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Efficacy and Safety of Ambervin® and Standard Therapy in Hospitalized Patients With COVID-19

Phase 3
Completed
Conditions
COVID-19
Interventions
Drug: Tyrosyl-D-alanyl-glycyl-phenylalanyl-leucyl-arginine succinate inhaled
Drug: Standard of care
Drug: Tyrosyl-D-alanyl-glycyl-phenylalanyl-leucyl-arginine succinate intramuscularly
Registration Number
NCT05656495
Lead Sponsor
Promomed, LLC
Brief Summary

This is open-labe randomized multicenter comparative Phase III study conducted in 8 medical facilities. The objective of the study is to assess the efficacy, safety and tolerability of Ambervin for intramuscular and inhaled administration in complex therapy COVID-19 compared with the Standard of care (SOC) in hospitalized patients with moderate COVID-19.

Detailed Description

Upon signing the informed consent form and screening, 313 eligible patients hospitalized with COVID-19 were randomized at a 1:1:1 ratio to receive either Ambervin intramuscular 1mg 1 times a day for 10 days or Ambervin inhaled 10mg 1 times a day for 10 days or SOC.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
313
Inclusion Criteria
  1. Availability of the Informed Consent Form of thePatient Information Leaflet (PIL) signed and dated bypatient.

  2. Men and women aged 18 to 80 years inclusive at thetime of signing the Informed Consent Form in PIL.

  3. Confirmed case of COVID-19 at the time ofscreening based on SARS-CoV-2 RNA test usingnucleic acid amplification (NAA) method. It isacceptable to include a patient with a presumptiveCOVID-19 diagnosis prior to receiving the results ofSARS-CoV-2 RNA test made at the screening stage.

  4. Hospital admission due to COVID-19.

  5. Moderate severity infection with SARS-CoV-2: Clinical signs (the presence of at least 2 of the following criteria):

    • body temperature > 38 °C;
    • RR > 22/min;
    • CT pattern typical of a viral lesion
    • shortness of breath on exertion;
    • SpO2 < 95%;
    • Serum CRP > 10 mg/L.
  6. Lesion volume is minimal or moderate; CT 1-2.

  7. Patient's consent to use reliable contraceptive methods through out the study and within 1 month for women and 3 months for men after its completion. Reliable means of contraception are: sexualabstinence, use of condom in combination withspermicide.

Women incapable of childbearing may also participate inthe study (with past history of: hysterectomy, tubal ligation,infertility, menopause for more than 2 years), as well asmen with infertility or a history of vasectomy

Exclusion Criteria
  1. Hypersensitivity to components of the study drug.
  2. Impossibility of CT procedure (for example, gypsumdressing or metal structures in the field of imaging).
  3. Obstacles or inability to perform intramuscular injections and / or inhalations
  4. Arterial hypotension (a decrease in blood pressure (BP) below 100/60 mm Hg) at the time of screening and / or a history of hypotensive crises.
  5. The need for the use of drugs from the list of prohibited therapies.
  6. Availability of criteria for severe and extremely severe disease at the time of screening
  7. Presence within 6 months prior to screening of a probable or confirmed case of moderate COVID-19
  8. History of presumptive or confirmed COVID-19 caseof moderate, severe and extremely severe course ofthe disease.
  9. Vaccination less than 4 weeks prior to screening.
  10. The need for treatment in the intensive care unit at the time of screening.
  11. Impaired liver function (AST and/or ALT ≥ 2 UNLand/or total bilirubin ≥ 1.5 UNL) at the time ofscreening.
  12. Renal impairment (GFR < 60 ml/min) at the time of screening.
  13. Positive testing for HIV, syphilis, hepatitis B and/or C.
  14. Chronic heart failure FC III-IV according to New York Heart Association (NYHA) functional classification.
  15. Malignancies in the past medical history.
  16. Alcohol, pharmacological and/or drug addiction in the past medical history and/or at the time of screening.
  17. Epilepsy in history.
  18. Schizophrenia, schizoaffective disorder, bipolardisorder, or other history of mental pathology orsuspicion of their presence at the time of screening.
  19. Severe, decompensated or unstable somatic diseases (any disease or condition that threaten thepatient's life or impair the patient's prognosis, and also make it impossible for him/her to participate in the clinical study).
  20. Any history data that the investigating physician believes could lead to complication in the interpretation of the study results or create an additional risk to the patient as a result of his/her participation in the study.
  21. Patient's unwillingness or inability to comply with procedures of the Study Protocol (in the opinion of physician investigator).
  22. Pregnant or nursing women or women planning pregnancy.
  23. Participation in another clinical study for 3 monthsprior to inclusion in the study.
  24. Other conditions that, according to the physicianinvestigator, prevent the patient from being includedin the study.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Ambervin inhaledTyrosyl-D-alanyl-glycyl-phenylalanyl-leucyl-arginine succinate inhaledArm 2 (n=105) receives the study drug Ambervin for inhalation administration 10 mg 1 time per day. The course of treatment is 10 days.
Standard of careStandard of careArm 3 (n=104) patients receive standard therapy prescribed in accordance with the recommended treatment regimens included in the InterimGuidelines for the prevention, diagnosis and treatment of new coronavirus infection (COVID-19) approved by the Russian Ministry of Health by decision of the investigator and taking into account the availability of drugs at the study site
Ambervin intramuscularlyTyrosyl-D-alanyl-glycyl-phenylalanyl-leucyl-arginine succinate intramuscularlyArm 1 (n=104) receives the study drug Ambervin for intramuscularly administration 1 mg 1 time per day. The course of treatment is 10 days.
Primary Outcome Measures
NameTimeMethod
Prevalence of patients with category 0-1 as per categorical ordinal clinical improvement WHO scaleFrom baseline to Visit 4 (days 14-15)

