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Clinical Trials/ACTRN12623000431628
ACTRN12623000431628
Withdrawn
Phase 1

A Phase 1 Study to Evaluate the Safety, Tolerability, and Pharmacokinetics of ELVN-002 in Healthy Adult Volunteers, Part B: Open-label Food Effect

Enliven Therapeutics, Inc.0 sites6 target enrollmentApril 28, 2023

Overview

Phase
Phase 1
Intervention
Not specified
Conditions
Not specified
Sponsor
Enliven Therapeutics, Inc.
Enrollment
6
Status
Withdrawn
Last Updated
last year

Overview

Brief Summary

No summary available.

Registry
who.int
Start Date
April 28, 2023
End Date
TBD
Last Updated
last year
Study Type
Interventional
Sex
All

Investigators

Eligibility Criteria

Inclusion Criteria

  • 1\. Male or female, aged more than 18 to less than 60 years old (both inclusive at the time of informed consent).
  • 2\. In good general health, with no significant medical history, and no clinically significant abnormalities on physical examination at Screening and/or before the first administration of IP at the discretion of the PI or designee.
  • 3\. Body mass index (BMI) greater than 18 and less than 32\.0 kg/m2 at Screening and weight more than 50 kg.
  • 4\. Non\-smoker (has not used any tobacco products). A participant who smokes less than 2 cigarettes or equivalent (eg, cigars, vaping, nicotine patches) per week within 3 months prior to Screening can be included in the study if willing and able to stop smoking for the duration of the study, at the discretion of the PI or designee.
  • 5\. Clinical laboratory values at Screening (including haematology, biochemistry, coagulation, and urinalysis) within normal range as specified by the testing laboratory, unless deemed not clinically significant by the PI or designee.
  • 6\. Acceptable estimated glomerular filtration rate (eGFR) for the study using the Chronic Kidney Disease Epidemiology Collaboration (CKD\-EPI) creatinine equation: greater than 89 mL/min/1\.73 for participants 18 to 59 years old, or greater than 84 mL/min/1\.73 for participants 60 years old).
  • 7\. Women of childbearing potential (WOCBP) must have a negative pregnancy test at Screening and Day \-1 and be willing to have additional pregnancy tests as required throughout the study.
  • 8\. Female participants who meet 1 of the following criteria will be included.
  • a. Female participants must not be pregnant or lactating, and must use acceptable, highly effective double contraception from Screening until 90 days after the last study procedure is completed. Females with same\-sex partners (abstinence from penile\-vaginal intercourse) or who are abstinent from heterosexual intercourse are not required to use contraception when this is their preferred and usual lifestyle. Effective forms of contraception include:
  • Simultaneous use of intrauterine device (IUD) (non\-hormonal) and condom for the male partner.

Exclusion Criteria

  • 1\. Has participated in previous studies of ELVN\-002\.
  • 2\. Underlying physical or psychological medical condition that, in the opinion of the PI, could impact on the participant’s safety, participant involvement in the study, or data integrity.
  • 3\. History or surgical records of any clinically significant renal, cardiovascular, hepatic, hematopoietic, neurological, pulmonary, or gastrointestinal pathology, or other conditions known to interfere with the absorption, distribution, metabolism, or excretion of the IP, as determined by the PI or designee.
  • 4\. History of severe allergic or anaphylactic reactions, or sensitivity to ELVN\-002, itraconazole, and phenytoin, or their constituents.
  • 5\. History of malignancy, except for non\-melanoma skin cancer, excised more than 2 years ago and cervical intraepithelial neoplasia that has been successfully cured more than 5 years prior to Screening (a general practitioner \[GP] letter or biopsy report for confirmation required).
  • 6\. History of symptomatic bacterial or viral infection within 2 weeks prior to Screening.
  • 7\. Abnormal ECG findings at Screening or Day \-1 (eg, repeated demonstration of a QTc interval greater than 450 ms (male) or greater than 470 ms (female) corrected by Fridericia's formula \[QTcF] or Bazett's formula \[QTcB]) that are considered by the PI or designee to be clinically significant.
  • 8\. History of clinically significant arrhythmia, cardiac conditions, or risk factors for Torsades de Pointes (eg, heart failure, current hypokalaemia, and family history of long QT syndrome).
  • 9\. Clinically significant findings in transthoracic echocardiogram at Screening, including less than normal left ventricular ejection fraction (LVEF).
  • 10\. Blood donation or significant blood loss (greater than 500 mL) within 60 days prior to the first administration of IP.

Outcomes

Primary Outcomes

Not specified

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