MedPath

A Study To Evaluate The Safety And Efficacy Of PF-06826647 In Participants With Moderate To Severe Ulcerative Colitis

Phase 2
Withdrawn
Conditions
Ulcerative Colitis
Interventions
Drug: PF-06826647 300 mg QD
Drug: Placebo
Drug: PF-06826647 100 mg QD
Drug: PF-06826647 600 mg QD
Drug: PF-6826647 400 mg QD
Registration Number
NCT04209556
Lead Sponsor
Pfizer
Brief Summary

The purpose of this study is to evaluate efficacy and safety of PF-06826647 in moderate to severe ulcerative colitis

Detailed Description

Not available

Recruitment & Eligibility

Status
WITHDRAWN
Sex
All
Target Recruitment
Not specified
Inclusion Criteria
  • Participants with moderate to severe UC as defined by a total Mayo score of ≥6, with a rectal bleeding subscore of ≥1 and an endoscopic subscore of ≥2;
  • Participants must have inadequate response to, loss of response to, or intolerance to at least one conventional therapy for UC: Oral, intravascular, or intramuscular corticosteroids; Immunosuppressants (azathioprine [AZA], 6-MP, or methotrexate [MTX]); Anti-tumor necrosis factor (TNF) inhibitors (eg, infliximab, adalimumab, or golimumab); Anti-integrin inhibitors (eg, vedolizumab); JAK inhibitor (eg, tofacitinib); Anti-IL-12/IL-23 inhibitors (eg, ustekinumab).
Read More
Exclusion Criteria
  • Presence of indeterminate colitis, microscopic colitis, ischemic colitis, infectious colitis, radiation colitis, and diverticular disease associated with colitis, or Crohn's disease
  • Participants displaying clinical signs of fulminant colitis or toxic megacolon;
  • Participants with evidence of colonic dysplasia, adenomas or neoplasia.
Read More

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PF-06826647 300 mg QDPF-06826647 300 mg QDPF-06826647 300 mg QD
PlaceboPlaceboPlacebo
PF-06826647 100 mg once a day (QD)PF-06826647 100 mg QDPF-06826647 100 mg once a day (QD)
PF-06826647 600 mg QDPF-06826647 600 mg QDPF-06826647 600 mg QD
Open Label Extension, PF-06826647 400 mg QDPF-6826647 400 mg QDPF-06826647 400 mg QD
Primary Outcome Measures
NameTimeMethod
Number of Participants With Clinical Laboratory AbnormalitiesAt Week 60

Following parameters will be analyzed for laboratory examination: hematology (hemoglobin, hematocrit, red blood cell count, platelet count, white blood cell count, total neutrophils, eosinophils, monocytes, basophils, lymphocytes); liver function (aspartate aminotransferase, alanine aminotransferase, total bilirubin, lactate dehydrogenase, alkaline phosphatase, albumin, total protein); renal function (blood urea nitrogen, creatinine, uric acid); electrolytes (sodium, potassium, chloride, calcium, phosphate, bicarbonate); clinical chemistry (glucose, creatine kinase); immunology (CRP); urinalysis (dipstick \[urine specific gravity, decimal logarithm of reciprocal of hydrogen ion activity {pH} of urine, glucose, protein, blood, ketones, bilirubin\], microscopy \[urine RBC, WBC, urate crystals, calcium, oxalate, miscellaneous \[urine mucus and leucocytes\]).

Percentage of participants achieving endoscopic responseAt Week 8

Endoscopic response is defined by Mayo endoscopic index \< 2

Number of Adverse Events (AEs), Serious Adverse Events (SAEs) based on severity and withdrawals due to adverse events (AEs)At Week 60
Percentage of participants with clinically significant changes in Electrocardiogram (ECG)At Week 60

Clinical significant changes in ECG

Number of Participants With Categorical changes from baseline in Vital Signs DataAt Week 60

Number of participants with increase from baseline in sitting SBP and DBP of greater than or equal to 30 mmHg at Week 60.

