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Safety, Tolerability, and Activity of ISIS 113715 in People With Type 2 Diabetes Mellitus Who Have Not Received Prior Treatment

Phase 2
Completed
Conditions
Type 2 Diabetes Mellitus
Registration Number
NCT00330330
Lead Sponsor
Ionis Pharmaceuticals, Inc.
Brief Summary

The aim of this study is to evaluate the safety, tolerability, and pharmacokinetics of five ISIS 113715 intravenous dose cohorts in drug-naïve type 2 diabetics.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
96
Inclusion Criteria
  • Type 2 Diabetes Mellitus of less than 5 years in duration
  • Have never received hypoglycemic therapy
  • Aged 18 to 65 years
  • Fasting blood glucose between 130 and 220 mg/dL (7.2 to 12.2 mmol/L) for Cohorts A-D and between 140 and 220 mg/dL (7.8 to 12.2 mmol/L) for Cohort E
  • HbA1c between 6.8 and 10.0% for Cohorts A-D and between 7.5 and 11.0% for Cohort E
  • Body Mass index > 25 and < 35 kg m -2
Exclusion Criteria
  • Medication that may affect glucose homeostasis (e.g. systemic glucocorticoid) within one month of screening
  • Clinically significant abnormalities in medical history or physical exam
  • Clinically significant abnormalities on laboratory examination
  • History of HIV infection
  • Active infection requiring antiviral or antimicrobial therapy
  • Malignancy (with the exception of basal or squamous cell carcinoma of the skin if adequately treated and no recurrence for > one year at the time of screening)
  • Any other concurrent condition which, in the opinion of the Investigator, would preclude participation in or interfere with compliance
  • Alcohol or drug abuse
  • Undergoing or have undergone treatment with another investigational drug, biologic agent or device within 90 days of screening
  • Abnormal serum creatinine concentration defined as > 1.5 mg/dL (132.6 micro mol/L) for males and > 1.2 mg/dL (106 micro mol/L) for females
  • Medications that may affect coagulation (heparin, warfarin, etc.) with the exception of acetylsalicylic acid or non-steroidal anti-inflammatory agents.
  • Allergy to sulfur-containing medications

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Primary Outcome Measures
NameTimeMethod
To evaluate the pharmacokinetic profile of ISIS 113715
To evaluate the safety and tolerability of ISIS 113715
To evaluate the pharmacologic activity of ISIS 113715
Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (10)

Close Corporation "MEDSI"

🇷🇺

Moscow, Russian Federation

NZOZ Specjalistyczny Osrodek Internistyczno Diabetologiczny

🇵🇱

Bialystok, Poland

Prywatna Praktyka Lekarska

🇵🇱

Radom, Poland

Clinic of Therapy of Postgraduate Education named after N.S. Molchanov

🇷🇺

St. Petersburg, Russian Federation

Oddzial Chorob Wewnetrznych ze Stacja Dializ Szpital w Wolominie

🇵🇱

Wolomin, Poland

Chair of Endocrinology and Diabetology of the Faculty of Advenced Training for Physicians

🇷🇺

Moscow, Russian Federation

Endocrinology Scientific Centre of RAMS

🇷🇺

Moscow, Russian Federation

Medical Institution "Polyclinic OAOA Gazprom"

🇷🇺

Moscow, Russian Federation

Moscow Regional Scientific-Research Clinical Institute named after I.F. Vladimirsky

🇷🇺

Moscow, Russian Federation

Chair of Endocrinology and Diabetology Central Clinical Hospital of the Ministry of Communications of RF

🇷🇺

Moscow, Russian Federation

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