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Effect of Combined Incretin-Based Therapy Plus Canagliflozin on Glycemic Control and the Compensatory Rise in Hepatic Glucose Production in Type 2 Diabetic Patients

Not Applicable
Completed
Conditions
Type 2 Diabetes Mellitus
Interventions
Registration Number
NCT02324842
Lead Sponsor
The University of Texas Health Science Center at San Antonio
Brief Summary

Specific Aim 1.To examine whether the combination of liraglutide plus canagliflozin can prevent the increase in Hepatic Glucose Production (HGP) following institution of canagliflozin therapy and produce an additive or even synergistic effect to lower the plasma glucose concentration and A1c.

Specific Aim 2: To examine whether combination therapy with liraglutide plus canagliflozin can produce an additive, or even synergistic, effect to promote weight loss and reduction in hepatic and visceral fat content.

Specific Aim 3. To examine whether combination therapy with liraglutide plus canagliflozin can produce an additive or even synergistic effect to reduce systolic/diastolic blood pressure and 24-hour integrated blood pressure.

Detailed Description

Specific Aim 1.To examine whether the combination of liraglutide plus canagliflozin can prevent the increase in HGP following institution of canagliflozin therapy and produce an additive or even synergistic effect to lower the plasma glucose concentration and A1c. We will examine this hypothesis by comparing the effect of administration of liraglutide alone, canagliflozin alone, and the combination of liraglutide plus canagliflozin on:(i) the rate of HGP; (ii) decrease in fasting plasma glucose concentration; (iii) counter-regulatory hormone response and (iv) A1c. We anticipate that the addition of liraglutide to canagliflozin will prevent the increase in plasma glucagon concentration, augment insulin secretion, and blunt/block the increase in HGP in response to canagliflozin, resulting in a greater decrease in fasting plasma glucose concentration and A1c than observed with each therapy alone.

Specific Aim 2: To examine whether combination therapy with liraglutide plus canagliflozin can produce an additive, or even synergistic, effect to promote weight loss and reduction in hepatic and visceral fat content.

Specific Aim 3. To examine whether combination therapy with liraglutide plus canagliflozin can produce an additive or even synergistic effect to reduce systolic/diastolic blood pressure and 24-hour integrated blood pressure.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
45
Inclusion Criteria
  • Male and female subjects between the ages of 18-70
  • Subjects with Type 2 Diabetes Mellitus (T2DM)
  • Drug naïve or on stable dose (more than 3 months) of metformin with or without sulfonylurea
  • Have an HbA1c levels ≥7.0% and <10.0%
  • Stable weight (± 3 lbs) over the preceding 3 months
Exclusion Criteria
  • Subjects taking drugs known to affect glucose metabolism (other than metformin) will be excluded.
  • Individuals with evidence of proliferative diabetic retinopathy or plasma creatinine >1.4 females or >1.5 males or estimated Glomerular Filtration Rate (eGFR)< 60 ml/min.172m2 will be excluded
  • Unstable body weight (change of greater than ±3 lbs over the preceding 3 months)
  • Participates in excessively heavy exercise program

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
CanagliflozinCanagliflozincanagliflozin (film-coated tablet), 100 mg/day, increased to 300 mg/day after week two if tolerated without side effects
liraglutideLiraglutideliraglutide, 1.2 mg/day, increased to 1.8 mg/day after week two if tolerated without side effects
canagliflozin plus liraglutideCanagliflozincanagliflozin, 100 mg/day, plus liraglutide, 1.2 mg/day, increased to 300 mg/day and 1.8 mg/day, respectively at week two, if tolerated without side effects
canagliflozin plus liraglutideLiraglutidecanagliflozin, 100 mg/day, plus liraglutide, 1.2 mg/day, increased to 300 mg/day and 1.8 mg/day, respectively at week two, if tolerated without side effects
Primary Outcome Measures
NameTimeMethod
HbA1c at 4 MonthsApproximately 4 months

Primary end point of the study is the HbA1c level in response to canagliflozin alone, liraglutide or canagliflozin with liraglutide.

Fasting Plasma Glucose (FPG) at 4 MonthsBaseline to Approximately 4 months

Values will be presented as the mean + (Standard Deviation) SD. The difference in HGP and all secondary endpoints at study end versus baseline will be calculated and compared between each active treatment group with ANOVA.

Secondary Outcome Measures
NameTimeMethod
Body Mass Index (BMI) at 4 MonthsApproximately 4 months

A measure of BMI at 4 months to examine effects of combination therapy with liraglutide plus canagliflozin.

Trial Locations

Locations (1)

University of Texas Health Science Center at San Antonio

🇺🇸

San Antonio, Texas, United States

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