MedPath

A Study of AV-101 (Dry Powder Inhaled Imatinib) in Patients With Pulmonary Arterial Hypertension (PAH)

Phase 2
Terminated
Conditions
Pulmonary Arterial Hypertension
Interventions
Drug: Placebo
Registration Number
NCT05036135
Lead Sponsor
Aerovate Therapeutics
Brief Summary

IMPAHCT: Inhaled iMatinib Pulmonary Arterial Hypertension Clinical Trial is a Phase 2b/Phase 3 study to evaluate the safety and efficacy of AV-101 (dry powder inhaled imatinib) in patients with Pulmonary Arterial Hypertension (PAH). The Phase 2b part of the study will assess three doses to establish an optimal dose for the Phase 3 part of the study. The Phase 2b primary endpoint will be the placebo corrected change in pulmonary vascular resistance (PVR). The Phase 3 primary endpoint will be the placebo corrected change in 6-minute walk distance (6MWD) after 24 weeks of treatment.

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
202
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
AV-101 10 mgAV-101-
AV-101 35 mgAV-101-
PlaceboPlacebo-
AV-101 70 mgAV-101-
Primary Outcome Measures
NameTimeMethod
Phase 2b: Change from Baseline in Pulmonary Vascular Resistance (PVR)24 weeks
Phase 3: Change from Baseline in Six Minute Walk Distance (6MWD)24 weeks
Secondary Outcome Measures
NameTimeMethod
Phase 2b: Change from Baseline in Six Minute Walk Distance (6MWD)24 weeks
Phase 2b: Time to Clinical Worsening24 weeks
Phase 2b: Change from Baseline in Registry to Evaluate Early and Long-Term PAH Disease Management (REVEAL) Lite 2.0 Risk Score24 weeks

REVEAL Lite 2.0 risk scores range from 1 to 14; a higher score represents higher risk

Phase 2b: Change from Baseline in N-terminal pro B-type natriuretic peptide (NT-proBNP)24 weeks
Phase 2b: Proportion of Subjects with Improvement in WHO Functional Class24 weeks
Phase 2b: Change from Baseline in Health-Related Quality of Life emPHasis-10 Questionnaire Score24 weeks

emPHasis-10 questionnaire scores range from 0 - 50; a higher score represents a higher symptom burden

Phase 3: Change from Baseline in NT-proBNP24 weeks
Phase 3: Time to Clinical Worsening24 weeks
Phase 3: Proportion of Subjects with Improvement in WHO Functional Class24 weeks
Phase 3: Change from Baseline in Registry to Evaluate Early and Long-Term PAH Disease Management (REVEAL) Lite 2.0 Risk Score24 weeks

REVEAL Lite 2.0 risk scores range from 1 to 14; a higher score represents higher risk

Phase 3: Change from Baseline in Pulmonary Arterial Hypertension-Symptoms and Impact (PAH-SYMPACT) Questionnaire Score24 weeks

PAH-SYMPACT is a patient reported outcome instrument developed to assess PAH symptoms and impacts

Trial Locations

Locations (128)

Tufts Medical Center, Inc.

๐Ÿ‡บ๐Ÿ‡ธ

Boston, Massachusetts, United States

AHEPA General Hospital of Thessaloniki

๐Ÿ‡ฌ๐Ÿ‡ท

Thessalonรญki, Greece

University of Minnesota

๐Ÿ‡บ๐Ÿ‡ธ

Minneapolis, Minnesota, United States

Duke University Medical Center - Duke South Clinic

๐Ÿ‡บ๐Ÿ‡ธ

Durham, North Carolina, United States

Vanderbilt University Medical Center

๐Ÿ‡บ๐Ÿ‡ธ

Nashville, Tennessee, United States

UCLA/David Geffen School of Medicine-Pulmonary and Criticial Care

๐Ÿ‡บ๐Ÿ‡ธ

Los Angeles, California, United States

Arizona Pulmonary Specialists, Ltd.

