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A Phase 3 Study to Confirm the Efficacy and Safety of Linzagolix to Treat Endometriosis-associated Pain

Phase 3
Terminated
Conditions
Endometriosis
Interventions
Registration Number
NCT03986944
Lead Sponsor
Kissei Pharmaceutical Co., Ltd.
Brief Summary

The primary objective of this study is to demonstrate the efficacy and safety of linzagolix administered orally once daily for 3 months at a dose of 75 mg alone or of 200 mg in combination with add-back hormone replacement therapy (ABT: estradiol (E2) 1 mg / norethisterone acetate (NETA) 0.5 mg) versus placebo, in the management of moderate to severe endometriosis-associated pain (EAP).

Detailed Description

This is a prospective, randomized, double-blind, placebo-controlled study to demonstrate the efficacy and safety of linzagolix administered orally once daily at doses of 75 mg alone and 200 mg in combination with low dose ABT (E2 1 mg/NETA 0.5 mg) versus placebo in the management of moderate to severe EAP in 450 women.

Eligible subjects who have completed the 6-month treatment period may enter a separate extension study for 6 additional months of active treatment (no placebo control). Subjects who do not continue in the extension study will enter a 6 month treatment-free follow-up phase.

Recruitment & Eligibility

Status
TERMINATED
Sex
Female
Target Recruitment
85
Inclusion Criteria

The subject must have:

  • Her most recent surgical and - if available - histological diagnosis of pelvic endometriosis up to 10 years before screening.
  • Moderate to severe endometriosis-associated pain during the screening period.
  • Regular menstrual cycles.
  • BMI ≥ 18 kg/m2 at the screening visit.

Key

Exclusion Criteria

The subject will be excluded if she:

  • Is pregnant or breast feeding or is planning a pregnancy within the duration of the treatment period of the study.
  • Is less than 6 months postpartum or 3 months postabortion/ miscarriage at the time of entry into the screening period.
  • Has had a surgical history of any major abdominal surgery within 6 months or any interventional surgery for endometriosis performed within a period of 2 months before screening.
  • Did not respond to prior treatment with GnRH agonists or GnRH antagonists for endometriosis.
  • Has a history of, or known, osteoporosis or other metabolic bone disease.
  • Has chronic pelvic pain that is not caused by endometriosis and requires chronic analgesic or other chronic therapy which would interfere with the assessment of endometriosis-associated pain.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Linzagolix 200 mg + Add-back (E2 1 mg / NETA 0.5 mg)Placebo tablet to match 75 mg linzagolix tablet-
PlaceboPlacebo tablet to match 75 mg linzagolix tablet-
PlaceboPlacebo tablet to match 200 mg linzagolix tablet-
Linzagolix 200 mg + Add-back (E2 1 mg / NETA 0.5 mg)200 mg linzagolix tablet-
PlaceboPlacebo capsule to match Add-back capsule-
Linzagolix 75 mgPlacebo tablet to match 200 mg linzagolix tablet-
Linzagolix 75 mgPlacebo capsule to match Add-back capsule-
Linzagolix 75 mg75 mg linzagolix tablet-
Linzagolix 200 mg + Add-back (E2 1 mg / NETA 0.5 mg)Add-back capsule (E2 1 mg / NETA 0.5 mg)-
Primary Outcome Measures
NameTimeMethod
DysmenorrheaBaseline to Month 3

Change at Month 3 from baseline in the mean daily assessment of dysmenorrhea (DYS) measured on a 4-point Verbal Rating Scale (VRS) using an electronicdiary

* The 4-point VRS scale for DYS ranges from 0 to 3 (0: No pain; 1: Mild pain; 2: Moderate pain; 3: Severe pain).

* A negative change in scores would be indicative of an improvement in the pain of DYS.

Non-menstrual Pelvic PainBaseline to Month 3

Change at Month 3 from baseline in the mean daily assessment of non-menstrual pelvic pain (NMPP) measured on a 4-point Verbal Rating Scale (VRS) using anelectronic diary

* The 4-point VRS scale for NMPP ranges from 0 to 3 (0: No pain; 1: Mild pain; 2: Moderate pain; 3: Severe pain).

* A negative change in scores would be indicative of an improvement in the NMPP.

