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The Effects of Epidermal Growth Factor Receptor (EGFR) Inhibition on Pulmonary Arterial Hypertension Associated with Systemic Sclerosis A phase II controlled open-label safety and efficacy study.

Phase 2
Withdrawn
Conditions
high pulmonary vascular pressure associated with scleroderma
10019280
10010761
10037454
Registration Number
NL-OMON30491
Lead Sponsor
Vrije Universiteit Medisch Centrum
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
Withdrawn
Sex
Not specified
Target Recruitment
20
Inclusion Criteria

A subject is eligible for inclusion in this study only if all of the following criteria apply:
1. Written informed consent
2. Systemic sclerosis
3. PAH with a mean PAP of above 25 mmHg measured during rest.
4. PVR above 300 dynes
5. TLC > 70 %
6. NYHA class III and/or 6 Minute Walk Test < 80% predicted
7.Conventional PAH treatment and/or bosentan and/or sildenafil treatment
8. Stability on medication during the previous 3 months (defined as stable or decrease of 6 MWT after 3 months of treatment).

Exclusion Criteria

A subject will be excluded from this study in case of the following criteria:
1. Left ventricular dysfunction
2. Valvular heart disease
3. Pericardial constriction
4 Wedge pressure >/= 15 mmHg
5. Chronic thromboembolic pulmonary hypertension
6. Uncontrolled sleep apnea.
7. History of malignancies
8. Overt right heart failure
9. History or presence of skin ulcerations
10. Women of child-bearing potential (WOCB) who are unwilling or unable to use contraceptives
11. Sexually active fertile man not using effective birth control if their partners are WOCB
12. Severe abnormality of the cornea
13. Inadequate hematologic function defined by an absolute neutrophil count < 1,500/mm3, platelet count < 80.000/mm3 and hemoblobin level of < 9 g/dL
14.-Inadequate hepatic function defined by a total bilirubin level 1.5 times the upper limit of normal (ULN) and ASAT levels 2.5 times ULN
15. Inadequate renal function defined by a serum creatinine level > 1,5 times ULN (alternative: Cockroft <50 ml/min).
16. Substances that inhibit CYP3A4 activity, such as rifampicin, phenytoin, ketoconazole, itraconazole (see section 6.4.5)
17. Severe interstitial fibrosis on HRCT

Study & Design

Study Type
Interventional
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
<p>To describe the safety of cetuximab in scleroderma associated PAH. </p><br>
Secondary Outcome Measures
NameTimeMethod
<p>To explore the efficacy of cetuximab in terms of: stroke volume, 6 minute walk<br /><br>test, changes on HRCT, changes in nailfold microcirculation, changes in<br /><br>molecular parameters (NT-proBNP) </p><br>
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