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A Study of ABBV-011 Alone and in Combination With Budigalimab (ABBV-181) in Participants With Relapsed or Refractory Small Cell Lung Cancer

Phase 1
Completed
Conditions
Small Cell Lung Cancer
Interventions
Registration Number
NCT03639194
Lead Sponsor
AbbVie
Brief Summary

This is a multicenter, open-label, Phase 1 study of ABBV-011 given as a single agent and in combination with budigalimab (ABBV-181) in participants with relapsed or refractory small cell lung cancer (SCLC). The study consists of 4 parts: Part A is a single-agent ABBV-011 dose regimen finding cohort; followed by Part B, a single-agent ABBV-011 dose expansion cohort; and then Part C, an ABBV-011 and budigalimab (ABBV-181) combination escalation and expansion cohort; Part D, single-agent ABBV-011 dose-evaluating cohort for Japan.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
132
Inclusion Criteria
  • Histologically or cytologically confirmed small cell lung cancer (SCLC) that is relapsed or refractory following at least 1 prior platinum-containing chemotherapy, but no more than 3 total prior lines of therapy, and with no curative therapy available.
  • Measurable disease, defined as at least 1 tumor lesion greater than or equal to 10 mm in the longest diameter or a lymph node greater than or equal to 15 mm in short axis measurement assessed by computed tomography (CT) scan, according to Response Evaluation Criteria in Solid Tumors (RECIST) version 1.1.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.
  • Minimum life expectancy of at least 12 weeks.
  • Recovery to at least Grade 1 of any clinically significant toxicity (excluding alopecia) prior to initiation of study drug administration.
  • Adequate hematologic, hepatic, neurologic, and renal function.
  • All participants in Part B and Part C will be required to have tumor tissue that tests positive for target expression.
  • Sponsor may elect for confirmed SCLC tumor tissue to test positive for target expression for Parts A and D participants as well.
  • Last dose of any prior anticancer therapy >= 4 weeks before the first dose of study drug.

Additional Inclusion Criteria for Study Part B and Part C:

  • SCLC tumor tissue that tests positive for seizure-related homolog 6 (SEZ6) by immunohistochemistry (IHC).
Exclusion Criteria
  • History of confirmed or suspected liver cirrhosis, hepatic veno-occlusive disease (VOD), sinusoidal obstruction syndrome (SOS), alcohol dependence, or ongoing excessive alcohol use.
  • Prior history of allogeneic or autologous stem cell transplantation.
  • Documented history of stroke or clinically significant cardiac disease as described in the protocol within 6 months prior to the first dose of study drug.
  • History of cardiac conduction abnormalities as described in the protocol.
  • Recent or ongoing serious infection, as described in the protocol.
  • Active SARS-CoV-2 infection.
  • Prior or concomitant malignancies with some exceptions, as described in the protocol.
  • Any significant medical or psychiatric condition, including any suggested by Screening laboratory findings, that in the opinion of the Investigator or Sponsor may place the participant at undue risk from the study treatment, interfere with interpretation of study results, or compromise ability to comply with protocol requirements.
  • Participants with a history of hypersensitivity to the active ingredients or any excipients of study drugs (ABBV-011 or budigalimab [ABBV-181]) will be excluded.

Additional Exclusion Criteria for Part C:

  • History of inflammatory bowel disease.
  • Peripheral neuropathy Grade 2 with pain, or Grade 3 or higher.
  • Body weight less than 35 kilograms.
  • Active pneumonitis or interstitial lung disease (ILD) or a history of pneumonitis/ILD requiring treatment with steroids.
  • Participants previously treated with an anti PD-1/PD-L1 targeting agent must meet additional criteria described in the protocol.
  • Participant is judged by the Investigator to have evidence of ongoing hemolysis.
  • Immunosuppressive use with exceptions as per protocol.
  • Participants who have received a live vaccine within 30 days of start of study treatment.
  • Active autoimmune disease with exceptions as indicated in the protocol.
  • History of primary immunodeficiency, solid organ transplantation, or previous clinical diagnosis of tuberculosis.
  • Participants with a history of Stevens-Johnson syndrome (SJS), toxic epidermal necrolysis (TEN), or drug reaction with eosinophilia and systemic symptoms (DRESS).

Additional exclusion criteria for Japanese and Korean participants:

  • Participants with a history of interstitial lung disease (pneumonitis) or current interstitial lung disease (pneumonitis).

