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An Exploratory Trial to Assess the Improvement of Adverse Events in Chronic Myelogenous Leukemia Patients Treated With Imatinib When Switched to Nilotinib Treatment

Phase 4
Completed
Conditions
Chronic Myelogenous Leukemia
Interventions
Registration Number
NCT00980018
Lead Sponsor
Novartis Pharmaceuticals
Brief Summary

The purpose of this exploratory study will be to examine changes in chronic low grade chronic adverse events, measured by Common Terminology Criteria for Adverse Events (CTCAE) grading, when patients are switched from imatinib to nilotinib therapy.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
52
Inclusion Criteria
  1. Male or female patients ≥ 18 years of age
  2. Eastern Cooperative Oncology Group (ECOG) 0, 1, or 2
  3. Diagnosis of CML-CP associated with Bcr-Abl quantifiable by RQ-PCR (IS)
  4. Patients must be an imatinib responder and achieved the following efficacy milestones as appropriate for the length of time on imatinib therapy as per protocol
  5. CML-CP patients initiated on any dose of imatinib
  6. Ability to provide written informed consent prior to any study related screening procedures being done
Exclusion Criteria
  1. Loss of CHR or cytogenetic response
  2. Prior accelerated phase or blast phase CML
  3. Previously documented T315I mutation
  4. Presence of chromosomal abnormalities (trisomy 8) and/or clonal evolution other than Ph+.
  5. Previous treatment with any other tyrosine kinase inhibitor except for imatinib.
  6. Treatment with other investigational agents within 30 days of Day 1.
  7. History of non-compliance to medical regimens or inability to grant consent.
  8. Women who are pregnant, breast feeding, or of childbearing potential without a negative serum test at baseline. Male or female patients of childbearing potential unwilling to use contraceptive precautions throughout the trial and 3 months following discontinuation of study drug. Post-menopausal women must be amenorrheic for at least 12 months to be considered of non-childbearing potential. Women of childbearing potential must have a negative serum pregnancy test prior to the first dose of nilotinib.

Other protocol-defined inclusion/exclusion criteria may apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
nilotinibNilotinibParticipants received two 150 \[a total of 300 mg at each dosing\] mg nilotinib capsules twice daily (bid) orally every morning and every evening approximately 12 hours apart and two 200 mg capsules \[a total of 400 mg at each dosing\] for patients enrolled prior to Protocol Amendment 1).
Primary Outcome Measures
NameTimeMethod
Percentage of Participants With Improvement in Imatinib Related Chronic Low Grade Non Hematologic Adverse Event (AE) After Switch to Treatment With Nilotinib at End of Cycle 3End of Cycles 1, 2, and 3

A patient was considered improved if 50% or more of the chronic imatinib-related chronic low grade nonhematologic AEs showed improvement (a decrease in CTCAE \[Common Terminology Criteria for Adverse Events\] grade or complete resolution).

Secondary Outcome Measures
NameTimeMethod
Percentage of Participants Achieving Complete Cytogenetic Response (CCyR) After Switching to Nilotinib for Participants Not Reporting CCyR at BaselineCycles 1, 2, 6, 9, and 12

Time to complete cytogenetic response is defined as time from baseline to first time of CCyR as documented by bone marrow cytogenetics. Cytogenetic response was assessed as applicable by bone marrow cytogenetics 6, 12, and 18 months after starting imatinib therapy. Assess CCyR by bone marrow cytogenics

Duration of Complete Cytogenetic Response18 months of follow up from the first documented response

Duration of Complete Cytogenetic Response is defined as the time from first CCyR to first loss of CCyR as documented by bone marrow cytogenetics, or by FISH assay, whichever is earlier. The duration of CCyR begins on the day of enrollment for patients reporting CCyR at baseline.

