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Hydroxycitrate: A Novel Therapy for Calcium Phosphate Urinary Stones

Phase 4
Recruiting
Conditions
Calcium Phosphate Kidney Stones
Interventions
Dietary Supplement: OHCit- low dose
Drug: Placebo
Dietary Supplement: OHCit- standard dose
Registration Number
NCT06003348
Lead Sponsor
University of Texas Southwestern Medical Center
Brief Summary

This study tests whether hydroxycitrate, a molecule closely related to citrate, can reduce calcium phosphate stone recurrence.

Detailed Description

In this double-blind, placebo-controlled, randomized, crossover study, each participant will undergo 4 phases of study, with the order randomized by a blocked randomization scheme. The 4 phases will be Placebo, Super CitriMax (hydroxycitrate) OHCit low dose, OHCit standard dose, or Potassium Citrate. Randomization will be stratified based on sex, concomitant thiazide use, and concomitant alkali use.

Each phase will be 1 week in duration, during which subjects will take assigned study medications. A minimum 1-week washout period will be imposed between phases. During the first 2 days of each phase, subjects will be instructed to adhere to a prescribed diet. On the last 5 days of each phase, subjects will be kept on a constant metabolic diet. Use of metabolic diet is essential to eliminate confounders that could occur from changes in dietary intake across phases. During the final two study days (days 6-7), two 24-hr urines will be collected for urine biochemistry and crystallization studies. Fasting blood will be obtained at the end of the last urine collection.

Study Medications: Subjects will receive three tablets twice daily during each phase. These will consist of either placebo, Potassium Citrate (KCit), or Super CitriMax (OHCit). Study tablets will be prepared by a compounding pharmacy, with placebo tablets similar in appearance and size to the active medication tablets.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
25
Inclusion Criteria
  • Calcium Phosphate stone formers
Exclusion Criteria
  • History of recurrent urinary tract infections
  • Chronic diarrhea
  • Estimated Glomerular Filtration Rate (eGFR) < 45 ml/min/1.73 m2
  • History of primary hyperparathyroidism
  • Hypokalemia
  • Hyperkalemia
  • Pregnancy

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Super CitriMax; OHCit-low doseOHCit- low doseSuper CitriMax 7 mEq 2 tabs, twice daily And Placebo 1 tab, twice daily Total Daily Dose: OHCit 28 mEq/d
PlaceboPlaceboPlacebo 3 tablets twice daily Total Daily Dose: None
Super CitriMax; OHCit-standard doseOHCit- standard doseSuper CitriMax 7 mEq 3 tabs, twice daily Total Daily Dose: OHCit 42 mEq/d
Potassium Citrate (Urocit®-K)Potassium CitratePotassium Citrate KCit 10 mEq 2 tabs, twice daily and Placebo 1 tab, twice daily Total Daily Dose: Citrate 40 mEq/d
Primary Outcome Measures
NameTimeMethod
Formation product (FP) for Calcium PhosphateAfter 1 week of treatment

FP is obtained by adding increasing amounts of Calcium Chloride (CaCl2) to a series of urine aliquots maintained at constant pH for 2 hours, and is identified by the point at which calcium phosphate (CaP) precipitates as detected by an absorbance microplate reader.

Calculated supersaturation using \[Calcium\] and \[Phosphate\] at that point represents FP.

Secondary Outcome Measures
NameTimeMethod
Calcium Phosphate supersaturationAfter 1 week of treatment

Supersaturation of calcium phosphate will be assessed by Joint Expert Speciation System (JESS).

Crystal growth of Calcium PhosphateAfter 1 week of treatment

We will assess crystal growth (CG) of CaP after seeding urine with a small amount of brushite (0.25 mg/ml urine) and incubating at 37°C for 3 hours (representing steady state) under constant stirring. A decrement in \[Calcium\]×\[Phosphate\] after seeding signifies crystal growth, while a \[Calcium\]×\[Phosphate\] increment represents crystal dissolution.

Trial Locations

Locations (1)

UT Southwestern Medical Center

🇺🇸

Dallas, Texas, United States

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