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Systemic Oxaliplatin or Intra-arterial Chemotherapy Combined With LV5FU2 +/- Irinotecan and an Target Therapy in First Line Treatment of Metastatic Colorectal Cancer Restricted to the Liver

Phase 3
Recruiting
Conditions
Colorectal Neoplasms
Interventions
Registration Number
NCT02885753
Lead Sponsor
Federation Francophone de Cancerologie Digestive
Brief Summary

Colorectal cancer is the 3rd most common cancer in France and the 2nd cause of death from cancer. Between 30 to 60% of patients develop limited or predominant liver metastases. Surgical resection of these metastases, only curative treatment is not immediately possible in 10-15% of cases. In unresectable patients, current palliative treatments are based on systemic chemotherapy associated or not with the targeted therapies (anti-EGFR (panitumumab), anti-VEGF (bevacizumab)). In this patient population, special attention was paid to intensified treatment regimens in order to improve their efficiency and improving the tumoral response rate, the intensity of the response and its earliness correlate with improved overall and progression-free survival.

The intra-arterial use of oxaliplatin coupled with IV chemotherapy has yielded OR levels of 64% in patients having survived one or more lines of chemotherapy IV and 62% in patients who have progressed on oxaliplatin IV. In addition, the HIA administration of oxaliplatin limits systemic and especially neurological toxicities, thanks to a greater hepatic clearance.

In conclusion, the combination of systemic chemotherapy, targeted therapy and HIAC with oxaliplatin has showed promising efficacy results associated with good tolerance from the first line onwards. Indeed, we can expect from the Phase II recent data, a control rate close to 100%, with high response rates associated with early maturity and depth responses as well as prolonged survival. However, to date, in the absence of randomized trial testing this combination, this strategy does not have sufficient evidence to be integrated in our routine practices, and HIAC remains limited to a few expert centers in treatment catch-up.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
348
Inclusion Criteria
  • Histologically proven colorectal adenocarcinoma with hepatic metastasis(es)
  • At least one measurable hepatic metastasis according to the criteria RECIST v1.1
  • No other metastatic sites except lung nodules if number ≤ 3 and < 10 mm
  • RAS mutation status known (determination of KRAS mutation (exons 2,3 and 4) and determination of the NRAS mutation (exons 2,3 and 4))
  • Age ≥ 18
  • WHO ≤ 2 (Appendix 4)
  • No prior treatment by chemotherapy except perioperative or adjuvant chemotherapy discontinued for more than 12 months
  • Life expectancy > 3 months
  • PNN > 1500/mm3, platelets > 100 000/mm3, Hb > 9 g/dLq
  • Bilirubin < 25 mmol/L, AST < 5x ULN, ALT < 5 x ULN, ALP < 5 x ULN, TP > 60%, proteinuria from 24H < 1 g
  • Creatinine clearance > 50 mL/min according to MDRD formula (Appendix 4)
  • Patient affiliated to a social security scheme
  • Patient information and signature of the informed consent
Exclusion Criteria
  • Contraindications specific to the installation of a KTHIA: thrombosis of the hepatic artery, arterial vascular anatomy may compromise a secondary hepatic resection.
  • Patient immediately eligible for a curative therapy (surgical and/or percutaneous) after discussion in CPR
  • Following alterations in the 6 months prior to inclusion: myocardial infarction, angina, severe/unstable angina, coronary artery bypass surgery, congestive heart failure NYHA class II, III or IV, stroke or transient ischemic attack
  • Hypertension not controlled by medical treatment (SBP > 140 mmHg and/or DBP> 90 mmHg with blood pressure taken according to the diagram of the HAS)
  • A history of abdominal fistula, gastrointestinal perforation, intra-abdominal abscess or active gastrointestinal bleeding in the 6 months preceding the start of treatment
  • Progressive gastroduodenal ulcer, wound or fractured bone
  • Abdominal or major extra-abdominal surgery (except diagnostic biopsy) or irradiation in the 4 weeks before starting the treatment
  • Transplant patients, HIV positive or other immune deficiency syndromes
  • Any progressive pathology not balanced over the past 6 months: hepatic failure, renal failure, respiratory failure
  • Peripheral neuropathy > 1
  • Patient with interstitial pneumonitis or pulmonary fibrosis
  • History of chronic diarrhea or inflammatory disease of the colon or rectum, or unresolved occlusion or sub-occlusion in symptomatic treatment
  • History of malignant pathologies during the past 5 years except basocellular skin carcinoma considered in complete remission or in situ cervical carcinoma, properly treated
  • Patient already included in another clinical trial with an experimental molecule
  • Any known specific contraindication or allergy or hypersensitivity to the drugs used in the study (cf RCP Appendix 7)
  • Known deficit in DPD
  • QT/QTc range > 450 msec for men and > 470 msec for women
  • K+ < LNL, Mg2+ < LNL, Ca2+ < LNL
  • Lack of effective contraception in patients (men and/or women) of childbearing age, pregnant or breastfeeding women, women of childbearing age not having had a pregnancy test
  • Persons deprived of liberty or under supervision
  • Impossibility of undergoing medical monitoring during the trial for geographic, social or psychological reasons

