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TST001 in Patients With CLDN18.2 Positive Previously Treated Advanced Biliary Tract Cancer

Phase 2
Completed
Conditions
Biliary Tract Neoplasms
Interventions
Drug: TST001
Registration Number
NCT05190575
Lead Sponsor
Shanghai Zhongshan Hospital
Brief Summary

TST001 is a recombinant humanized anti-Claudin 18.2 (CLDN18.2) IgG1 monoclonal antibody. This is an open-label, single-arm phase II study to evaluate the efficacy and safety of TST001 for patients with CLDN18.2 positive previously treated unresectable advanced or metastatic Biliary Tract Cancer.

Detailed Description

TST001 is a recombinant humanized anti-Claudin 18.2 (CLDN18.2) IgG1 monoclonal antibody. Claudin18.2 (CLDN18.2) protein is one of the family of tetraspanning proteins expressed at epithelial tight junctions and primarily expressed only in normal gastric tissues . CLDN18.2 protein is a pancancer target expressed in primary lesions and metastases of variouscancer types, including gastric cancer, biliary tract cancer and others. Current available information indicates that CLDN18.2 is a promising therapeutic target for the treatment of solid tumors.

This is an open-label, single-arm phase II study to evaluate the efficacy and safety of TST001 for patients with CLDN18.2 positive previously treated unresectable advanced or metastatic Biliary Tract Cancer. Eligible patients will be treated with TST001 until disease progression or other discontinuation criteria met. If there is ≥ one objective response among the first 15 enrolled patients, then the trial continues to enroll a total of 40 patients; if not, then the trial discontinues.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
8
Inclusion Criteria
  • Histologically confirmed, unresectable advanced or metastatic biliary tract cancer.
  • Patients failed at least one prior line of systemic medications; if patients had disease progression during or within 6 months after the completion of adjuvant therapy or neoadjuvant therapy, the adjuvant therapy or neoadjuvant therapy could be regarded as one line of therapy.
  • CLDN18.2 expression positive confirmed through tumor tissue.
  • Patients with at least one measurable disease according to RECISTv1.1.
  • ECOG PS of 0 or 1.
  • Patients have predicted life expectancy ≥ 12 weeks.
  • Paitients with adequate cardica, liver, renal function, etc.
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Exclusion Criteria
  • • History of another concurrent primary malignancy.

    • Untreated or symptomatic CNS metastases.
    • Prior treatment targeting CLDN18.2.
    • Major surgical procedure, prior locoregional therapy such as radioembolization within 28 days prior to the first dose of study drug.
    • Prior serious hypersensitivity to monoclonal antibody or any component of the investigational drug.
    • Patients had any of the following within 6 months prior to first dose of study treatment: cerebrovascular accident, transient ischemic attack, myocardial infarction or unstable angina pectoris, heart failure NYHA III or IV degree, or uncontolled uarrhythmia requiring intervention.
    • Patients who are pregnant or lactating.
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Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
TST001TST001Drug: TST001 IV infusion every 3 weeks until disease progression or other discontinuation criteria.
Primary Outcome Measures
NameTimeMethod
ORR18 months

ORR according to RECIST 1.1 using investigator assessment

Secondary Outcome Measures
NameTimeMethod
PFS18 months

PFS accorridng RECSIST1.1 using investigator assessment

DoR18 months

DoR accroding to RECSIST1.1 using investigator assessment

DCR18 months

Patients who were assessed as partial response, complete response or stable disease

Safety & tolerability18 months

Adverse events will be graded according to NCI-CTC AE v5.0

Overall survival18 months

Time from enrollment to death of any cause

Trial Locations

Locations (1)

Zhongshan hospital

🇨🇳

Shanghai, China

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