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (112)

CMEP/CMU health / ID # 812

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Saginaw, Michigan, United States

Center for Women's Health / ID # 761

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Greenwood Village, Colorado, United States

Physicians Research Options, LLC / Red Rocks Ob/Gyn / ID # 732

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Lakewood, Colorado, United States

Visions Clinical Research-Tucson / ID # 754

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Tucson, Arizona, United States

Join Clinical Trials / ID # 778

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Huntington Park, California, United States

Lynn Institute of the Ozarks / ID # 826

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Little Rock, Arkansas, United States

Mesa Obstetricians and Gyneocologists / ID # 790

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Mesa, Arizona, United States

Synexus Clinical Research US, Inc. / ID # 725

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Orlando, Florida, United States

Sensible Healthcare / ID # 749

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Ocoee, Florida, United States

Praetorian Pharmaceutical Research / ID # 739

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Marrero, Louisiana, United States

University of South Florida / ID # 738

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Tampa, Florida, United States

Cypress Medical Research Center, LLC / ID # 755

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Wichita, Kansas, United States

Pharmasite Research Inc / ID # 838

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Baltimore, Maryland, United States

Universal Axon Clinical Research / ID # 769

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Doral, Florida, United States

Futura Research, Org / ID # 781

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Norwalk, California, United States

National Research Institute / ID # 805

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Panorama City, California, United States

Women Under Study, LLC / ID # 820

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New Orleans, Louisiana, United States

A Premier Medical Research of Florida, LLC / ID # 752

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Orange City, Florida, United States

Johns Hopkins University, School Of Medicine / ID # 816

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Baltimore, Maryland, United States

Continental Clinical Solutions, LLC / ID # 777

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Towson, Maryland, United States

Providea Health Partners LLC / ID # 734

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Evergreen Park, Illinois, United States

Physician Care Clinical Research LLC / ID # 810

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Sarasota, Florida, United States

NECCR Fall River, LLC / Id # 712

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Fall River, Massachusetts, United States

Global Health Research Center, Inc. / ID # 787

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Miami Lakes, Florida, United States

Clinical Associates of Orlando, LLC / ID # 779

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Orlando, Florida, United States

Carolina Medical Trials, LLC / ID # 788

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Winston-Salem, North Carolina, United States

Women Partners in Health / ID # 836

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Austin, Texas, United States

Accel Research Sites, DeLand Clinical Research Unit / ID # 713

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DeLand, Florida, United States

Saginaw Valley Medical Research Group, LLC / ID # 743

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Saginaw, Michigan, United States

Christina Sebestyen MD, P.A. dba OBGYN North / ID # 764

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Austin, Texas, United States

Georgetown OB/GYN / ID # 770

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Georgetown, Texas, United States

Hilltop OBGYN / ID # 711

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Franklin, Ohio, United States

UT Southwestern Medical Center / ID # 823

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Dallas, Texas, United States

Clinical Neuroscience Solutions, Inc. / ID # 731

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Orlando, Florida, United States

Albuquerque Clinical Trials, Inc. / ID # 707

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Albuquerque, New Mexico, United States

Omega Research Orlando, LLC / ID # 785

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Orlando, Florida, United States

Valley OBGYN / ID # 704

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Saginaw, Michigan, United States

Christus St. Elizabeth Gadolin Research, LLC / ID # 774

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Beaumont, Texas, United States

HCWC dba DiscoveryClinical Trials / ID # 771

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Dallas, Texas, United States

Wright State Physicians / ID # 733

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Dayton, Ohio, United States

Austin Area ObGyn PLLC / ID # 701

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Austin, Texas, United States

Lawrence OB/GYN clinical Research, LLC / ID # 742

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Lawrenceville, New Jersey, United States

Carolina Institute for Clinical Research / ID # 728

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Fayetteville, North Carolina, United States

MacArthur OB-Gyn Research / ID # 840

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Irving, Texas, United States

FMC Science / ID # 730

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Lampasas, Texas, United States

Penn State Health Milton S. Hershey Medical Center / ID # 804

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Hershey, Pennsylvania, United States

WR-ClinSearch, LLC / ID # 821

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Chattanooga, Tennessee, United States

University of Tennessee Medical Center / ID # 780

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Knoxville, Tennessee, United States

DCT-AACT, LLC dba Discovery Clinical Trials / ID # 815

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Pflugerville, Texas, United States

Matrix Clinical Research / ID # 751

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Los Angeles, California, United States

Coral Way Research / ID # 799

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Miami, Florida, United States

Suncoast Research Group, LLC / ID # 756

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Miami, Florida, United States

Biotech Pharmaceutical Group LLC / ID # 786

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Miami, Florida, United States

La Salud Research Clinic, Inc. / ID # 824

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Miami, Florida, United States

Suncoast Research Associates, LLC / ID # 760

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Miami, Florida, United States

LCC Medical Research Institute / ID # 814

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Miami, Florida, United States

Atlanta Women's Research Institute, Inc. / ID # 727

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Atlanta, Georgia, United States

Office of Edmond Pack, MD / Id # 818

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Las Vegas, Nevada, United States

Complete Healthcare for Women / ID # 801

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Columbus, Ohio, United States