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Reference arm FOLFOX with oxaliplatin intravenous + targeted therapy to RAS statusOxaliplatin intravenousPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm FOLFOX with oxaliplatin intraarterial + targeted therapy to RAS status5 FU continuousPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intraarterially Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm FOLFOX with oxaliplatin intraarterial + targeted therapy to RAS statusOxaliplatin intra-arterielPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intraarterially Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Reference arm FOLFOX with oxaliplatin intravenous + targeted therapy to RAS status5 FU bolusPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm mFOLFIRINOX with oxaliplatin intraarterial + BevacizumabOxaliplatin intra-arterielBevacizumab (5 mg/Kg) Oxaliplatin (85 mg/m²) intraarterially Irinotecan (150 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 2400 mg/m² intravenously over 46 hours
Reference arm FOLFOX with oxaliplatin intravenous + targeted therapy to RAS status5 FU continuousPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm FOLFOX with oxaliplatin intraarterial + targeted therapy to RAS status5 FU bolusPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intraarterially Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm mFOLFIRINOX with oxaliplatin intraarterial + Bevacizumab5 FU continuousBevacizumab (5 mg/Kg) Oxaliplatin (85 mg/m²) intraarterially Irinotecan (150 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 2400 mg/m² intravenously over 46 hours
Reference arm mFOLFIRINOX with oxaliplatin intravenous + BevacizumabOxaliplatin intravenousBevacizumab (5 mg/Kg) Oxaliplatin (85 mg/m²) intravenously Irinotecan (150 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 2400 mg/m² intravenously over 46 hours
Reference arm mFOLFIRINOX with oxaliplatin intravenous + Bevacizumab5 FU continuousBevacizumab (5 mg/Kg) Oxaliplatin (85 mg/m²) intravenously Irinotecan (150 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm FOLFOX with oxaliplatin intraarterial + targeted therapy to RAS statusFolinic acidPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intraarterially Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm FOLFOX with oxaliplatin intraarterial + targeted therapy to RAS statusPanitumumabPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intraarterially Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm FOLFOX with oxaliplatin intraarterial + targeted therapy to RAS statusBevacizumabPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intraarterially Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Reference arm FOLFOX with oxaliplatin intravenous + targeted therapy to RAS statusFolinic acidPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Reference arm FOLFOX with oxaliplatin intravenous + targeted therapy to RAS statusPanitumumabPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Reference arm FOLFOX with oxaliplatin intravenous + targeted therapy to RAS statusBevacizumabPanitumumab (6 mg/kg if RAS wild) or Bevacizumab (5 mg/Kg if RAS mutated) Oxaliplatin (85 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 400 mg/m² in bolus of 10 minutes 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm mFOLFIRINOX with oxaliplatin intraarterial + BevacizumabFolinic acidBevacizumab (5 mg/Kg) Oxaliplatin (85 mg/m²) intraarterially Irinotecan (150 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm mFOLFIRINOX with oxaliplatin intraarterial + BevacizumabBevacizumabBevacizumab (5 mg/Kg) Oxaliplatin (85 mg/m²) intraarterially Irinotecan (150 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 2400 mg/m² intravenously over 46 hours
Experimental arm mFOLFIRINOX with oxaliplatin intraarterial + BevacizumabIrinotecanBevacizumab (5 mg/Kg) Oxaliplatin (85 mg/m²) intraarterially Irinotecan (150 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 2400 mg/m² intravenously over 46 hours
Reference arm mFOLFIRINOX with oxaliplatin intravenous + BevacizumabFolinic acidBevacizumab (5 mg/Kg) Oxaliplatin (85 mg/m²) intravenously Irinotecan (150 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 2400 mg/m² intravenously over 46 hours
Reference arm mFOLFIRINOX with oxaliplatin intravenous + BevacizumabBevacizumabBevacizumab (5 mg/Kg) Oxaliplatin (85 mg/m²) intravenously Irinotecan (150 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 2400 mg/m² intravenously over 46 hours
Reference arm mFOLFIRINOX with oxaliplatin intravenous + BevacizumabIrinotecanBevacizumab (5 mg/Kg) Oxaliplatin (85 mg/m²) intravenously Irinotecan (150 mg/m²) intravenously Folinic Acid (400 mg/m²) intravenously 5Fu: 2400 mg/m² intravenously over 46 hours
Primary Outcome Measures
NameTimeMethod
progression-free survival24 months after randomization