The proportion of patients with category 0-1 as per the categorical ordinal clinical improvement scale

Secondary Outcome Measures
NameTimeMethod
Prevalence of patients with clinical status less than 4 points on the categorical ordinal WHO scale of clinical improvementFrom baseline to Visit 3 (days 11-12) and 4 (days 14-15)

The proportion of patients with clinical status less than 4 points on the categorical ordinal WHO scale of clinical improvement

Frequency of improvement in clinical status on a categorical ordinal WHO scale of clinical improvement of 2 or more categoriesFrom baseline to Visit 3 (days 11-12) and 4 (days 14-15)

The proportion of patients with clinical status on a categorical ordinal WHO scale of clinical improvement of 2 or more categories

Time to improve clinical status on a categorical ordinal scale of clinical improvement by ≥ 1 point.From baseline to Visit 6 (study completion, day 28±1)

Number of days to improve clinical status on a categorical ordinal scale of clinical improvement by ≥ 1 point.

Prevalence of patients eligible for discharge to continue outpatient treatment according to BMRFrom baseline to Visit 2 (days 6-7), 3 (days 11-12)

The proportion of patients eligible for discharge to continue outpatient treatment according to current Cuidelines

Prevalence of patients with RR < 22/minFrom baseline to Visit 2 (days 6-7), 3 (days 11-12)

The proportion of patients with RR \< 22/min

Prevalence of patients with CRP level < 10 mg/lFrom baseline to Visit 2 (days 6-7), 3 (days 11-12)

The proportion of patients with CRP level \< 10 mg/l

Prevalence of patients with blood lymphocytes > 1.2 x 10(9)/LFrom baseline to Visit 2 (days 6-7), 3 (days 11-12)

The proportion of patients with blood lymphocytes \> 1.2 x 10(9)/L

Assessment of the degree of lung damage according to CTFrom baseline to Visit 4 (days 14-15)

The degree of lung damage according to CT

Prevalence of patients with SpO2 ≥ 95% on 2 consecutive daysFrom baseline to Visit 2 (days 6-7), 3 (days 11-12), 4 (days 14-15)

The proportion of patients with SpO2 ≥ 95% on 2 consecutive days

The frequency of transfer of patients to the intensive care unit and intensive careFrom baseline to Visit 6 (study completion, day 28±1)

The proportion of patients transferred to the intensive care unit and intensive care

The frequency of cases of the use of high flow oxygen therapy, non-invasive and invasive ventilation of lung, ECMOFrom baseline to Visit 6 (study completion, day 28±1)

The proportion of patients who used high flow oxygen therapy, non-invasive and invasive ventilation of lung, ECMO

The frequency of cases of ARDSFrom baseline to Visit 6 (study completion, day 28±1)

The proportion of patients with ARDS

The frequency of patients with a fatal outcomeFrom baseline to Visit 6 (study completion, day 28±1)

The proportion of patients with a fatal outcome

Trial Locations

Locations (10)

Ryazan State Medical University named after academician I.P. Pavlov of Ministry of Health of the Russian Federation

🇷🇺

Ryazan, Russian Federation

Voronezh Regional Clinical Hospital No.1

🇷🇺

Voronezh, Russian Federation

Infectious Clinical Hospital No.1

🇷🇺

Moscow, Russian Federation

Regional Clinical Hospital

🇷🇺

Ryazan, Russian Federation

City Hospital No. 40 Kurortny District

🇷🇺

Sestroretsk, Russian Federation

Ogarev Mordova State University of Ministry of Health of the Russian Federation

🇷🇺

Saransk, Russian Federation

Regional State Budget Healthcare Institution "Clinical hospital No. 1"

🇷🇺

Smolensk, Russian Federation

Budgetary institution of the Chuvash Republic "Emergency Hospital"

🇷🇺

Cheboksary, Russian Federation

City clinical Hospital №24

🇷🇺

Moscow, Russian Federation

State Budgetary Healthcare Institution City Clinical Hospital named after S. I. Spasokukotskiy of Moscow Healthcare Department

🇷🇺

Moscow, Russian Federation

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