MedPath

Adjunctive Zonisamide in Primary Generalised Tonic Clonic Seizures

Phase 3
Terminated
Conditions
Epilepsy
Interventions
Drug: Placebo
Registration Number
NCT00692003
Lead Sponsor
Eisai Limited
Brief Summary

Zonisamide is already marketed for the treatment of partial seizures in epilepsy. This study is intended to provide evidence that zonisamide is safe and effective in the treatment of primary generalised tonic-clonic seizures. The total trial duration will be 5.5-6.5 months. After that subjects who have completed the study will be eligible to enrol in an open-label extension study until zonisamide is marketed for this indication or further development in this indication stops. This extension study will be described in a separate protocol (E2090-E044-316).

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
21
Inclusion Criteria
  1. Subject is male or female and aged 6-65 years.
  2. Subject has ≥ 3 PGTCS over the two months before screening and during the eight weeks Baseline Period with at least one seizure in each one month period. PGTCS must occur in the context of Idiopathic Generalized Epilepsy (IGE) and may be accompanied by other primary generalized seizures, provided these are also consistent with a diagnosis of IGE.
  3. Subject (or parent/caregiver, for subjects below the age of consent) is willing to sign an informed consent form. For subjects below the age of consent in their country, where appropriate they must be willing to give informed (written or verbal) assent. Subjects from the age specified in local regulations will be required to sign an appropriate informed consent form.
  4. Subject is taking a stable regimen of one or two other Antiepileptic Drugs (AEDs) for at least two weeks prior to Visit 1 (start of the Baseline Period).
  5. Subject has a clinical diagnosis of any type of idiopathic generalized epilepsy which has PGTCS (and which may be accompanied by other generalized seizure types), according to the International League Against Epilepsy (ILAE) Classification of Epileptic Seizures (1981) and the ILAE Classification of Epilepsies and Epileptic Syndromes (1989). Diagnosis should have been established by clinical history, electroencephalogram (EEG) and computed tomography/magnetic resonance imaging (CT/MRI) of the brain consistent with idiopathic generalized epilepsy. CT/MRI scan should have been performed within five years of the screening visit or, if not available from this period, should be performed in the Baseline Period.
  6. EEG should have been performed within one year of the screening visit or, if not available from this period, should be performed in the Baseline Period.
  7. Female subjects are pre-menarchal, or if of childbearing potential, are not pregnant or lactating or are post-menopausal.
  8. Female subjects of childbearing potential must abide by the one of the following medically acceptable contraceptive measures: oral contraception pill, contraceptive injections, implants or patches, intrauterine device in place for at least three months or vasectomised partner or abstinence throughout the study.
  9. Subject has a body weight ≥ 20 kg.
Exclusion Criteria
  1. Subject has progressive or focal neurological disease (as determined by pre-existing brain imaging such as CT or MRI performed maximally five years before the screening visit), or clinically significant organic disease.
  2. Subject has a history of, or results of clinical investigations (including EEG data) that are suggestive of, partial seizures as defined by the ILAE, including generalized tonic clonic seizures which are suspected to be secondarily generalized.
  3. Subjects with cryptogenic or symptomatic generalized epilepsy.
  4. Subjects with psychogenic seizures.
  5. Subject has a history of status epilepticus within a year of screening while complying with AEDs.
  6. Subject has seizures that only occur in clustered patterns.
  7. Subject has a history of renal calculi or renal insufficiency (above the upper normal limits of creatinine).
  8. Subject has a known diagnosis of human immunodeficiency virus (HIV) or hepatitis B or C.
  9. Subject had a predisposing condition that might interfere with absorption, distribution, or excretion of zonisamide.
  10. Subject has a history of sensitivity to sulfonamide drugs or zonisamide and its excipients.
  11. Subject has a recent history of excessive alcohol use or drug abuse.
  12. Subject has a history of suicide attempt in the five years before the screening visit..
  13. Subject has abnormal screening laboratory values that were clinically significant.
  14. Subject has a history of demonstrated non-compliance with treatment or the subject or parent/caregiver can be reasonably expected not to be compliant with study procedures or to complete the study.
  15. Subject has participated in a study of an investigational drug or device within 30 days prior to screening.
  16. Subject has received previous treatment with zonisamide.
  17. Subject is treated with ketogenic diet or vagus nerve stimulator.
  18. Subject has a history of necessary treatment with rescue benzodiazepines which is foreseen to continue during the study. Rescue benzodiazepines will not be allowed in this study (stable dosing with a benzodiazepine as (one of the) baseline anti-epileptic drug(s) is allowed).
  19. Current psychosis or moderate to severe depression, or use of anti-psychotic drugs, MAOIs, tricyclic antidepressants, benzodiazepine or barbiturate treatment for disorders other than epilepsy, and stimulants (amphetamine derivatives) within 28 days before the screening visit.
  20. Concomitant use of acetazolamide, carbonic anhydrase inhibitors such as topiramate and drugs with anticholinergic activity.
  21. Concomitant use of felbamate or use of felbamate within two months prior to Visit 1.
  22. Subject is not able to swallow capsules.
  23. Subject is not in general good health as determined by medical history, physical exam and screening laboratory results.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
ZonisamideZonisamide-
PlaceboPlacebo-
Primary Outcome Measures
NameTimeMethod
Number of Participants Considered Responders as Assessed During the Maintenance PeriodBaseline (Week -8/-4 to Week 0) and Maintenance Phase (Week 4 to Week 16)