comparison of radiological/clinical progression free survival

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (85)

Hôpital André Mignot

🇫🇷

Le Chesnay, France

Hôpital Belle Isle

🇫🇷

Metz, France

CHR

🇫🇷

Orleans, France

CH d'Auxerre

🇫🇷

Auxerre, France

CHIC

🇫🇷

Quimper, France

CHU de Pont Chaillou

🇫🇷

Rennes CEDEX 9, France

CHU Charles Nicolle

🇫🇷

Rouen CEDEX 01, France

Centre Paul Strauss

🇫🇷

Strasbourg, France

Hôpital Sainte Musse

🇫🇷

Toulon, France

Institut de cancérologie de Lorraine

🇫🇷

Vandœuvre-lès-Nancy, France

Centre Hospitalier de Saint Malo

🇫🇷

Saint-Malo, France

Hôpital Paul BROUSSE

🇫🇷

Villejuif, France

CAC - Gustave Roussy

🇫🇷

Villejuif, France

CH D'Abbeville

🇫🇷

Abbeville CEDEX, France

CHU - Hôtel Dieu

🇫🇷

Nantes, France

Centre François Baclesse

🇫🇷

Caen, France

Hôpital Privé d'Antony

🇫🇷

Antony, France

CH de Beauvais

🇫🇷

Beauvais, France

Centre de Radiothérapie Pierre Curie

🇫🇷

Beuvry, France

PRIVE - Infirmerie Protestante de Lyon

🇫🇷

Caluire-et-Cuire, France

Centre Hospitalier Métropole Savoie

🇫🇷

Chambéry CEDEX, France

CH William Morey

🇫🇷

Chalon-sur-Saône, France

Centre Georges-François Leclerc

🇫🇷

Dijon, France

Hôpital Henri Mondor

🇫🇷

Créteil CEDEX, France

GHM Institut Daniel Hollard

🇫🇷

Grenoble CEDEX 1, France

CHU Grenoble - Hôpital Albert Michallon

🇫🇷

La Tronche, France

Ch - Chd Vendee

🇫🇷

La Roche Sur Yon, France

CMC Les Ormeaux

🇫🇷

Le Havre, France

CH Annecy Genevois

🇫🇷

Pringy, France

Polyclinique Francheville

🇫🇷

Périgueux, France

Hôpial Privé du Confluent Le Confluent Centre Catherine de Sienne

🇫🇷

Nantes, France

CHU - Hôpital Européen George Pompidou

🇫🇷

Paris, France

CH - Pau

🇫🇷

Pau, France

Institut Curie

🇫🇷

Paris, France

CH René Dubois

🇫🇷

Pontoise, France

CHU Robert Debré

🇫🇷

Reims CEDEX, France

Hôpital Drome Nord

🇫🇷

Romans-sur-Isère, France

CAC - Eugène Marquis

🇫🇷

Rennes, France

Clinique Mutualiste de l'Estuaire - Cité Sanitaire

🇫🇷

Saint Nazaire, France

PRIVE - Saint Grégoire

🇫🇷

Saint-Grégoire, France

Chu - Hopital Nord Chu Saint Etienne

🇫🇷

Saint-Priest-en-Jarez, France

Clinique Trenel