Secondary Outcome Measures
NameTimeMethod
Percentage of participants achieving endoscopic remissionAt Week 8 and 60

Endoscopic remission is defined as Mayo endoscopic index of 0

Number of Participants With Clinical Laboratory AbnormalitiesAt Week 8

Following parameters will be analyzed for laboratory examination: hematology (hemoglobin, hematocrit, red blood cell count, platelet count, white blood cell count, total neutrophils, eosinophils, monocytes, basophils, lymphocytes); liver function (aspartate aminotransferase, alanine aminotransferase, total bilirubin, lactate dehydrogenase, alkaline phosphatase, albumin, total protein); renal function (blood urea nitrogen, creatinine, uric acid); electrolytes (sodium, potassium, chloride, calcium, phosphate, bicarbonate); clinical chemistry (glucose, creatine kinase); immunology (CRP); urinalysis (dipstick \[urine specific gravity, decimal logarithm of reciprocal of hydrogen ion activity {pH} of urine, glucose, protein, blood, ketones, bilirubin\], microscopy \[urine RBC, WBC, urate crystals, calcium, oxalate, miscellaneous \[urine mucus and leucocytes\]).

Percentage of participants achieving clinical remissionAt Week 8 and 60

Clinical remission is defined by total Mayo score of ≤ 2 with no individual subscore of \> 1

Change from baseline in total Mayo scoreAt Week 8 and 60
Percentage of participants with clinically significant changes in Electrocardiogram (ECG)At Week 8

Clinically significant changes from baseline in ECG (heart rate, QT, QTc, PR and QRS intervals)

Number of Participants With Categorical Vital Signs DataAt Week 8

Number of participants with increase from baseline in sitting SBP and DBP of greater than or equal to 30 mmHg at Week 8.

Percentage of participants achieving mucosal healingAt Week 8 and 60

Mucosal healing is defined as both total Mayo score and histologic index of ≤ 1.

Percentage of participants achieving clinical responseAt Week 8 and 60

Clinical response is defined as a decrease from baseline of at least 3 points in total Mayo score with at least 30% change, accompanied by at least one point decrease or absolute score of 0 or 1 in rectal bleeding subscore.

Mean change from baseline in partial Mayo score over timeUp to 60 weeks
Number of Adverse Events (AEs), Serious Adverse Events (SAEs) based on severity and withdrawals due to adverse events (AEs)At Week 8

Trial Locations

Locations (24)

ADVA Clinical Research

🇺🇸

Inglewood, California, United States

Hope Clinical Research

🇺🇸

Canoga Park, California, United States

Gastroenterology Consultants P.C.

🇺🇸

Roswell, Georgia, United States

Centinela Valley Endoscopy Center

🇺🇸

Inglewood, California, United States

Inglewood Imaging Center

🇺🇸

Inglewood, California, United States

Renaissance Imaging Center (CT/Xray)

🇺🇸

Northridge, California, United States

Valley Endoscopy Center (Colonoscopy/Flexible sigmoidoscopy)

🇺🇸

Tarzana, California, United States

Gastroenterology Associates of New Jersey, LLC (c/o TrialSpark, Inc.)

🇺🇸

Clifton, New Jersey, United States

Associates in Gastroenterology (c/o TrialSpark, inc)

🇺🇸

Woodbridge, Virginia, United States

Surinder Saini, M.D., Inc.

🇺🇸

Newport Beach, California, United States

Saludmax Medical Corp.

🇺🇸

Miami, Florida, United States

Alliance Clinical Research of Tampa

🇺🇸

Tampa, Florida, United States

Internal Medicine Associates (c/o TrialSpark, Inc.)

🇺🇸

Merrillville, Indiana, United States

Physicians Ambulatory Surgery Center, LLC, dba Physicians Endoscopy Center

🇺🇸

Houston, Texas, United States

Memorial Hermann SW Surgery Center

🇺🇸

Houston, Texas, United States

Gastroenterology Associates of Northern Virginia

🇺🇸

Fairfax, Virginia, United States

Verity Research, Inc.

🇺🇸

Fairfax, Virginia, United States

Houston Digestive Diseases Consultants, P.A.

🇺🇸

Houston, Texas, United States

Sugar Lakes Family Practice, PA

🇺🇸

Sugar Land, Texas, United States

Gastroenterolgy Associates of Northern Virginia

🇺🇸

Fairfax, Virginia, United States

Gastroenterology Consultants of San Antonio

🇺🇸

San Antonio, Texas, United States

Victorium Clinical Research

🇺🇸

San Antonio, Texas, United States

South Texas Radiology Imaging Center

🇺🇸

San Antonio, Texas, United States

Fair Oaks Imaging Center- Reston Radiology Consultants

🇺🇸

Fairfax, Virginia, United States

© Copyright 2025. All Rights Reserved by MedPath