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Telitacicept for the Treatment of Connective Tissue Disease-associated Thrombocytopenia

Phase 2
Recruiting
Conditions
Connective Tissue Diseases
Thrombocytopenia
Interventions
Registration Number
NCT05998759
Lead Sponsor
Beijing Hospital
Brief Summary

The goal of this clinical trial is to evaluate the efficacy and safety of Telitacicept for the treatment of connective tissue disease-associated thrombocytopenia.

Detailed Description

In this randomized, double-blind placebo-controlled study, the investigators aim to evaluate the efficacy and safety of Telitacicept for the treatment of connective tissue disease-associated thrombocytopenia. After screening, eligible participants will be randomized at a 1: 1 ratio to receive either subcutaneous Telitacicept 160 mg or placebo once a week for 24 weeks. The background standard therapy is maintained stable during the whole treatment period.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
296
Inclusion Criteria
  • Subjects who have been diagnosed with connective tissue disease (CTD)-associated thrombocytopenia. And CTD includes primary Sjögren syndrome (according to the 2002 American College of Rheumatology (ACR)/ European League against Rheumatism (EULAR) classification criteria), systemic lupus erythematosus (SLE, according to the 1997 or the 2009 ACR classification criteria), and undifferentiated connective tissue disease (according to the 1999 international classification criteria)
  • Refractory thrombocytopenia defined as:

Either: Failure to maintain sustained remission after treatment by glucocorticoid and at least one immunosuppressant (i.e. cyclophosphamide, cyclosporine, mycophenolate mofetil, azathioprine, tacrolimus, methotrexate, leflunomide and hydroxychloroquine, et al.) Or: Relapse during oral glucocorticoid tapering or after withdrawal

  • 50×10^9/L>PLT
  • anti-nuclear antibody (ANA) positive (≥1:80, any karyotype) detected in the laboratory of each research center
  • Standard therapy should be maintained stable for at least 14 days prior to the first dose of the experimental drug or placebo. Standard therapy refers to the following treatment (monotherapy or in combination): glucocorticoid, hydroxychloroquine, and other immunosuppressants (i.e. cyclophosphamide, cyclosporine, mycophenolate mofetil, azathioprine, tacrolimus, methotrexate and leflunomide, et al.)
  • Signed informed consent form, willing or able to participate in all required study evaluations and procedures
Exclusion Criteria
  • Vital organ lethal bleeding (including but not limited to central nervous system bleeding, digestive tract bleeding) at screening, or intracranial bleeding 6 months prior to screening
  • Antiphospholipid syndrome, thrombotic thrombocytopenia purpura, hemolytic uremic syndrome, or thrombocytopenia secondary to other causes (such as sepsis, Epstein-Barr virus infection, cytomegalovirus infection, Corona Virus Disease-19 (COVID-19) infection, drugs, etc.)
  • Hematopoietic system disorders, such as myelodysplastic syndrome, paroxysmal sleep hemoglobinuria, aplastic anemia, leukemia, lymphoma, myelofibrosis and so on
  • Severe cardiovascular system disease, including: unstable or uncontrollable disease or condition affecting the function of the heart (such as angina pectoris, congestive heart failure, uncontrolled hypertension or arrhythmia)
  • Arteriovenous thromboembolism events
  • Receiving antiplatelet or anticoagulant therapy at screening
  • Clinically significant electrocardiogram changes
  • corrected Q-T interval (QTc)>450ms for male, QTc>470ms for female
  • Severe pulmonary disease, including: unstable or uncontrollable disease or condition affecting respiratory function [e.g., diffuse alveolar hemorrhage, severe pulmonary hypertension, severe pulmonary interstitial disease (peripheral blood oxygen saturation <92% at rest without oxygen, or forced vital capacity (FVC)<50%, or carbon monoxide diffusing capacity (DLCO)<50%)]
  • Severe kidney disease, including: severe lupus nephritis (urinary protein > 6 g/24 hours or endogenous creatinine clearance < 30 ml /min) 8 weeks prior to randomization, active nephritis requiring current protocol disallowed drugs, severe renal insufficiency requiring hemodialysis or prednisone ≥100mg/ day (or equivalent) for ≥14 days
  • SLE or non-SLE related central nervous system disease (including epilepsy, psychosis, organic encephalopathy syndrome, cerebrovascular accident, encephalitis, central nervous system vasculitis) 8 weeks prior to randomization
  • Active hepatitis, a history of severe liver disease. Subjects positive for hepatitis B surface antigen (HBsAg) or antibodies to hepatitis C virus are excluded. As for subjects with antibodies to hepatitis B core antigen (HBcAb), further hepatitis B virus (HBV)-DNA should be tested. If HBV-DNA is negative, subjects could be enrolled; otherwise, subjects should be excluded
  • Abnormal laboratory results (including but not limited to: alanine aminotransferase (ALT) or aspertate aminotransferase (AST)≥3×ULN (upper limit of normal), white blood cell count <1.5×10^9/L)
  • Subjects with known active infections (e.g., shingles, COVID-19, HIV, active tuberculosis, etc.), and active or recurrent gastrointestinal ulcers
  • Pregnant or lactating women, and subjects with a during plan during the trial
  • Allergic reaction: history of allergic reactions to human biological products
  • Treatment with B cell-targeting agents such as Rituximab or Epratuzumab or Belimumab six months prior to randomization
  • Treatment with tumor necrosis factor (TNF) inhibitors or TNF-receptor blockers six months prior to randomization
  • Participating in clinical trial 28 days or 5 drug half-lives of the investigational agents prior to randomization
  • Received live vaccine 28 days prior to randomization
  • Treatment with unstable dosage of thrombopoietin receptor agonists such as Eltrombopag or Romiplostim 14 days prior to randomization
  • Subjects with depression or suicidal thoughts
  • Previous treatment with telitacicept
  • B cell targeting drug therapy is not tolerated or responsive
  • Investigator considers candidates not appropriating for the study