๐Ÿ‡บ๐Ÿ‡ธ

Phoenix, Arizona, United States

Cedars-Sinai Medical Center, Pulmonary & Critical Care

๐Ÿ‡บ๐Ÿ‡ธ

Los Angeles, California, United States

Dept of Veterans Affairs Greater Los Angeles Healthcare System

๐Ÿ‡บ๐Ÿ‡ธ

Los Angeles, California, United States

University of California

๐Ÿ‡บ๐Ÿ‡ธ

San Francisco, California, United States

George Washington University Medical Faculty Associates, Inc.

๐Ÿ‡บ๐Ÿ‡ธ

Washington, District of Columbia, United States

Indiana University Health

๐Ÿ‡บ๐Ÿ‡ธ

Indianapolis, Indiana, United States

The Unviersity of New Mexico - UNM Hospitals

๐Ÿ‡บ๐Ÿ‡ธ

Albuquerque, New Mexico, United States

New York-Presbyterian Brooklyn Methodist Hospital

๐Ÿ‡บ๐Ÿ‡ธ

Brooklyn, New York, United States

The Lindner Center for Research and Education

๐Ÿ‡บ๐Ÿ‡ธ

Cincinnati, Ohio, United States

University of Cincinnati

๐Ÿ‡บ๐Ÿ‡ธ

Cincinnati, Ohio, United States

Stat Care Pulmonary Consultants, PLLC

๐Ÿ‡บ๐Ÿ‡ธ

Knoxville, Tennessee, United States

Sentara Medical Group - Sentara Pulmonary & Critical Care Specialists

๐Ÿ‡บ๐Ÿ‡ธ

Norfolk, Virginia, United States

Houston Methodist Hospital

๐Ÿ‡บ๐Ÿ‡ธ

Houston, Texas, United States

Hospital Britanico de Buenos Aires

๐Ÿ‡ฆ๐Ÿ‡ท

Buenos Aires, Argentina

Hospital Dr. Jose Maria Cullen

๐Ÿ‡ฆ๐Ÿ‡ท

Santa Fe, Argentina

Concord Repatriation General Hospital

๐Ÿ‡ฆ๐Ÿ‡บ

Concord West, New South Wales, Australia

Nepean Hospital

๐Ÿ‡ฆ๐Ÿ‡บ

Kingswood, New South Wales, Australia

Westmead Hospital

๐Ÿ‡ฆ๐Ÿ‡บ

Westmead, New South Wales, Australia

Washington University School of Medicine

๐Ÿ‡บ๐Ÿ‡ธ

Saint Louis, Missouri, United States

Sunshine Coast University Hospital

๐Ÿ‡ฆ๐Ÿ‡บ

Birtinya, Queensland, Australia

The Prince Charles Hospital

๐Ÿ‡ฆ๐Ÿ‡บ

Chermside, Queensland, Australia

Fiona Stanley Hospital

๐Ÿ‡ฆ๐Ÿ‡บ

Murdoch, Australia

The Alfred Hospital

๐Ÿ‡ฆ๐Ÿ‡บ

Melbourne, Victoria, Australia

AKH - Medizinische Universitat Wien

๐Ÿ‡ฆ๐Ÿ‡น

Vienna, Austria

Hopital Erasme - Cliniques Universitaires de Bruxelles

๐Ÿ‡ง๐Ÿ‡ช

Brussels, Belgium

The Governors of the University of Calgary

๐Ÿ‡จ๐Ÿ‡ฆ

Calgary, Alberta, Canada

Santa Casa de Misericordia de Porto Alegre

๐Ÿ‡ง๐Ÿ‡ท

Porto Alegre, Brazil

UZ Leuven

๐Ÿ‡ง๐Ÿ‡ช

Leuven, Belgium

