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Clinical Trials/NCT00550212
NCT00550212
Completed
Phase 1

An Open-Label, Single-Dose Study of the Mass Balance and Metabolic Disposition of Orally Administered [14C]-Labeled HKI-272 in Healthy Male Subjects

Puma Biotechnology, Inc.0 sites6 target enrollmentStarted: March 2008Last updated:
ConditionsHealthy
Interventionsneratinib

Overview

Phase
Phase 1
Status
Completed
Enrollment
6
Primary Endpoint
Mass balance, metabolic distribution, PK

Overview

Brief Summary

The purpose of this study is to evaluate the mass balance and metabolic distribution of C14-labeled HKI-272 in healthy male subjects.

Study Design

Study Type
Interventional
Allocation
Non Randomized
Intervention Model
Single Group
Primary Purpose
Treatment
Masking
None

Eligibility Criteria

Ages
18 Years to 50 Years (Adult)
Sex
Male
Accepts Healthy Volunteers
Yes

Inclusion Criteria

  • Healthy male subjects, aged 18 to 50 years.

Exclusion Criteria

  • Female subjects

Arms & Interventions

1

Experimental

240 mg

Intervention: neratinib (Drug)

Outcomes

Primary Outcomes

Mass balance, metabolic distribution, PK

Time Frame: 10 days

Secondary Outcomes

No secondary outcomes reported

Investigators

Sponsor Class
Industry
Responsible Party
Sponsor

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