The number of participants who were considered responders during the 12 week Maintenance Period (Week 4 to Week 16). A responder was defined as a participant with a decrease from baseline in Primary Generalised Tonic-Clonic Seizures (PGTCS) frequency of \>= 50% (i.e. 28-day PGTC seizure frequency in the period from Week 4 to the Week 16 visit compared to Week -8/-4 to randomization at Week 0). Each participant's response to treatment was assessed on the basis of their seizure diaries. The diary was dispensed at the Screening Visit and maintained by the participant (parent/caregiver) through out the titration and maintenance treatment periods until the Early termination Visit at Week 16. Due to early termination of the study by the Sponsor, no formal analyses were conducted.

Secondary Outcome Measures
NameTimeMethod
Absolute Change From Baseline in 28-day PGTC Seizure FrequencyBaseline and up to 16 weeks

Absolute Change from Baseline in 28-day PGTC Seizure Frequency was assessed both for the Maintenance Period alone (Week 4 to Week 16) and for the entire double-blind treatment period (Week 0 to Week 16). Due to early termination of the study by the Sponsor, no formal analyses were conducted.

Trial Locations

Locations (71)

Fakultni nemocnice Plzen

🇨🇿

Plzen, Czech Republic

West-Tallinn Central Hospital

🇪🇪

Tallinn, Estonia

Wojewodzki Szpital Specjalistyczny im. M. Kopernika

🇵🇱

Gdansk, Poland

Centrum Neurologii Klinicznej

🇵🇱

Krakow, Poland

GOU VPO Novosibirsk State Medical University of Roszdrav

🇷🇺

Novosibirsk, Russian Federation

Yaroslavskaya State Medical Academy

🇷🇺

Yaroslavl, Russian Federation

CH Split

🇭🇷

Split, HR, Croatia

Kaunas Medical University Hospital

🇱🇹

Kaunas, Lithuania

Vilnius University Hospital Santariskiu klinikos

🇱🇹

Vilnius, Lithuania

Heim Pal Hospital

🇭🇺

Budapest, Hungary

UHC Zagreb

🇭🇷

Zagreb, HR, Croatia

Fakultni nemocnice s poliklinikou Ostrava

🇨🇿

Ostrava, Czech Republic

Centrum neurologicke pece

🇨🇿

Rychnov nad Kneznou, Czech Republic

Neurologicke oddeleni

🇨🇿

Hradec Kralove, Czech Republic

Private Neurologi Office

🇨🇿

Kromeriz, Czech Republic

Oulu University Central Hospital

🇫🇮

Oulu, Finland

Uniwersytet Medyczny

🇵🇱

Poznan, Poland

GOU VPO Smolensk State Medical Academy of Roszdrav

🇷🇺

Smolensk, Russian Federation

Derzhavna Ustanova Institut Nevrologiy

🇺🇦

Kharkiv, Ukraine

Neurodiagnostica AP OY

🇪🇪

Tallinn, Estonia

Neuromeda

🇱🇹

Kaunas, Lithuania

National Institute of Psychiatry and Neurology

🇭🇺

Budapest, Hungary

Bekes County Pandy Kalman Hospital

🇭🇺

Gyula, Hungary

Vas County Markusovszky Hospital

🇭🇺

Szombathely, Hungary

Szpital im. M. Kopernika

🇵🇱

Lodz, Poland

Spitalul Clinic Judetean de Urgenta Tg Mures

🇷🇴

Tg Mures, Romania

Szent Istvan Hospital

🇭🇺

Budapest, Hungary

FGU Moscow Research Institute of Psychiatry of Roszdrav

🇷🇺

Moscow, Russian Federation

Niepubliczny ZOZ KENDRON