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Part A: ABBV-011 Dose EscalationABBV-011ABBV-011 via intravenous administration at various doses and dosing regimens until the maximum tolerated dose and/or the recommended Part B dose(s) is declared.
Part C: ABBV-011 + Budigalimab Escalation and ExpansionABBV-011ABBV-011 via intravenous administration at various doses and dosing regimens starting at least 1 dose level below the recommended single-agent dose of ABBV-011 for Part B plus Budigalimab via intravenous administration at fixed doses and various dosing regimens.
Part B: ABBV-011 Dose ExpansionABBV-011ABBV-011 via intravenous administration at dose regimen(s) that will not exceed the maximum tolerated dose determined in Part A.
Part D: ABBV-011 Dose Evaluation for JapanABBV-011ABBV-011 via intravenous administration will be administered every 3 weeks (Q3wk), on Day 1 of each 21-day cycle or alternate dosing regimens.
Part C: ABBV-011 + Budigalimab Escalation and ExpansionBudigalimabABBV-011 via intravenous administration at various doses and dosing regimens starting at least 1 dose level below the recommended single-agent dose of ABBV-011 for Part B plus Budigalimab via intravenous administration at fixed doses and various dosing regimens.
Primary Outcome Measures
NameTimeMethod
Number of Participants With Adverse EventsUp to approximately 5 years after the first participant receives first dose of study drug

An adverse event (AE) is defined as any untoward medical occurrence in a patient or clinical investigation participant administered a pharmaceutical product which does not necessarily have a causal relationship with this treatment. The investigator assesses the relationship of each event to the use of study. A serious adverse event (SAE) is an event that results in death, is life-threatening, requires or prolongs hospitalization, results in a congenital anomaly, persistent or significant disability/incapacity or is an important medical event that, based on medical judgment, may jeopardize the participant and may require medical or surgical intervention to prevent any of the outcomes listed above.

Maximum Tolerated Dose (MTD) and/or the Recommended Phase 2 Dose (RPTD) of ABBV-011Up to approximately 5 years after the first participant receives first dose of study drug

The Maximum Tolerated Dose (MTD) and/or the Recommended Phase 2 Dose (RPTD) of ABBV-011 will be determined during the Part A dose escalation cohort.

Maximum Tolerated Dose (MTD) and/or the Recommended Phase 2 Dose (RPTD) of ABBV-011 in Combination with BudigalimabUp to approximately 5 years after the first participant receives first dose of study drug

The Maximum Tolerated Dose (MTD) and/or the Recommended Phase 2 Dose (RPTD) of ABBV-011 in combination with budigalimab will be determined during the Part C dose escalation cohort.

Number of Participants With Dose Limiting Toxicities (DLTs)Up to approximately 5 years after the first participant receives first dose of study drug

DLTs are adverse events as described in the protocol.

Mean Change from Baseline in Vital SignsUp to approximately 5 years after the first participant receives first dose of study drug

Mean change from Baseline in vital signs like blood pressure will be assessed.

Incidence of Laboratory AbnormaitiesUp to approximately 5 years after the first participant receives first dose of study drug

Number of participants with lab abnormalities will be assessed.

Mean Change from Baseline in Electrocardiogram (ECG) ParametersUp to approximately 5 years after the first participant receives first dose of study drug

Mean change from Baseline in ECG parameters like QTc interval will be assessed.

Secondary Outcome Measures
NameTimeMethod
Time to Maximum Serum Concentration (Tmax) of ABBV-011Up to approximately 5 years after the first participant receives first dose of study drug

Time to maximum serum concentration (Tmax) of ABBV-011.

Maximum Serum Concentration (Cmax) of ABBV-011Up to approximately 5 years after the first participant receives first dose of study drug

Maximum Serum Concentration (Cmax) of ABBV-011.

Area Under the Serum Concentration-Time Curve (AUCinf) of ABBV-011Up to approximately 5 years after the first participant receives first dose of study drug

Area under the serum concentration-time curve within a dosing interval of ABBV-011.

Area Under the Serum Concentration-Time Curve within a Dosing Interval (AUC0-t) of ABBV-011Up to approximately 5 years after the first participant receives first dose of study drug

Area under the serum concentration-time curve within a dosing interval (AUC0-t) of ABBV-011.

Observed Serum Concentration at Trough (Ctrough) of ABBV-011Up to approximately 5 years after the first participant receives first dose of study drug

Observed serum concentration at trough (Ctrough) of ABBV-011.

Apparent Terminal Half-Life (T1/2) of ABBV-011Up to approximately 5 years after the first participant receives first dose of study drug

Apparent terminal half-life (T1/2) of ABBV-011.

Accumulation Ratio of ABBV-011Up to approximately 5 years after the first participant receives first dose of study drug

Accumulation ratio of ABBV-011.

Steady State Volume of Distribution (Vss) of ABBV-011Up to approximately 5 years after the first participant receives first dose of study drug

Steady state volume of distribution (Vss) of ABBV-011.

Overall Survival (OS)Up to approximately 5 years after the first participant receives first dose of study drug

OS is defined as the time from the subject's first dose date to death due to any cause.

Serum Clearance (CL) of ABBV-011Up to approximately 5 years after the first participant receives first dose of study drug

Serum clearance of ABBV011.

