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Local Anesthetic Properties of Neosaxitoxin

Phase 1
Completed
Conditions
Healthy Volunteers
Registration Number
NCT00273065
Lead Sponsor
University of Chile
Brief Summary

The purpose of this study is to evaluate the local anesthetic properties of neosaxitoxin in humans

Detailed Description

Neosaxitoxin is a phycotoxins that reversible block the voltage-gated sodium channels at neuronal level. Its activity is express as blocking the axonal conduction, stopping the propagation of the nerve impulse. The objective of the present work is to evaluate the neosaxitoxin efficacy and safety as local anesthetic in a human trial

Methods: Randomized, double-blind, placebo-controlled trial, with 10 healthy volunteers. The anesthetic effect will be evaluated using a standardized human sensory and pain model. TSA Neurosensory analyser and Von Frey Technique will be used to evaluate five parameters: sensory threshold for warm and cold, pain thresholds for heat and cold and mechanical touch perception threshold.

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
10
Inclusion Criteria
  • Healthy males with the abilities to understand and respond the tests to perform
Exclusion Criteria
  • Use of any oral analgesics at least ten days before the study
  • Drugs abuse history
  • Showing at the clinical examination any signal of psychiatric disorder

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Primary Outcome Measures
NameTimeMethod
Neural blockade of five parameters:
sensory threshold for warm
sensory threshold for cold
pain thresholds for heat
pain thresholds for cold
mechanical touch perception threshold
Measurements at 1,3,6,9,12,16,24 and 48 hrs after the injections
Secondary Outcome Measures
NameTimeMethod
Pain on injection (VAS Score 0-10)
Blood sample at 1 hour
Orine sample at 4 hours after the injection, in order to determine amounts of neosaxitoxin

Trial Locations

Locations (1)

Henry Mayer Center, Hospital Clínico Universidad de Chile

🇨🇱

Santiago, Chile

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