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Placebo plus standard therapyPlaceboPlacebo combined with standard therapy. Standard therapy refers to the following treatment (monotherapy or in combination): glucocorticoid, hydroxychloroquine, and other immunosuppressants (i.e. cyclophosphamide, cyclosporine, mycophenolate mofetil, azathioprine, tacrolimus, methotrexate and leflunomide, et al.).
Telitacicept plus standard therapyTelitaciceptTelitacicept (160mg ih qw for 24 weeks) combined with standard therapy. Standard therapy refers to the following treatment (monotherapy or in combination): glucocorticoid, hydroxychloroquine, and other immunosuppressants (i.e. cyclophosphamide, cyclosporine, mycophenolate mofetil, azathioprine, tacrolimus, methotrexate and leflunomide, et al.).
Primary Outcome Measures
NameTimeMethod
Overall response (CR + PR) rateat week 24

Response is deemed as complete (CR) if the platelet (PLT) count is ≥ 100×10\^9/L, partial (PR) if the platelet count ranges from 50×10\^9/L to 100×10\^9/L and at least doubled from baseline. No active bleeding is allowed in participants classified as CR or PR.

Secondary Outcome Measures
NameTimeMethod
Overall response (CR + PR) rateat week 12

Response is deemed as complete (CR) if the platelet count is ≥ 100×10\^9/L, partial (PR) if the platelet count ranges from 50×10\^9/L to 100×10\^9/L and at least doubled from baseline. No active bleeding is allowed in participants classified as CR or PR.

Rescue treatment rateat week 24

Rescue treatment is initiated if the platelet count is \<10×10\^9/L, or the participant is with active bleeding, or based on the investigator's judgement when the platelet count ranges from 10×10\^9/L to 30×10\^9/L.

Time to rescue treatmentat week 24

Time to rescue treatment refers to period duration from the initiation of Telitacicept or placebo (day 1) to rescue treatment.

Relapse rateat week 24

No response refers to the platelet count is \< 50×10\^9/L, or increases for less than 1-fold from baseline, or with active central nervous system or digestive tract bleeding, or rescue treatment is initiated. Relapse is defined as no response recurring after a complete or partial response lasting for at least 7 days with treatment.

Time to relapseat week 24

Time to relapse refers to period duration from the initiation of Telitacicept or placebo (day 1) to relapse.

treatment related adverse eventat week 24

According to the NCI CTCAE 5.0

treatment related severe adverse eventat week 24

According to the NCI CTCAE 5.0

bleeding scaleat week 24

According to the ITP bleeding scale (IBLS). The IBLS comprises of 11 grades from 0 (none) to 2 (marked bleeding) by history over the previous week or by exam; 2 being worse. These 11 grades include: skin by physical exam, oral by physical exam, skin by history, oral by history, epistaxis, gastrointestinal, urinary, gynecological, pulmonary, intracranial hemorrhage, and subconjunctival hemorrhage.

Trial Locations

Locations (23)

The First Affiliated Hospital of Anhui Medical College

🇨🇳

Hefei, Anhui, China

The First Affiliated Hospital of China University of Science and Technology (Anhui Provincial)

🇨🇳

Hefei, Anhui, China

Beijing Hospital

🇨🇳

Beijing, Beijing, China

Peking University People's Hospital

🇨🇳

Beijing, Beijing, China

Peking University Third Hospital

🇨🇳

Beijing, Beijing, China

First Affiliated Hospital, Sun Yat-Sen University

🇨🇳

Guangzhou, Guangdong, China

Guangdong Provincial People's Hospital

🇨🇳

Guangzhou, Guangdong, China

The First Affiliated Hospital of Zhengzhou University

🇨🇳

Zhengzhou, Henan, China

Wuhan Union Hospital, China

🇨🇳

Wuhan, Hubei, China

Second Xiangya Hospital of Central South University

🇨🇳

Changsha, Hunan, China

Xiangya Hospital of Central South University

🇨🇳

Changsha, Hunan, China

The Affiliated Hospital of Inner Mongolia Medical University

🇨🇳

Hohhot, Inner Mongolia Autonomous Region, China

First Hospital of China Medical University

🇨🇳

Shenyang, Liaoning, China

Shandong Provincial Hospital

🇨🇳

Jinan, Shandong, China

Changhai Hospital

🇨🇳

Shanghai, Shanghai, China

RenJi Hospital

🇨🇳

Shanghai, Shanghai, China

Shanxi Bethune Hospital

🇨🇳

Taiyuan, Shanxi, China

West China Hospital

🇨🇳

Chengdu, Sichuan, China

Institute of Hematology & Blood Diseases Hospital

🇨🇳

Tianjin, Tianjin, China

Tianjin First Central Hospital

🇨🇳

Tianjin, Tianjin, China

Tianjin Medical University General Hospital

🇨🇳

Tianjin, Tianjin, China

People's Hospital of Xinjiang Uygur Autonomous Region

🇨🇳

Ürümqi, Xinjiang Uygur Autonomous Region, China

The First People's Hospital of Yunnan

🇨🇳

Kunming, Yunnan, China

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