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Clinical Trials/NCT01937767
NCT01937767
Completed
Phase 2

A Randomized, Single-blind Phase II Study Evaluating the Efficacy, Safety and Pharmacokinetics of Remimazolam in General Anesthesia in Adult Patients Undergoing Cardiac Surgery, Including Follow-up Sedation in the PACU/ICU

Paion UK Ltd.1 site in 1 country90 target enrollmentAugust 2013

Overview

Phase
Phase 2
Intervention
Propofol
Conditions
General Anesthesia
Sponsor
Paion UK Ltd.
Enrollment
90
Locations
1
Primary Endpoint
Proportion of patients with successful anesthesia
Status
Completed
Last Updated
6 years ago

Overview

Brief Summary

This phase II study in patients undergoing elective cardiac surgery will evaluate the efficacy, safety, and pharmacokinetics of remimazolam, compared with propofol and sevoflurane, during the induction and maintenance of general anesthesia.

Registry
clinicaltrials.gov
Start Date
August 2013
End Date
February 19, 2014
Last Updated
6 years ago
Study Type
Interventional
Study Design
Parallel
Sex
All

Investigators

Responsible Party
Sponsor

Eligibility Criteria

Inclusion Criteria

  • scheduled for major elective cardiac surgery.
  • scheduled for mechanical ventilation via tracheal intubation.

Exclusion Criteria

  • thoraco-abdominal replacement of the aorta or other procedure expected to be accompanied by a massive hemorrhage (at least 15% of the circulating blood volume).

Arms & Interventions

Propofol

Induction: Propofol, fentanyl, rocuronium. Maintenance: Sevoflurane, remifentanil.

Intervention: Propofol

Propofol

Induction: Propofol, fentanyl, rocuronium. Maintenance: Sevoflurane, remifentanil.

Intervention: Sevoflurane

Propofol

Induction: Propofol, fentanyl, rocuronium. Maintenance: Sevoflurane, remifentanil.

Intervention: Remifentanil

Propofol

Induction: Propofol, fentanyl, rocuronium. Maintenance: Sevoflurane, remifentanil.

Intervention: Fentanyl

Propofol

Induction: Propofol, fentanyl, rocuronium. Maintenance: Sevoflurane, remifentanil.

Intervention: Rocuronium

Remimazolam 6 mg/kg/hr

Induction: Remimazolam 6 mg/kg/hr, fentanyl, rocuronium. Maintenance: Remimazolam up to 2 mg/kg/hr titrated to effect, remifentanil.

Intervention: Remimazolam

Remimazolam 6 mg/kg/hr

Induction: Remimazolam 6 mg/kg/hr, fentanyl, rocuronium. Maintenance: Remimazolam up to 2 mg/kg/hr titrated to effect, remifentanil.

Intervention: Remifentanil

Remimazolam 6 mg/kg/hr

Induction: Remimazolam 6 mg/kg/hr, fentanyl, rocuronium. Maintenance: Remimazolam up to 2 mg/kg/hr titrated to effect, remifentanil.

Intervention: Fentanyl

Remimazolam 6 mg/kg/hr

Induction: Remimazolam 6 mg/kg/hr, fentanyl, rocuronium. Maintenance: Remimazolam up to 2 mg/kg/hr titrated to effect, remifentanil.

Intervention: Rocuronium

Remimazolam 12 mg/kg/hr

Induction: Remimazolam 12 mg/kg/hr, fentanyl, rocuronium. Maintenance: Remimazolam up to 2 mg/kg/hr titrated to effect, remifentanil.

Intervention: Remimazolam

Remimazolam 12 mg/kg/hr

Induction: Remimazolam 12 mg/kg/hr, fentanyl, rocuronium. Maintenance: Remimazolam up to 2 mg/kg/hr titrated to effect, remifentanil.

Intervention: Remifentanil

Remimazolam 12 mg/kg/hr

Induction: Remimazolam 12 mg/kg/hr, fentanyl, rocuronium. Maintenance: Remimazolam up to 2 mg/kg/hr titrated to effect, remifentanil.

Intervention: Fentanyl

Remimazolam 12 mg/kg/hr

Induction: Remimazolam 12 mg/kg/hr, fentanyl, rocuronium. Maintenance: Remimazolam up to 2 mg/kg/hr titrated to effect, remifentanil.

Intervention: Rocuronium

Outcomes

Primary Outcomes

Proportion of patients with successful anesthesia

Time Frame: Between the start of study medication and the end of the surgical procedure (up to approx 12 hours)

Successful anesthesia was defined as no use of rescue sedative medication between start of the study medication and end of the surgical procedure completion of last skin suture.

Study Sites (1)

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