Ventavia Research Group, LLC / ID # 729

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Houston, Texas, United States

Vilo Research Group / ID # 709

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Houston, Texas, United States

UT Health Clinical Res Ctr / ID # 828

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Houston, Texas, United States

TMC Life Research, Inc. / ID # 809

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Houston, Texas, United States

Seattle Reproductive Medicine / ID # 811

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Seattle, Washington, United States

Precision Research Institute / ID # 792

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San Diego, California, United States

MD Strategies Research Centers / ID # 765

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San Diego, California, United States

Wasatch Clinical Research / ID # 746

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Salt Lake City, Utah, United States

Highland Clinical Research / ID # 708

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Salt Lake City, Utah, United States

Clinical Research Associates Inc / ID # 802

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Nashville, Tennessee, United States

Precision Trials AZ, LLC / ID # 783

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Phoenix, Arizona, United States

Quality of LIfe Medical & Research Center, LLC / ID # 813

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Tucson, Arizona, United States

Applied Research Center of Arkansas / ID # 735

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Little Rock, Arkansas, United States

Long Beach Clinical Trials, LLC / ID # 768

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Long Beach, California, United States

Dr. David I. Lubetkin, LLC / ID # 703

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Boca Raton, Florida, United States

Helix Biomedics Clincial Research, LLC / ID # 750

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Boynton Beach, Florida, United States

Clinical Neuroscience Solutions, Inc. / ID # 773

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Jacksonville, Florida, United States

South Florida Clinical Research Institute / ID # 747

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Margate, Florida, United States

Sonara Clinical Research, LLC / ID # 720

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Meridian, Idaho, United States

GCP Clinical Research, LLC / ID # 825

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Tampa, Florida, United States

Moore Health Wellness Research Institute, LLC / ID # 795

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Chicago, Illinois, United States

Horizon Research Group of Opelousas, LLC / ID # 757

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Eunice, Louisiana, United States

Onyx Clinical Research / ID # 793

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Flint, Michigan, United States

Unified Women's Clinical Research - Green Valley OBGYN / ID # 719

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Greensboro, North Carolina, United States

Eastern Carolina Women's Center / Id # 794

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New Bern, North Carolina, United States

ClinOhio Research Services, LLC / ID # 722

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Columbus, Ohio, United States

Unified Women's Clinical Research - Raleigh / Id # 714

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Raleigh, North Carolina, United States

OB/GYN Associates of Erie / ID # 706

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Erie, Pennsylvania, United States

The Clinical Trial Center / ID # 744

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Jenkintown, Pennsylvania, United States

VitaLink Research - Upstate / ID # 789

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Greenville, South Carolina, United States

Clinical Trials of South Carolina / ID # 741

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North Charleston, South Carolina, United States

VitaLink Research Spartanburg / ID # 753

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Spartanburg, South Carolina, United States

Clinical Neuroscience Solutions, Inc / ID # 772

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Memphis, Tennessee, United States

Signature Gyn Services / ID # 726

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Fort Worth, Texas, United States

Medical Colleagues of Texas / ID # 819

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Katy, Texas, United States

Maximos OB/GYN / ID # 737

🇺🇸

League City, Texas, United States

DCT-McAllen Primary Care Research, LLC dba Discovery Clinical Trials / ID # 803

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McAllen, Texas, United States

Northeast Clinical Research of San Antonio, LLC / ID # 710

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Schertz, Texas, United States

Physicians Research Options PRO / ID # 766

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Draper, Utah, United States

Physicians' Res Options - PG / ID # 833

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Pleasant Grove, Utah, United States

Clinical Research Partners, LLC / ID # 715

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Richmond, Virginia, United States

Clinical Research Partners, LLC / ID # 775

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Richmond, Virginia, United States

Seattle Women's: Health, Research, Gynecology / ID # 702

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Seattle, Washington, United States

CARe Clinic / ID # 872

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Red Deer, Alberta, Canada

McMaster University Medical Centre / ID # 870

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Hamilton, Ontario, Canada

Victory Reproductive Care / ID # 873

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Windsor, Ontario, Canada

Ponce Medical SChool Foundation Inc./ CAIMED Center / ID # 891

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Ponce, Puerto Rico

Puerto Rico Medical Research Inc. / ID # 890

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Ponce, Puerto Rico

Birmingham OBGYN / ID # 740

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Birmingham, Alabama, United States

Downtown Women's Health Care / ID # 718

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Denver, Colorado, United States

Oregon Health & Science University / ID # 791

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Portland, Oregon, United States

Seasons at Bristol / ID # 705

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Bristol, Tennessee, United States

Tidewater Clinical Research The Group for Women / ID # 716

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Virginia Beach, Virginia, United States

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