Time to Optimal Imatinib-related Adverse Event Improvement18 months of follow up from the date of the first dose of study drug to the time to maximum decrease in CTCAE grade of these events

Time to optimal improvement is defined as the time when the sum of the total CTCAE toxicity grades for a patient's chronic low-grade imatinib-related adverse events reaches its minimum value.

Percentage of Participants Achieving Major Molecular Response (MMR) After the Switch in the Therapy for Participants Not Reporting MMR at BaselineCycles 1,2,3,6,9,12

Major Molecular Response (MMR) value at Molecular MD is designated a percentage, which is equivalent to a 3-log reduction from a standardized baseline value from the International Randomized Interferon versus STI571 (IRIS) study or 0.1% per International Scale (IS). Time to MMR is defined as time from baseline to first time of MMR as documented by RQ-PCR

Log Change in BCR-Abl Transcript Level From Baseline After the Switch TherapyCycles 1,2,3,6,9, and 12

Levels of BCR-ABL transcripts were determined by quantitative RQ-PCR testing of peripheral blood and analyzed at a central testing laboratory. Log reduction in BCR-ABL transcripts levels from the standardized baseline value will be calculated for each sample from the reported percent ratio of BCR-ABL transcripts versus control gene transcripts converted to a reference standard.

Time to Major Molecular Response (MMR) in Participants With MMR Absent at BaselineCycles 1,2,3,6,9,12

For time to MMR, an event is defined as achievement of MMR documented by RQ-PCR. Patients with MMR at the Screening RQ-PCR assay are counted as having time to MMR equal to 0.

Time to Complete Cytogenetic Response in Participants Not Reporting at BaselineCycle 12

For time to CCyR, an event is defined as achievement of CCyR documented by bone marrow cytogenetics.

Duration of Major Molecular Response18 months of follow up from the first documented response

Duration of Major Molecular Response is defined as the time from first MMR to first loss of MMR as documented by RQ-PCR. The duration of MMR begins on the day of enrollment for patients reporting MMR at baseline.

Trial Locations

Locations (20)

Presbyterian Hospital of Dallas TexasOncology@PresbyterianHosp

🇺🇸

Dallas, Texas, United States

Texas Oncology Texas Oncology - Sugar Land

🇺🇸

Dallas, Texas, United States

Rocky Mountain Cancer Centers RMCC - Aurora

🇺🇸

Greenwood Village, Colorado, United States

USC Norris Cancer Center LAC & USC Medical Center

🇺🇸

Los Angeles, California, United States

Highlands Oncology Group

🇺🇸

Fayetteville, Arkansas, United States

Hematology Oncology Services of Arkansas SC

🇺🇸

Little Rock, Arkansas, United States

Southwest Cancer Care Murrieta

🇺🇸

Poway, California, United States

Florida Cancer Institute

🇺🇸

New Port Richey, Florida, United States

St. Louis University Cancer Center

🇺🇸

Saint Louis, Missouri, United States

Stroger Cook County Hospital John H. Stroger Hospital

🇺🇸

Chicago, Illinois, United States

Cancer Centers of Florida PA Cancer Centers of FL-Orlando-4

🇺🇸

Ocoee, Florida, United States

St. Agnes Hospital

🇺🇸

Baltimore, Maryland, United States

St. Francis Hospital and Health Centers IndianaBlood&MarrowTransplantn

🇺🇸

Beech Grove, Indiana, United States

Northwest Cancer Specialists Salmon Creek Office

🇺🇸

Portland, Oregon, United States

Oregon Health Sciences University

🇺🇸

Portland, Oregon, United States

The Jones Clinic

🇺🇸

Germantown, Tennessee, United States

Texas Oncology, P.A.

🇺🇸

Bedford, Texas, United States

Cancer Care Centers of South Texas / HOAST CCC of So. TX- San Antonio(2)

🇺🇸

San Antonio, Texas, United States

MD Anderson Cancer Center/University of Texas

🇺🇸

Houston, Texas, United States

Novartis Investigative Site

🇨🇦

Montreal, Quebec, Canada

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