Duration of Clinical Benefit (DOCB)Up to approximately 5 years after the first participant receives first dose of study drug

(DOCB) is defined as the time from the participant's initial observation of clinical benefit (CR or PR or SD) to PD or death due to any cause, whichever occurs first.

Progression-Free Survival (PFS)Up to approximately 5 years after the first participant receives first dose of study drug

PFS time is defined as the time from the subject's first dose of study drug (Day 1) to either the subject's disease progression (PD) or death due to any cause, whichever occurs first.

Incidence of Antidrug Antibodies (ADA) Against ABBV-011 or Budigalimab (ABBV-181)Up to approximately 5 years after the first participant receives first dose of study drug

Number of participants with incidence of ADAs against ABBV-011 or budigalimab will be assessed.

Objective Response Rate (ORR) as Assessed by Response Evaluation Criteria in Solid Tumors version 1.1 (RECIST v1.1)Up to approximately 5 years after the first participant receives first dose of study drug

ORR is defined as the percentage of participants with confirmed Complete Response (CR) or Partial Response (PR).

Clinical Benefit Rate (CBR)Up to approximately 5 years after the first participant receives first dose of study drug

CBR is defined as the percentage of participants with best overall response (confirmed or unconfirmed) of CR, PR or stable disease (SD).

Duration of Response (DOR)Up to approximately 5 years after the first participant receives first dose of study drug

DOR is defined as the time from the participant's initial objective response (CR or PR) to Progressive Disease (PD) or death due to any cause, whichever occurs first.

Trial Locations

Locations (32)

UH Cleveland Medical Center /ID# 207561

🇺🇸

Cleveland, Ohio, United States

The Ohio State University /ID# 207552

🇺🇸

Columbus, Ohio, United States

Highlands Oncology Group, PA /ID# 207176

🇺🇸

Springdale, Arkansas, United States

NEXT Oncology /ID# 207167

🇺🇸

San Antonio, Texas, United States

Massachusetts General Hospital /ID# 207549

🇺🇸

Boston, Massachusetts, United States

University of Michigan Comprehensive Cancer Center /ID# 207177

🇺🇸

Ann Arbor, Michigan, United States

Univ of Wisconsin Hosp/Clinics /ID# 207556

🇺🇸

Madison, Wisconsin, United States

Dana-Farber Cancer Institute /ID# 213032

🇺🇸

Boston, Massachusetts, United States

University of Washington /ID# 207557

🇺🇸

Seattle, Washington, United States

Shizuoka Cancer Center /ID# 230911

🇯🇵

Sunto-gun, Shizuoka, Japan

Duke Cancer Center /ID# 207547

🇺🇸

Durham, North Carolina, United States

Wakayama Medical University Hospital /ID# 229111

🇯🇵

Wakayama-shi, Wakayama, Japan

Seoul National University Bundang Hospital /ID# 234274

🇰🇷

Seongnam, Gyeonggido, Korea, Republic of

Tennessee Oncology, PLLC /ID# 207175

🇺🇸

Nashville, Tennessee, United States

Memorial Sloan Kettering Cancer Center-Koch Center /ID# 208216

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New York, New York, United States

Hokkaido Cancer Center /ID# 229101

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Sapporo-shi, Hokkaido, Japan

National Cheng Kung University Hospital /ID# 234267

🇨🇳

Tainan, Taiwan

National Cancer Center Hospital East /ID# 230943

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Kashiwa-shi, Chiba, Japan

Asan Medical Center /ID# 234273

🇰🇷

Seoul, Korea, Republic of

Yale School of Medicine /ID# 207559

🇺🇸

New Haven, Connecticut, United States

University of Iowa Hospitals and Clinics /ID# 207560

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Iowa City, Iowa, United States

Washington University-School of Medicine /ID# 207168

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Saint Louis, Missouri, United States

Henry Ford Hospital /ID# 233539

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Detroit, Michigan, United States

Vanderbilt Ingram Cancer Center /ID# 207551

🇺🇸

Nashville, Tennessee, United States

National Cancer Center /ID# 240169

🇰🇷

Goyang, Gyeonggido, Korea, Republic of

Yonsei University Health System Severance Hospital /ID# 239515

🇰🇷

Seoul, Seoul Teugbyeolsi, Korea, Republic of

Seoul National University Hospital /ID# 234272

🇰🇷

Seoul, Korea, Republic of

University of Alabama at Birmingham - Main /ID# 207295

🇺🇸

Birmingham, Alabama, United States

University of Kentucky Chandler Medical Center /ID# 208217

🇺🇸

Lexington, Kentucky, United States

University of California, Davis Comprehensive Cancer Center /ID# 207548

🇺🇸

Sacramento, California, United States

University of Utah /ID# 207553

🇺🇸

Salt Lake City, Utah, United States

National Hospital Organization Shikoku Cancer Center /ID# 229737

🇯🇵

Matsuyama-shi, Ehime, Japan

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