Heart Institute - University of Sao Paulo

๐Ÿ‡ง๐Ÿ‡ท

Sรฃo Paulo, Brazil

London Health Science Centre

๐Ÿ‡จ๐Ÿ‡ฆ

London, Ontario, Canada

Jewish General Hospital

๐Ÿ‡จ๐Ÿ‡ฆ

Montrรฉal, Quebec, Canada

Centro de Investigaciones Clinicas de la Universidad Catolica

๐Ÿ‡จ๐Ÿ‡ฑ

Santiago, Chile

Peking Union Medical College Hospital

๐Ÿ‡จ๐Ÿ‡ณ

Beijing, China

Chongqing Medical University - The First Affiliated Hospital

๐Ÿ‡จ๐Ÿ‡ณ

Chongqing, China

Guangdong Provincial People's Hospital

๐Ÿ‡จ๐Ÿ‡ณ

Guangdong, China

Central South University - The Second Xiangya Hospital

๐Ÿ‡จ๐Ÿ‡ณ

Hunan, China

Yanan Hospital of Kunming City

๐Ÿ‡จ๐Ÿ‡ณ

Kunming, China

Gansu Provincial People's Hospital

๐Ÿ‡จ๐Ÿ‡ณ

Lanzhou, China

Tianjin Medical University General Hospital

๐Ÿ‡จ๐Ÿ‡ณ

Tianjin, China

Southeast University (SEU) - Zhongda Hospital

๐Ÿ‡จ๐Ÿ‡ณ

Nanjing, China

Shanghai Pulmonary Hospital

๐Ÿ‡จ๐Ÿ‡ณ

Shanghai, China

Vseobecna fakultni nemocnice v Praze

๐Ÿ‡จ๐Ÿ‡ฟ

Praha, Czechia

Groupement Hospitalier Sud - Hรดpital Bicรชtre

๐Ÿ‡ซ๐Ÿ‡ท

Le Kremlin-Bicรชtre, Cedex, France

Hรดpital Cardio-Vasculaire et Pneumologique Louis Pradel

๐Ÿ‡ซ๐Ÿ‡ท

Bron, France

Universitaetsklinikum Carl Gustav Carus TU Dresden

๐Ÿ‡ฉ๐Ÿ‡ช

Dresden, Germany

Hopital Arnaud de Villeneuve

๐Ÿ‡ซ๐Ÿ‡ท

Montpellier, France

Hรดpital Nord - CHU Marseille

๐Ÿ‡ซ๐Ÿ‡ท

Marseille, France

Les Hรดpitaux Universitaires de Strasbourg

๐Ÿ‡ซ๐Ÿ‡ท

Strasbourg, France

Mรผnchen Klinik Bogenhausen

๐Ÿ‡ฉ๐Ÿ‡ช

Mรผnchen, Germany

University General Hospital Attikon

๐Ÿ‡ฌ๐Ÿ‡ท

Athens, Greece

Cardiosurgery Hospital

๐Ÿ‡ฌ๐Ÿ‡ท

Kallithรฉa, Greece

Hadassah University Hospital - Ein Kerem

๐Ÿ‡ฎ๐Ÿ‡ฑ

Jerusalem, Israel

Azienda Ospedaliero Universitaria Ospedali Riuniti - Foggia

๐Ÿ‡ฎ๐Ÿ‡น

Foggia, Italy

Ospedale San Giuseppe - Fatebenefratelli

๐Ÿ‡ฎ๐Ÿ‡น

Milan, Italy

Tel Aviv Sourasky Medical Center

๐Ÿ‡ฎ๐Ÿ‡ฑ

Tel Aviv, Israel

Azienda Socio Sanitaria Territoriale di Monza

๐Ÿ‡ฎ๐Ÿ‡น

Monza, Italy

Azienda Ospedaliera Vincenzo Monaldi

๐Ÿ‡ฎ๐Ÿ‡น

Napoli, Italy

Fondazione IRCCS Policlinico San Matteo

๐Ÿ‡ฎ๐Ÿ‡น

Pavia, Italy

Azienda Ospedaliera Universitaria Policlinico Umberto I

๐Ÿ‡ฎ๐Ÿ‡น

Rome, Italy

Unidad de Investigacion Clinica en Medicina S.C.

