinically significant medical history.
  4. Understands the study procedures in the Informed consent form (ICF), and be willing and able to comply with the protocol.
Exclusion Criteria
  1. History or presence of clinically significant medical or psychiatric condition or disease.
  2. Positive results at screening for human immunodeficiency virus (HIV), hepatitis B surface antigen (HBsAg) or hepatitis C virus (HCV).
  3. Seated blood pressure is less than 100/65 mmHg or greater than 140/90 mmHg at screening.
  4. Plasma donation within a month prior to the first dose of study drug.
  5. Participation in another clinical trial within 3 months prior to the first dose of study drug(s).

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Sequence AFimasartan + AmlodipinePeriod 1(Treatment A) - Period 2(Treatment A) - Period 3(Treatment B) There will be a washout of 14 days between the each period.
Sequence AFimasartan/AmlodipinePeriod 1(Treatment A) - Period 2(Treatment A) - Period 3(Treatment B) There will be a washout of 14 days between the each period.
Sequency CFimasartan/AmlodipinePeriod 1(Treatment B) - Period 2(Treatment A) - Period 3(Treatment A) There will be a washout of 14 days between the each period.
Sequency CFimasartan + AmlodipinePeriod 1(Treatment B) - Period 2(Treatment A) - Period 3(Treatment A) There will be a washout of 14 days between the each period.
Sequence BFimasartan/AmlodipinePeriod 1(Treatment A) - Period 2(Treatment B) - Period 3(Treatment A) There will be a washout of 14 days between the each period.
Sequence BFimasartan + AmlodipinePeriod 1(Treatment A) - Period 2(Treatment B) - Period 3(Treatment A) There will be a washout of 14 days between the each period.
Primary Outcome Measures
NameTimeMethod
Cmax and AUClast of Fimasartan, AmlodipineTime Frame: 0~144 hour after medication
Secondary Outcome Measures
NameTimeMethod
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