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A Study of RNK05047 in Subjects With Advanced Solid Tumors/Diffuse Large B-cell Lymphoma (CHAMP-1)

Phase 1
Recruiting
Conditions
DLBCL
Advanced Solid Tumor
Interventions
Registration Number
NCT05487170
Lead Sponsor
Ranok Therapeutics (Hangzhou) Co., Ltd.
Brief Summary

This is a first in human, Phase 1/2 open-label multi-center, dose escalation and expansion study to evaluate the safety, tolerability, PK, PD and efficacy of RNK05047 when administered an intravenous (IV) infusion to subjects with advanced solid tumors, including diffuse large B-cell lymphoma (DLBCL).

This is a 2-part study (dose escalation, cohort expansion) with sequential enrollment.

Detailed Description

In Part 1, enrolled subjects will receive IV RNK05047 once weekly for 3 consecutive weeks in a 4-week cycle (no treatment in the fourth week). The dose-escalation phase will follow a standard 3+3 design, with 3 subjects enrolled into the first dosing cohort to receive RNK05047 at the starting dose of 0.75 mg/kg.

In Part 2, once RP2D has been established, additional subjects (3 to 5 cohorts of approximately 15 subjects per cohort) will be enrolled in the cohort-expansion phase of the study. Tumor types for these cohorts will be determined based on data from the dose-escalation phase of the study and emerging results from preclinical studies or other scientific data. These dose expansion cohorts in all groups may be done concurrently.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
32
Inclusion Criteria
  • Pathologically documented locally advanced or metastatic solid tumor
  • Refractory or intolerant to all available standard-of-care therapies for advanced disease
  • Measurable disease
  • Archived tumor tissue collected
  • ECOG Performance Status of 0 or 1
  • BMI ≥ 18 kg/m2
  • Adequate liver, renal, hematologic, and coagulation parameters
  • Negative serum pregnancy test (for women of childbearing potential) at Screening and a negative urine or serum pregnancy test on Day 1 prior to the first infusion
  • Males and females of childbearing potential must agree to use a highly effective method of contraception during treatment and for at least 4 months after the last dose of study treatment.
  • Must be able to understand and comply with the conditions of the protocol and must have read and understood the consent form and provided written informed consent.
Exclusion Criteria
  • Concurrent anticancer therapy: Radiotherapy, chemotherapy, biological therapy, or other anticancer investigational agents NOTE: at least 5 half-lives must have been ensued for any prior systemic cancer therapy agent before subject received the study drug on Day 1
  • Unresolved toxicities from prior anticancer therapy, defined as not having resolved according to CTCAE version 5.0 Grade ≤ 1, excluding Grade 1 alopecia
  • Presence or suspicion of active central nervous system (CNS) metastases and/or leptomeningeal carcinomatosis
  • Peripheral neurotoxicity ≥ Grade 2 according to CTCAE v5.0
  • Known active infection with HIV, HTLV-1, hepatitis B or C
  • Women who are pregnant or breastfeeding
  • History of another malignancy unless the subject has been treated with curative intent for this malignancy

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
RNK05047RNK05047Dose-escalation of RNK05047 IV infusion
Primary Outcome Measures
NameTimeMethod
Part 1: Incidence of DLTsthrough 1 cycle/4 weeks
Part 2: Incidence of TEAEsthrough study completion, an average of 1 year
Part 1: Incidence of TEAEsthrough study completion, an average of 1 year
Part 2: Objective response rate (ORR) based on RECIST 1.1/RECIL 2017through study completion, an average of 1 year
Part 2: Duration of response (DoR) based on RECIST 1.1/RECIL 2017through study completion, an average of 1 year
Part 2: Disease Control Rate (DCR) based on RECIST 1.1/RECIL 2017through study completion, an average of 1 year
Part 2: Progression-free Survival (PFS) based on RECIST 1.1/RECIL 2017through study completion, an average of 1 year
Secondary Outcome Measures
NameTimeMethod
Part 1: ORR based on RECIST 1.1/RECIL 2017through study completion, an average of 1 year
Part 2: Overall Survival (OS)through study completion, an average of 1 year
Part 2: Plasma concentration RNK05047Through Cycle 3/approximately 12 weeks
Part 1: PFS based on RECIST 1.1/RECIL 2017through study completion, an average of 1 year
Part 1: Plasma concentration RNK05047Through Cycle 3/approximately 12 weeks
Part 1: DoR based on RECIST 1.1/RECIL 2017through study completion, an average of 1 year
Part 1: DCR based on RECIST 1.1/RECIL 2017through study completion, an average of 1 year

Trial Locations

Locations (5)

Cancer Hospital, Chinese Academy of Medical Sciences

🇨🇳

Beijing, Beijing, China

Beijing Cancer Hospital

🇨🇳

Beijing, Beijing, China

Emory University Winship Cancer Institute

🇺🇸

Atlanta, Georgia, United States

Norton Cancer Institute

🇺🇸

Louisville, Kentucky, United States

Weill Cornell - NY Presbyterian Hospital

🇺🇸

New York, New York, United States

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