๐Ÿ‡ฒ๐Ÿ‡ฝ

Monterrey, Nuevo Leรณn, Mexico

Instituto Nacional de Cardiologia Dr Ignacio Chavez Rivera

๐Ÿ‡ฒ๐Ÿ‡ฝ

Mexico City, Mexico

Universidad Autonoma de Nuevo Leon, Hospital Universitario

๐Ÿ‡ฒ๐Ÿ‡ฝ

Monterrey, Mexico

Amsterdam UMC, Locatie VUMC

๐Ÿ‡ณ๐Ÿ‡ฑ

Amsterdam, Netherlands

Uniwersytecki Szpital Kliniczny im. Jana Mikulicza-Radeckiego

๐Ÿ‡ต๐Ÿ‡ฑ

Wrocล‚aw, Poland

Krakowski Szpital Specjalistyczny im. Jana Pawla II

๐Ÿ‡ต๐Ÿ‡ฑ

Krakow, Poland

Szpital Kliniczny Przemienienia Paล„skiego UM im. Marcinkowskiego

๐Ÿ‡ต๐Ÿ‡ฑ

Poznaล„, Poland

Hospital Pulido Valente

๐Ÿ‡ต๐Ÿ‡น

Lisboa, Portugal

Bieganski Provincial Specialist Hospital

๐Ÿ‡ต๐Ÿ‡ฑ

ลรณdลบ, Poland

Hospital Garcia de Orta, EPE

๐Ÿ‡ต๐Ÿ‡น

Almada, Portugal

Cardiopulmonary Research Center

๐Ÿ‡ต๐Ÿ‡ท

Guaynabo, Puerto Rico

CHUPorto

๐Ÿ‡ต๐Ÿ‡น

Porto, Portugal

National University Hospital

๐Ÿ‡ธ๐Ÿ‡ฌ

Singapore, Singapore

Tan Tock Seng Hospital

๐Ÿ‡ธ๐Ÿ‡ฌ

Singapore, Singapore

Hospital Universitari Vall d'Hebron

๐Ÿ‡ช๐Ÿ‡ธ

Barcelona, Spain

Center of Chest Disease Johannesburg

๐Ÿ‡ฟ๐Ÿ‡ฆ

Johannesburg, South Africa

Hosp. Universitario Gran Canaria Doctor Negrin

๐Ÿ‡ช๐Ÿ‡ธ

Las Palmas de Gran Canaria, Spain

Hospital Universitario de Toledo

๐Ÿ‡ช๐Ÿ‡ธ

Toledo, Spain

Hospital universtario de Salamanca

๐Ÿ‡ช๐Ÿ‡ธ

Salamanca, Spain

Hosp. Universitario Marques de Valdecilla

๐Ÿ‡ช๐Ÿ‡ธ

Santander, Spain

Norrlands Universitetssjukhus

๐Ÿ‡ธ๐Ÿ‡ช

Umeรฅ, Sweden

Golden Jubilee National Hospital

๐Ÿ‡ฌ๐Ÿ‡ง

Glasgow, United Kingdom

The Newcastle upon Tyne Hospitals NHS Foundation Trust

๐Ÿ‡ฌ๐Ÿ‡ง

Newcastle, United Kingdom

National Jewish Health

๐Ÿ‡บ๐Ÿ‡ธ

Denver, Colorado, United States

University of Nebraska Medical Center- Hematology/Oncology Section

๐Ÿ‡บ๐Ÿ‡ธ

Omaha, Nebraska, United States

Hospital Clinic de Barcelona

๐Ÿ‡ช๐Ÿ‡ธ

Barcelona, Spain

Hospital 12 de Octubre

๐Ÿ‡ช๐Ÿ‡ธ

Madrid, Spain

Universidad Autonoma de Madrid

๐Ÿ‡ช๐Ÿ‡ธ

Madrid, Spain

Hospital Universitario Virgen de la Victoria

๐Ÿ‡ช๐Ÿ‡ธ

Mรกlaga, Spain

Universitaetsklinikum Giessen und Marburg GmbH Standort Giessen

๐Ÿ‡ฉ๐Ÿ‡ช

Giesen, Germany

Universitaetsklinikum Heidelberg

๐Ÿ‡ฉ๐Ÿ‡ช

Heidelberg, Germany

The Lady Davis Carmel Medical Center

๐Ÿ‡ฎ๐Ÿ‡ฑ

Haifa, Israel

Royal Prince Alfred Hospital

๐Ÿ‡ฆ๐Ÿ‡บ

