MedPath

Futibatinib and Pembrolizumab Combination in the Treatment of Advanced or Metastatic Urothelial Carcinoma

Phase 2
Active, not recruiting
Conditions
Advanced and Metastatic Urothelial Cancer
Interventions
Registration Number
NCT04601857
Lead Sponsor
Taiho Oncology, Inc.
Brief Summary

The purpose of the trial is to evaluate the antitumor activity and confirm the safety for the combination of Fibroblast Growth Factor Receptor (FGFR) inhibitor futibatinib and anti-programmed cell death-1 (PD-1) antibody pembrolizumab in patients with advanced or metastatic urothelial cancer who are not candidates to receive a platinum-based treatment regimens.

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
43
Inclusion Criteria
  1. Willing and able to provide written informed consent for the trial.

  2. Age ≥ 18 years of age

  3. Histologically confirmed advanced or metastatic urothelial carcinoma who have not received systemic treatment for advanced metastatic disease.

    1. Cohort A: must have an FGFR3 mutation or FGFR1-4 fusion/rearrangement.
    2. Cohort B: all other patients with UC (including patients with other FGFR or non-FGFR genetic aberrations and patients with wild-type [non-mutated] tumors)
  4. Unfit for or intolerant to standard platinum-based chemotherapy.

  5. Have an Eastern Cooperative Oncology Group (ECOG) performance status (PS) of 0 to 1.

  6. Adequate organ function.

  7. Have a measurable disease per RECIST 1.1

Exclusion Criteria
  1. Have received prior therapy with anti-PD-1, anti-PD-L1/L2 agent or FGFR inhibitor.

  2. History and/or current evidence of any of the following disorders:

    1. Non-tumor related alteration of the calcium-phosphorus homeostasis that is considered clinically significant in the opinion of the Investigator.
    2. Ectopic mineralization/calcification considered clinically significant in the opinion of the Investigator.
    3. Retinal or corneal disorder considered clinically significant in the opinion of the Investigator.
  3. Has received a live vaccine within 30 days prior to the first dose of study drug.

  4. Have an active autoimmune disease that has required systemic treatment in the past 2 years.

  5. Have a history of (noninfectious) pneumonitis that required steroids or has current pneumonitis.

  6. Have had an allogenic tissue/ organ transplant.

  7. Has known human immunodeficiency virus (HIV) and/or history of Hepatitis B or C infections, or known to be positive for Hepatitis B antigen (HBsAg)/ Hepatitis B virus (HBV) DNA or Hepatitis C Antibody or RNA.

  8. Have known active central nervous system metastases and/or carcinomatous meningitis.

  9. Has a diagnosis of immunodeficiency or is receiving chronic systemic steroid therapy.

  10. Has severe hypersensitivity (≥Grade 3) to pembrolizumab and/or any of its excipients.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
futibatinib and pembrolizumab (Cohort A)futibatinib and pembrolizumab (KEYTRUDA®))Patients with UC and FGFR3 mutation or FGFR1-4 fusion/rearrangement.
futibatinib and pembrolizumab (Cohort B)futibatinib and pembrolizumab (KEYTRUDA®))All other patients than in Cohort A with UC (including patients with other FGFR or non-FGFR genetic aberrations and patients with wild-type \[non-mutated\] tumors).
Primary Outcome Measures
NameTimeMethod
Objective response rate (ORR)Approximately 12 months

Objective response rate (ORR), defined as the proportion of patients experiencing a best overall response of partial response (PR) or complete response (CR).

Secondary Outcome Measures
NameTimeMethod
Incidence of treatment-emergent Adverse Events (AE)[Safety and Tolerability]Approximately 8 months

Safety and tolerability of the futibatinib and pembolizumab combination therapy based on reported AEs, graded according to the NCI-CTCAE, Version 5.0

Duration of response (DOR)Approximately 8 months

DOR defined as the time from the first documentation of response (CR or PR) to the first documentation of objective tumor progression or death due to any cause, whichever occurs first.

Disease control rate (DCR)Approximately 8 months

DCR defined as the proportion of patients experiencing a best overall response of stable disease (SD), PR, or CR.

Progression-free survival (PFS)Approximately 8 months

PFS defined as the time from the first dose of study therapy to the date of death (any cause) or disease progression, whichever occurs first.

Overall survival (OS)Approximately 18 months

OS defined as the time from the date of the first dose to the death date.

Trial Locations

Locations (18)

Dana Farber Cancer Institute

🇺🇸

Boston, Massachusetts, United States

Institut Paoli Calmettes - Hôpital de jour

🇫🇷

Marseille, Bouches-du-Rhône, France

Henry Ford Hospital

🇺🇸

Detroit, Michigan, United States

Centre Georges-François Leclerc

🇫🇷

Dijon, Côte d'Or, France

Centre Regional de Lutte Contre le Cancer de Lorraine

🇫🇷

Vandœuvre-lès-Nancy, France

Centre Leon Berard - departement d'oncologie medicale

🇫🇷

Lyon, Rhone, France

ALTHAIA, Xarxa Assistencial Universitària de Manresa

🇪🇸

Manresa, Brcelona, Spain

Institut De Cancerologie Gustave Roussy

🇫🇷

Villejuif, France

Hospital Clinic de Barcelona

🇪🇸

Barcelona, Spain

Hospital de La Santa Creu i Sant Pau

🇪🇸

Barcelona, Spain

Hospital Universitario Vall d'Hebrón

🇪🇸

Barcelona, Spain

Hospital Universitario Reina Sofia

🇪🇸

Córdoba, Spain

Hospital Universitario HMN Sanchinarro

🇪🇸

Madrid, Spain

Hospital la Fe

🇪🇸

Valencia, Spain

Hospital Universitario Marqués de Valdecilla

🇪🇸

Santander, Spain

Comprehensive Care Centers of Nevada

🇺🇸

Las Vegas, Nevada, United States

ICANS - Institut de cancérologie de Strasbourg Europe

🇫🇷

Strasbourg, Bas-Rhin, France

UCSF Helen Diller Family Comprehensive Cancer Center

🇺🇸

San Francisco, California, United States

© Copyright 2025. All Rights Reserved by MedPath