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AZD5423 Single Ascending Dose Study

Phase 1
Completed
Conditions
Healthy Volunteers
Interventions
Drug: Placebo
Registration Number
NCT00963183
Lead Sponsor
AstraZeneca
Brief Summary

The aim of the study is to assess the safety, tolerability, pharmacokinetics and pharmacodynamics of AZD5423 following single ascending dose administrations in healthy male subjects.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
72
Inclusion Criteria
  • Provision of signed, written and dated informed consent prior to any study specific procedures
  • Have a body mass index (BMI) between 18 and 30 kg/m2 and weigh at least 50 kg and no more than 100 kg
Exclusion Criteria
  • Any clinically significant disease or disorder
  • Any clinically significant abnormalities at screening examination
  • Use of any prescribed or non-prescribed medication

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
BPlaceboDrug: Placebo
AAZD5423Drug: AZD5423
Primary Outcome Measures
NameTimeMethod
Safety variables (ECG, adverse events, blood pressure, pulse, body temp, safety lab), lung function and physical examinationFrequent sampling occasions during study days
Secondary Outcome Measures
NameTimeMethod
Pharmacokinetics - Maximum plasma concentration (Cmax), time to Cmax (tmax), area under the plasma concentration-time curve from zero to the time of the last measurable concentration [AUC(0-t)] and from zero to infinity (AUC)Frequent sampling occasions during study days
Add'l pharmacokinetics - Terminal rate constant (λz); terminal half-life (t½λz), Apparent plasma clearance (CL/F), apparent volume of distribution during terminal phase (Vz/F), mean residence time (MRT).Frequent sampling occasions during study days
Pharmacodynamics - Plasma cortisol concentrationsFrequent sampling occasions during study days

Trial Locations

Locations (1)

Research Site

🇬🇧

London, United Kingdom

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