🇵🇱

Bialystok, Poland

Spitalul Clinic Judetean de Urgenta Sf Spiridon Iasi

🇷🇴

Iasi, Romania

Clinical Center of Nis

🇷🇸

Nis, Serbia

The Royal Melbourne Hospital

🇦🇺

Melbourne, Victoria, Australia

Fakultni nemocnice Olomouc

🇨🇿

Olomouc, Czech Republic

Institut fur Diagnostik der Epilepsien

🇩🇪

Berlin, Germany

Neurologische Gemeinschaftspraxis

🇩🇪

Munchen, Germany

Austin Health

🇦🇺

Heidelburg, Victoria, Australia

St. Vincents Hospital

🇦🇺

Melbourne, Australia

Interdisziplinares Epilepsiezentrum am Klinikum der Philipps-Universitat Marburg

🇩🇪

Marburg, Germany

Tartu University Hospital

🇪🇪

Tartu, Estonia

Bacs-Kiskun County ONK Hospital

🇭🇺

Kecskemet, Hungary

Specjalistyczny Szpital Wieloprofilowy

🇵🇱

Katowice, Poland

Orszagos Idegsebeszeti Tudomanyos Intezet

🇭🇺

Budapest, Hungary

GOU VPO Krasnoyarskaya State Medical Academy of Roszdrav

🇷🇺

Krasnoyarsk, Russian Federation

GOU VPO Russian State Medical University of Roszdrav

🇷🇺

Moscow, Russian Federation

Odesskyy Derzhavnyy Medychnyy Universitet

🇺🇦

Odesa, Ukraine

Strategic Health Evaluators Pty Ltd

🇦🇺

Chatswood, New South Wales, Australia

The Prince of Wales Hospital

🇦🇺

Randwick, New South Wales, Australia

CH Sestre Milosrdnice University Hospital

🇭🇷

Zagreb, HR, Croatia

Nemocnice Na Homolce

🇨🇿

Praha 5, Czech Republic

Kuopio Epilepsy Center

🇫🇮

Kuopio, SF, Finland

Neurochirurgische Klinik der Universitat Freiburg

🇩🇪

Freiburg, Germany

Universitatsklinikum Ulm

🇩🇪

Ulm, Germany

Bethesda Hospital for Children

🇭🇺

Budapest, Hungary

Veszpem County Csolnoky F. Hospital

🇭🇺

Veszpem, Hungary

Spitalul Clinic de Psihiatrie

🇷🇴

Bucharest, Romania

Spitalul Universitar de Urgenta Bucuresti

🇷🇴

Bucharest, Romania

Spitalul Clinic Judetean de Urgenta Cluj

🇷🇴

Cluj-Napoca, Romania

Spitalul Clinic de Urgenta Sfanta Treime

🇷🇴

Iasi, Romania

Centrul Medical Sana

🇷🇴

Bucharest, Romania

GOU VPO Moscow State University of Medicine and Dentistry of Roszdrav

🇷🇺

Moscow, Russian Federation

St. Petersburg State Medical Pediatric Academy

🇷🇺

St. Petersburg, Russian Federation

GU St. Petersburg Research Institute of Psychoneurology

🇷🇺

St.Petersburg, Russian Federation

GOU VPO St. Petersburg State Medical University

🇷🇺

St.Petersburg, Russian Federation

Clinical Center of Serbia

🇷🇸

Belgrade, Serbia

University Medical Center Zvezdara

🇷🇸

Belgrade, Serbia

Clinical Center Kragujevac

🇷🇸

Kragujevac, Serbia

Kyiv City Psychiatric Hospital #2, Poliklinichne Viddilenya

🇺🇦

Kyiv, Ukraine

Tsentr Psihosomatychnoyi Patologiyi Dnipropetrovskoyi oblasnoyi klinichnoyi likarni imeni Mechnikova

🇺🇦

Dniepropetrovsk, Ukraine

Miska Klinichna psihonevrologichna Tsentr Epilepsiyi

🇺🇦

Kyiv, Ukraine

Lvivskyiy oblasnyi Protyepileptuchnyy tsentr

🇺🇦

Lviv, Ukraine

Vinnitskyy Natsionalnyy Medychnyy Universitet

🇺🇦

Vinnitsa, Ukraine

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