MedPath

Fluconazole Prophylaxis for the Prevention of Candidiasis in Infants Less Than 750 Grams Birthweight

Phase 3
Completed
Conditions
Candidiasis
Interventions
Drug: placebo
Registration Number
NCT00734539
Lead Sponsor
Daniel Benjamin
Brief Summary

The most common etiology of infection-related death or neurodevelopmental impairment in neonates with birthweight \<750 g is invasive candidiasis. Over 70% of the premature neonates who develop invasive candidiasis will die or suffer severe, permanent neurologic impairment. Fluconazole has been commonly used off-label in the neonatal intensive care unit, but definitive recommendations for its use in the nursery have been hampered by the limited number of well-designed trials. In neonates weighing \<750 g, appropriate dosing is not known, definitive safety and long-term follow up trials have not been completed, and there have not been well-powered trials conducted to establish the efficacy of the product using mortality as part of the primary endpoint. Three recent proof-of-concept studies suggest that fluconazole will be safe and effective, and a recently completed pharmacokinetic study is providing data to give preliminary dosing guidance. The next logical step in drug development is proposed by this research: to conduct a pivotal trial to determine the safety and efficacy of fluconazole in premature neonates with 2-year neurodevelopmental follow-up assessment.

362 neonates, with a birthweight \<750g, were randomized at 33 US centers, to twice weekly fluconazole (6 mg/kg) or placebo for the first 6 weeks of life. The primary efficacy endpoint will be Candida-free survival at study day 49. The research will establish definitive dosing, safety, and efficacy of fluconazole; it will also provide critical information on the effects of fluconazole on neurodevelopmental impairment and antifungal resistance.

Potential Impact:

Approximately 17,000 neonates are born \<750 grams each year in the United States. Over 5000 will die or develop invasive Candida infections. Demonstrating safety and efficacy of fluconazole in preterm neonates will improve the survivability and long term outcomes for these neonates.

Detailed Description

362 subjects were randomized to the study at 33 US sites. Final study visits of Month 18-22 corrected age long term follow up were completed. Study database is locked.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
362
Inclusion Criteria
  • Informed consent from the legally authorized representative.
  • > 48 hours of age and < 120 hours old at time of first drug administration
  • < 750 g birth weight
  • Negative blood cultures for Candida
Exclusion Criteria
  • History of a hypersensitivity or severe vasomotor reaction to any azole
  • receiving antifungal therapy for suspected/proven invasive fungal infection
  • medical condition, in the opinion of the Investigator, may create an unacceptable additional risk
  • diagnosed with invasive candidiasis or congenital Candida infection.
  • liver failure (AST and ALT > 250 U/L)
  • renal failure (creatinine > 2 mg/dL)
  • major lethal congenital or genetic anomalies
  • triplet or higher multiple gestations

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
2placeboPlacebo IV or PO twice weekly for 6 weeks
1fluconazolefluconazole 6mg/kg IV or PO twice weekly for 6 weeks
Primary Outcome Measures
NameTimeMethod
Death or Candidiasisstudy day 49

The primary endpoint for the study is death or candidiasis.

1. Death prior to study day 49.

2. Candidiasis prior to study day 49

1. Definite: isolation of Candida from normally sterile body fluid (blood, CSF, urine \[obtained via sterile catheterization or suprapubic tap\], peritoneal fluid).

2. Probable:

i. \> 5 days of consecutive antifungal therapy

AND both:

ii. Thrombocytopenia \<150,000/mm3 iii. Positive Candida culture from nonsterile site (ETS, bag urine)

Secondary Outcome Measures
NameTimeMethod
Focal Intestinal Perforationprior to hospital discharge, up to 15 ½ months
Neurodevelopmental Impairment18-22 months corrected gestational age

Bayley-III cognition composite score of less than 70, blindness, deafness, or cerebral palsy

Candidiasisprior to hospital discharge, up to 15 ½ months

Definite or probable

Stage II or Higher Necrotizing Enterocolitisprior to hospital discharge, up to 15 ½ months
Chronic Lung Disease36 weeks corrected gestational age
Patent Ductus Arterious Requiring Surgical Ligationprior to hospital discharge, up to 15 ½ months
Retinopathy of Prematurity Requiring Laser Surgeryprior to hospital discharge, up to 15 ½ months
Periventricular Leukomalaciaprior to hospital discharge, up to 15 ½ months
Length of Hospitalizationprior to hospital discharge, up to 15 ½ months
Positive Bacterial Infection From a Sterile Siteprior to hospital discharge, up to 15 ½ months
Intraventricular Hemorrhageprior to hospital discharge, up to 15 ½ months

Grade 3 or 4

Trial Locations

Locations (33)

University of California-San Diego

🇺🇸

San Diego, California, United States

Riley Hospital

🇺🇸

Indianapolis, Indiana, United States

West Jersey Hospital - Voorhees

🇺🇸

Voorhees, New Jersey, United States

Pennsylvania Hospital

🇺🇸

Philadelphia, Pennsylvania, United States

Parkland Memorial Hospital

🇺🇸

Dallas, Texas, United States

Texas Children's Hospital/Baylor College of Medicine

🇺🇸

Houston, Texas, United States

University of Nevada School of Medicine

🇺🇸

Las Vegas, Nevada, United States

Cooks Children's Medical Center

🇺🇸

Fort Worth, Texas, United States

Columbia University Medical Center

🇺🇸

New York, New York, United States

SUNY Dowstate Medical Center

🇺🇸

Brooklyn, New York, United States

University of Texas Medical Branch

🇺🇸

Galveston, Texas, United States

Baptist Medical Center

🇺🇸

Jacksonville, Florida, United States

Arkansas Childrens Hospital

🇺🇸

Little Rock, Arkansas, United States

Pitt County Memorial Hospital

🇺🇸

Greenville, North Carolina, United States

University of Arkansas for Medical Sciences

🇺🇸

Little Rock, Arkansas, United States

University of Texas - Houston

🇺🇸

Houston, Texas, United States

Duke University Medical Center

🇺🇸

Durham, North Carolina, United States

Memorial Hospital

🇺🇸

South Bend, Indiana, United States

Tulane University School of Medicine

🇺🇸

New Orleans, Louisiana, United States

Brookdale University Medical Center

🇺🇸

Brooklyn, New York, United States

University of Minnesota, Fairview Medical Center

🇺🇸

Minneapolis, Minnesota, United States

Wesley Medical Center

🇺🇸

Wichita, Kansas, United States

Shands Jacksonville Medical Center

🇺🇸

Jacksonville, Florida, United States

Kings County Hospital Center

🇺🇸

Brooklyn, New York, United States

University of Tennessee

🇺🇸

Memphis, Tennessee, United States

Akron Children's Hospital

🇺🇸

Akron, Ohio, United States

University of Florida

🇺🇸

Gainesville, Florida, United States

University of Miami

🇺🇸

Miami, Florida, United States

Children's Hospital of Orange County

🇺🇸

Orange, California, United States

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

Wayne State University

🇺🇸

Detroit, Michigan, United States

Oregon Health Sciences Center

🇺🇸

Portland, Oregon, United States

Kosair Children's Hospital

🇺🇸

Louisville, Kentucky, United States

© Copyright 2025. All Rights Reserved by MedPath