🇫🇷

Sainte Colombe, France

CHU de Saint Etienne - Hôpital Nord

🇫🇷

Saint-Priest-en-Jarez, France

CHU Nancy-Brabois

🇫🇷

Vandœuvre-lès-Nancy, France

Hôpitaux du Leman

🇫🇷

Thonon-les-Bains, France

Hôpital Sud

🇫🇷

Amiens, France

Centre Hospitalier du pays d'Aix

🇫🇷

Aix-en-Provence, France

PRIVE - Polyclinique Bordeaux Nord

🇫🇷

Bordeaux, France

CH - Côte Basque

🇫🇷

Bayonne CEDEX, France

PRIVE - Sainte Catherine

🇫🇷

Avignon, France

CH Jean Minjoz

🇫🇷

Besançon, France

CMCO Côte d'Opale

🇫🇷

Boulogne-sur-Mer, France

Hôpital Duchenne

🇫🇷

Boulogne-sur-Mer, France

Institut Bergonié

🇫🇷

Bordeaux CEDEX, France

Hôpital Louis Pasteur

🇫🇷

Chartres, France

Clinique Saint Côme

🇫🇷

Compiègne CEDEX, France

Hôpital Privé Sainte Marie

🇫🇷

Chalon-sur-Saône, France

CH - Sud Francilien

🇫🇷

Corbeil-Essonnes, France

Hopitaux Civils de Colmar

🇫🇷

Colmar, France

CHU - Hôpital François Mitterand

🇫🇷

Dijon, France

Institut de Cancérologie de Bourgogne - GRRECC

🇫🇷

Dijon, France

CH Marne La Vallée-Jossigny - Hôpital André Mignot

🇫🇷

Jossigny, France

CH du Mans

🇫🇷

Le Mans CEDEX 9, France

CAC - Léon Bernard

🇫🇷

Lyon, France

Hôpital de Bicêtre

🇫🇷

Le Kremlin-Bicêtre, France

CH - Saint Joseph

🇫🇷

Marseille, France

Hôpital Edouard Herriot

🇫🇷

Lyon, France

CHU La Timone

🇫🇷

Marseille CEDEX 5, France

Hôpital Francobritannique

🇫🇷

Levallois-Perret, France

CH de Meaux

🇫🇷

Meaux, France

PRIVE - Hôpital Européen

🇫🇷

Marseille, France

Centre Hospitalier

🇫🇷

Montélimar, France

Centre d'Imagerie médicale du Confluent- IRIS GRIM

🇫🇷

Nantes, France

Hôpital Saint Antoine

🇫🇷

Paris, France

Hôpital Cochin

🇫🇷

Paris, France

CHU - Saint Louis

🇫🇷

Paris, France

PRIVE - Saint Joseph

🇫🇷

Paris, France

CH - Centre Hospitalier de Pau

🇫🇷

Pau, France

CHU - Haut Lévêque

🇫🇷

Pessac, France

CH

🇫🇷

Soissons CEDEX, France

CH Lyon Sud

🇫🇷

Pierre-Bénite CEDEX, France

CHU

🇫🇷

Poitiers, France

CAC - ICO Site René Gauducheau

🇫🇷

Saint-Herblain, France

CHU - Rangueil

🇫🇷

Toulouse, France

CH - Kantonsspital Baden

🇨🇭

Baden, Switzerland

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