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Study to Assess Analgesic Efficacy and Safety of ASP3662 in Subjects With Painful Diabetic Peripheral Neuropathy

Phase 2
Terminated
Conditions
Painful Diabetic Peripheral Neuropathy (PDPN)
Interventions
Registration Number
NCT02372578
Lead Sponsor
Astellas Pharma Global Development, Inc.
Brief Summary

The purpose of this study is to assess analgesic efficacy of ASP3662 relative to placebo in subjects with painful diabetic peripheral neuropathy (PDPN) as well as assess the safety and tolerability of ASP3662 relative to placebo.

The analgesic effect is evaluated by measuring percent responders, change in daily worst pain score, change in average daily pain score, Patient Global Impression of Change (PGIC) and Clinical Global Impression of Change (CGIC).

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
115
Inclusion Criteria
  • Subject has a BMI ≤ 40.

  • Subject has all of the following:

    1. Established diagnosis of diabetes (Type I or II) with painful diabetic peripheral neuropathy and glycosylated hemoglobin (HgbA1c) ≤ 9.5% at Screening or Randomization.
    2. Stable diabetic drug regimen for at least 3 months prior to Screening.
    3. At least a 1 year history of PDPN.
    4. Diagnosis of PDPN to be confirmed by a score of ≥ 3 on the Michigan Neuropathy Screening Instrument (MNSI) at Screening.
  • Subject has pain intensity score(s) ≥ 4 or ≤ 9 on an 11-point numeric pain rating scale (NPRS) at Screening Visit and prior to Randomization.

  • Subject agrees to complete pain diaries and is complaint with the daily pain recording prior to Randomization as defined by the completion of a minimum of 5 of 7 daily pain ratings, 3 of which are required in the last 4 days.

  • Subject's anti-diabetic regimen is anticipated to be stable throughout the study.

  • Subject must be willing to washout of all medications currently being taken for his/her PDPN (chronic and occasional/as needed) and remain off of those pain medications while participating in the study.

Exclusion Criteria
  • Subject has received prior treatment with pregabalin for PDPN and was considered unresponsive or intolerant.
  • Subject has tried and failed 3 or more drugs to treat PDPN within the past 3 years. Drugs must have been administered at therapeutic doses and have been administered for an adequate period of time.
  • Subject has a known hypersensitivity to ASP3662, pregabalin, gabapentin or acetaminophen, or their formulation components.
  • Subject has significant pain (moderate or above) due to causes other than PDPN.
  • Subject has a history of painful peripheral neuropathy due to a cause other than diabetes.
  • Subject has any lower extremity amputation
  • Subject has a current or previous foot ulcer within the past 3 months as described by medical history and/or medical examination.
  • Subject has an active malignancy or a history of malignancy (except for treated non-melanoma skin cancer) within 5 years.
  • Subject has clinically significant abnormalities in clinical chemistry, hematology, or urinalysis, or a serum creatinine at Screening.
  • Subject has creatinine clearance < 60 mL/min (estimated from serum creatinine, body weight, age, and sex using the Cockcroft and Gault equation) at Screening.
  • Subject tests positive for hepatitis B surface antigen (HBsAg) or hepatitis C antibody at Screening or has a known history of a positive test for human immunodeficiency virus (HIV) infection.
  • Subject has a positive drug screen for alcohol or drugs of abuse at Screening and/or Randomization. Subjects who are on low doses of benzodiazepines for sleep with a legitimate prescription will be allowed into the study. In addition, subjects with a positive drug screen at Randomization will be excluded.
  • Subject is currently using protocol specified non-permitted medications including OTC products and is unable or does not choose to discontinue them.
  • Subject has planned an elective surgery during planned study participation.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
ASP3662pregabalin placeboASP3662 once daily (QD) and pregabalin placebo 3 times daily (TID) for Weeks 1 - 6. ASP3662 placebo QD and pregabalin placebo TID for Week 7.
pregabalinpregabalinpregabalin TID and ASP3662 placebo QD for Weeks 1 - 7.
PlaceboASP3662 placeboASP3662 placebo QD and pregabalin placebo TID for Weeks 1 - 7.
Placebopregabalin placeboASP3662 placebo QD and pregabalin placebo TID for Weeks 1 - 7.
pregabalinASP3662 placebopregabalin TID and ASP3662 placebo QD for Weeks 1 - 7.
ASP3662ASP3662ASP3662 once daily (QD) and pregabalin placebo 3 times daily (TID) for Weeks 1 - 6. ASP3662 placebo QD and pregabalin placebo TID for Week 7.
ASP3662ASP3662 placeboASP3662 once daily (QD) and pregabalin placebo 3 times daily (TID) for Weeks 1 - 6. ASP3662 placebo QD and pregabalin placebo TID for Week 7.
Primary Outcome Measures
NameTimeMethod
Change from Baseline in mean 24-hour average pain intensity as reported on the NPRSBaseline to Week 6/ End of Treatment (EOT)

Numerical Pain Rating Scale (NPRS)

Secondary Outcome Measures
NameTimeMethod
Percentage of Responders in mean 24-hour average pain intensity scoreBaseline to Week 6/ EOT
Change from Baseline in mean of 24-hour average pain intensity scoreBaseline to Weeks 1, 2, 3, 4, 5 and 6
Change from Baseline in mean daily worst pain scoreBaseline to Week 6/ EOT
Change from Baseline in mean daily average pain scoreBaseline to Week 6/ EOT
Patient Global Impression Change (PGIC)Week 6/ EOT
Clinical Global Impression of Change (CGIC)Week 6/ EOT

Trial Locations

Locations (37)

Site US10013

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Kettering, Ohio, United States

Site US10039

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Phoenix, Arizona, United States

Site US10051

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Boston, Massachusetts, United States

Site US10033

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Salt Lake City, Utah, United States

Site US10001

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Anniston, Alabama, United States

Site US10054

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Fresno, California, United States

Site US10047

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Santa Monica, California, United States

Site US10049

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The Villages, Florida, United States

Site US10064

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Metairie, Louisiana, United States

Site US10053

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Fairfield, Connecticut, United States

Site US10003

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Oviedo, Florida, United States

Site US10034

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Austin, Texas, United States

Site US10008

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Ormond Beach, Florida, United States

Site US10018

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Clearwater, Florida, United States

Site US10009

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Aurora, Illinois, United States

Site US10036

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Chicago, Illinois, United States

Site US10019

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DeLand, Florida, United States

Site US10015

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Greer, South Carolina, United States

Site US10026

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New Bedford, Massachusetts, United States

Site US10063

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Quincy, Massachusetts, United States

Site US10040

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Houston, Texas, United States

Site US10032

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San Antonio, Texas, United States

Site US10045

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Renton, Washington, United States

Site US10004

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Homestead, Florida, United States

Site US10007

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Jupiter, Florida, United States

Site US10042

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Jacksonville, Florida, United States

Site US10017

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Tustin, California, United States

Site US10020

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Lomita, California, United States

Site US10023

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Bradenton, Florida, United States

Site US10041

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Miami Lakes, Florida, United States

Site US10014

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Duncansville, Pennsylvania, United States

Site US10043

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Hazelwood, Missouri, United States

Site US10031

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San Antonio, Texas, United States

Site US10005

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Boynton Beach, Florida, United States

Site US10046

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Orlando, Florida, United States

Site US10055

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Walnut Creek, California, United States

Site US10025

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Evansville, Indiana, United States

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