Camperdown, New South Wales, Australia

Cardiologรญa Palermo

๐Ÿ‡ฆ๐Ÿ‡ท

Caba, Argentina

Nexo Salud Investigaciรณn Clรญnica

๐Ÿ‡ฆ๐Ÿ‡ท

Buenos Aires, Argentina

Sanatorio de la Trinidad Mitre

๐Ÿ‡ฆ๐Ÿ‡ท

Buenos Aires, Argentina

Insituto Medico DAMIC

๐Ÿ‡ฆ๐Ÿ‡ท

Cรณrdoba, Argentina

Hospital Italiano de Cordoba

๐Ÿ‡ฆ๐Ÿ‡ท

Cรณrdoba, Argentina

UC Davis Medical Center

๐Ÿ‡บ๐Ÿ‡ธ

Sacramento, California, United States

University of Colorado Denver

๐Ÿ‡บ๐Ÿ‡ธ

Aurora, Colorado, United States

Kaiser Permanente Los Angeles Medical Center

๐Ÿ‡บ๐Ÿ‡ธ

Los Angeles, California, United States

LA Biomedical Research Institute Harbor

๐Ÿ‡บ๐Ÿ‡ธ

Torrance, California, United States

Mayo Clinic Florida

๐Ÿ‡บ๐Ÿ‡ธ

Jacksonville, Florida, United States

Emory University

๐Ÿ‡บ๐Ÿ‡ธ

Atlanta, Georgia, United States

University of Iowa Hospitals & Clinics

๐Ÿ‡บ๐Ÿ‡ธ

Iowa City, Iowa, United States

NYU Langone Seaport

๐Ÿ‡บ๐Ÿ‡ธ

New York, New York, United States

The Ohio State University Wexner Medical Center

๐Ÿ‡บ๐Ÿ‡ธ

Columbus, Ohio, United States

Bend Memorial Clinic

๐Ÿ‡บ๐Ÿ‡ธ

Oregon City, Oregon, United States

Hospital of the University of Pennsylvania

๐Ÿ‡บ๐Ÿ‡ธ

Philadelphia, Pennsylvania, United States

UPMC Presbyterian Hospital

๐Ÿ‡บ๐Ÿ‡ธ

Pittsburgh, Pennsylvania, United States

Baylor University Medical Center

๐Ÿ‡บ๐Ÿ‡ธ

Dallas, Texas, United States

Royal Adelaide Hospital

๐Ÿ‡ฆ๐Ÿ‡บ

Adelaide, Australia

Istituto Mediterraneo per i Trapianti e Terapie ad Alta Specializzazione

๐Ÿ‡ฎ๐Ÿ‡น

Palermo, Italy

Orlando Heart Center

๐Ÿ‡บ๐Ÿ‡ธ

Orlando, Florida, United States

University of Michigan

๐Ÿ‡บ๐Ÿ‡ธ

Ann Arbor, Michigan, United States

Pauls Stradins Clinical University Hospital

๐Ÿ‡ฑ๐Ÿ‡ป

Riga, Latvia

CICUM San Miguel

๐Ÿ‡ฒ๐Ÿ‡ฝ

Guadalajara, Jalisco, Mexico

Imperial College Healthcare NHS Trust

๐Ÿ‡ฌ๐Ÿ‡ง

London, England, United Kingdom

University of Alberta Hospital

๐Ÿ‡จ๐Ÿ‡ฆ

Edmonton, Alberta, Canada

University of Arizona, Department of Medicine

๐Ÿ‡บ๐Ÿ‡ธ

Tucson, Arizona, United States

Royal Brompton Hospital

๐Ÿ‡ฌ๐Ÿ‡ง

London, United Kingdom

University of Kansas Medical Center

๐Ÿ‡บ๐Ÿ‡ธ

Kansas City, Kansas, United States

Thomas Jefferson University

๐Ÿ‡บ๐Ÿ‡ธ

Philadelphia, Pennsylvania, United States

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