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Acute Consequences Of Food-induced Glucocorticoid Secretion In Healthy Individuals

Early Phase 1
Completed
Conditions
Glucocorticoid Effect
Interventions
Registration Number
NCT05167084
Lead Sponsor
Eleonora Seelig
Brief Summary

In a randomized, cross-over study, 20 healthy volunteers will receive a block and replace therapy that mimics physiological GC rhythm (metyrapone plus hydrocortisone) or placebo. Participants will undergo two identical overfeeding periods with each treatment. With the block and replace therapy, food-induced GC peak will be suppressed. Metabolic and autonomic parameters will be compared to reveal, whether GCs mediate the physiological adaptions to excessive food intake.

Understanding acute effects of GCs upon food intake is critical, since repetitive disruptions of GC secretion may become harmful in chronic conditions.

Detailed Description

Obesity is one of the most serious health problems of the 21st century. To understand how we regulate our body weight is crucial for developing new treatment targets. Even though body mass index of populations is increasing, the body weight of adults is usually kept stable over time. Indeed, acute excessive food intake triggers a set of adaptions in order to prevent weight gain. The signal that triggers these beneficial adaptions is still unknown. Glucocorticoid (GC) secretion increases with acute food intake and many physiological adaptions to overfeeding coincide with classical glucocorticoid actions. The investigators therefore hypothesize that GCs are the signal that prevents weight gain during acute overfeeding.

The objective of this project is to test whether food-induced GCs represent the physiological signal that defends against weight gain.

The primary objective is to investigate whether reduction in insulin sensitivity is abolished with the block and replace therapy.

Secondary objectives are to investigate whether suppression of GC secretion during excessive food intake impairs the activation of sympathetic nervous system, satiety, satiation, energy expenditure, substrate utilization, blood pressure, secretion of neuroendocrine hormones, lipids and immune cells.

This is a double-blind, randomized, placebo-controlled cross-over study. After screening, subjects will be randomized to two crossover 8-day study periods with a washout period of 28 days:

A) Participants will receive hydrocortisone 19.9 mg/d subcutaneously via a pump in a pulsed fashion (eight times/day) and metyrapone per os (starting with a dose of 500 mg/d on day 1 to 2500mg/d on day 4, and then will be kept constant until day 8)

B) Participants will receive placebo (0,9% NaCl solution) 19.9 mg/d subcutaneously via a pump in a pulsed fashion and placebo pills per os (starting with a dose of 500 mg/d on day 1 to 2500mg/d on day 4, and then will be kept constant until day 8)

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
20
Inclusion Criteria
  • BMI 18.5 - 25 kg/m2
Exclusion Criteria
  • Previous medical history for any chronic condition in the last three months, active disease or abnormal physical examination as verified by a qualified physician.
  • Casual smoking (>6 cigarettes per day)
  • Frequent, heavy alcohol consumption (>30g/day)
  • Frequent, heavy caffeine consumption (>4 caffeinated drinks/day)
  • Regular physical exercise (>4hrs per week)
  • Shift workers
  • Participation in an investigational drug trail within the past two months
  • Intake of any drugs (prescribed, over the counter or recreational) including topical steroids and inhalers, within 48 hours of the study initiation
  • Known allergy to metyrapone
  • Inability or unwillingness to provide informed consent

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Metyrapone And HydrocortisoneMetyrapone 250 mg Oral TabletsDuring one of the study periods, subjects receive hydrocortisone 19.9 mg/d subcutaneously via a pump in a pulsed fashion (eight times/day) and metyrapone per os (starting with a dose of 500 mg/d, then the dose will be increased the next days until 2500mg/d is achieved).
Metyrapone And HydrocortisoneHydrocortisone 19,9mg s.c., pulsatile with a flow rate of 10μl/sDuring one of the study periods, subjects receive hydrocortisone 19.9 mg/d subcutaneously via a pump in a pulsed fashion (eight times/day) and metyrapone per os (starting with a dose of 500 mg/d, then the dose will be increased the next days until 2500mg/d is achieved).
PlaceboPlacebo (0,9% NaCl solution)During the other study period, subjects receive placebo (0,9% NaCl solution) 19.9 mg/d subcutaneously via a pump in a pulsed fashion and the same dose of placebo tablets p.o instead of metyrapone.
PlaceboPlacebo 250 mg TabletsDuring the other study period, subjects receive placebo (0,9% NaCl solution) 19.9 mg/d subcutaneously via a pump in a pulsed fashion and the same dose of placebo tablets p.o instead of metyrapone.
Primary Outcome Measures
NameTimeMethod
Insulin sensitivityTwo 8-day intervention periods

Change in insulin sensitivity assessed with a mixed meal tolerance test

Secondary Outcome Measures
NameTimeMethod
GLP-1 (nmol/l)Two 8-day intervention periods

Blood sample

PYY (pg/ml)Two 8-day intervention periods

Blood Sample

Aldosterone (Adrenal Steroid Hormones)Two 8-day intervention periods

Blood Sample

17-Hydroxypregnenolon (Adrenal Steroid Hormones)Two 8-day intervention periods

Blood Sample

Substrate utilisationTwo 8-day intervention periods

Respiratory quotient assessed with indirect calorimetry

Systolic and diastolic blood pressureTwo 8-day intervention periods

Assessment of blood pressure with a standard blood pressure monitor.

ReninTwo 8-day intervention periods

Blood Sample

Pregnenolon (Adrenal Steroid Hormones)Two 8-day intervention periods

Blood Sample

TSH (mIU/l)Two 8-day intervention periods

Blood Sample

WeightTwo 8-day intervention periods

Measurement of weight with a standard scale

Energy expenditureTwo 8-day intervention periods

Basal metabolic rate measured with indirect calorimetry

Progesteron (Adrenal Steroid Hormones)Two 8-day intervention periods

Blood Sample

11-Deoxycorticosteron (Adrenal Steroid Hormones)Two 8-day intervention periods

Blood Sample

T3 (nmol/l)Two 8-day intervention periods

Blood Sample

SatietyTwo 8-day intervention periods

Appetite rating with visual analogue scale (VAS) from 0mm-100mm (0mm=not at all and 100mm=extreme)

SatiationTwo 8-day intervention periods

Amount of food intake with ad libitum buffet

Cortisol (nmol/l) total and freeTwo 8-day intervention periods

Blood sample

Corticosteron (Adrenal Steroid Hormones)Two 8-day intervention periods

Blood Sample

18-Hydroxycorticosteron (Adrenal Steroid Hormones)Two 8-day intervention periods

Blood Sample

17-Hydroxyprogesteron (Adrenal Steroid Hormones)Two 8-day intervention periods

Blood Sample

11-Deoxycortisol (Adrenal Steroid Hormones)Two 8-day intervention periods

Blood Sample

GIP (nmol/l)Two 8-day intervention periods

Blood Sample

T4 (nmol/l)Two 8-day intervention periods

Blood Sample

Lipids (mmol/l) ((total cholesterol, LDL-cholesterol, HDL-cholesterol and triglycerides)Two 8-day intervention periods

Blood Sample

HGH (mIU/l)Two 8-day intervention periods

Blood Sample

GDF-15 (pg/mL)Two 8-day intervention periods

Blood Sample

Sympathetic nervous system activityTwo 8-day intervention periods

Heart rate variability analysis

Trial Locations

Locations (1)

University Hospital Basel

🇨🇭

Basel, Basel-Stadt, Switzerland

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