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Effect of Food on Bioavailability of a Modified Release Formulation of Imatinib

Phase 1
Completed
Conditions
Healthy
Interventions
Registration Number
NCT00422825
Lead Sponsor
Novartis Pharmaceuticals
Brief Summary

This is a single center, four-treatment, four period, crossover study to evaluate the effect of food on the relative bioavailability of a single dose of imatinib (STI571) given as a 800 mg modified release tablet, MR2 compared to twice-daily doses of 400 mg film-coated imatinib tablets. There will be a 10 day wash out phase between treatments and a 1 week safety period at the end of the study. Each participant will receive all four treatments

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
16
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Imatinib 800mgimatinib-
Imatinib 400mgimatinib-
Primary Outcome Measures
NameTimeMethod
Assess the effect of food on bioavailability and pharmacokinetics of modified and immediate release formulations of imatinib
Secondary Outcome Measures
NameTimeMethod
To compare the relative bioavailability of a single dose 800 mg modified release formulation (with a low fat breakfast) with the marketed 400 mg immediate release tablet administered (with a low fat breakfast) twice daily
To compare safety and tolerability of 800 mg modified release formulation with or without food.
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