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Orexin Receptor Antagonists as Modulators of Threat Sensitivity in Individuals With Alcohol Use Disorder

Early Phase 1
Active, not recruiting
Conditions
Alcohol Use Disorder
Interventions
Other: Placebo
Registration Number
NCT05656534
Lead Sponsor
Ohio State University
Brief Summary

The goal of this double-blind clinical trial is to further explore if, how, and for whom orexin antagonism modifies brain-behavior stress targets in moderate to severe alcohol use disorder (AUD). The main questions it aims to answer are:

* Does an acute dose of suvorexant (SUV) and/or daily use of SUV modify brain-behavior targets of AUD dysfunction?

* Does daily SUV use change alcohol behavior and if so, is this change in behavior linked to brain-behavior change?

Participants will be randomized to a treatment group (SUV or placebo) and protocol arm, electromyography (EMG) only or EMG+functional magnetic resonance imaging (fMRI). Participants will be asked to complete the following:

* Baseline lab visit(s) that include the psychophysiological stress paradigm (EMG only or EMG+fMRI, dependent upon randomization).

* Acute drug challenge where the participant will return to the lab to repeat the stress paradigm following administration of a single dose of either 10mg SUV or placebo.

* Medication trial where participants will be instructed to take 10mg capsules of SUV or placebo orally each night before bedtime for 4-weeks.

* Daily reports of medication adherence, side-effects, sleep, alcohol use, and mood will be collected via smartphones during the 4-week medication trial.

* Post-treatment lab visit(s) where participants will return to the lab at the end of the medication trial and complete the same stress paradigm from baseline (EMG only or EMG+fMRI, dependent upon randomization).

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
71
Inclusion Criteria
  • Age 18-65.
  • Participant is able to give informed consent.
  • Generally medically and physically healthy as confirmed by medical history.
  • Meet DSM-5 diagnostic criteria for current moderate or severe AUD.
  • Engage in heavy alcohol use defined as drinking equal or greater than 14 standard drinks per week if male and equal or greater than 7 standard drinks per week if female.
Exclusion Criteria
  • Clinically significant medical or neurological condition (e.g., liver disease, narcolepsy, complex sleep behaviors, severe hepatic impairment, COPD, severe obstructive sleep apnea).
  • Current cognitive dysfunction (traumatic brain injury, mental retardation, organic mental syndrome, pervasive developmental disorder, or dementia).
  • Current use of antihistamines, strong or moderate inhibitors of CYP3A liver enzymes, strong CYP3A inducers, or digoxin.
  • Current or past DSM-5 diagnosis of mania, schizophrenia, psychosis, suicidality, major depressive disorder, or obsessive compulsive disorder.
  • Current substance use disorder other than alcohol or mild cannabis use disorder.
  • Treatment seeking for AUD.
  • Recent psychotropic medication use in the past 2 months.
  • Currently smokes 5 or more cigarettes (or electronic equivalent) per day.
  • BMI equal or greater than 35.
  • Engage in night-shift work.
  • Lack of fluency in English.
  • Presence of ferrous-containing metal in the body.
  • Inability to tolerate small, enclosed spaces.
  • Deafness in one or both ears.
  • Currently pregnant (positive pregnancy test), lactating, or not agreeing to use birth control methods during the duration of the trial.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Suvorexant TreatmentSuvorexantIndividuals will take 10mg of suvorexant (Merck \& Co Inc.) during the Acute Drug Challenge and daily for 28 days.
ControlPlaceboIndividuals will take a placebo pill during the Acute Drug Challenge and daily for 28 days.
Primary Outcome Measures
NameTimeMethod
Startle reactivity to stress with an acute dose of suvorexant.Change from baseline to 2 hours post-ingestion of an acute dose of suvorexant.

Changes in acoustic startle electromyographic (EMG) response during stress anticipation following an acute dose of suvorexant.

Alcohol behavior and daily use of suvorexant.Change from baseline to post-treatment, up to 1.5-2 months.

Changes in proportion of heavy drinking days and drinks per drinking day following daily use of suvorexant.

Startle reactivity to stress with daily use of suvorexant.Change from baseline to post-treatment, up to 1.5-2 months.

Changes in acoustic startle electromyographic (EMG) response during stress anticipation following daily use of suvorexant.

Secondary Outcome Measures
NameTimeMethod
Brain change and daily use of suvorexant.Change from baseline to post-treatment, up to 1.5-2 months.

Changes in the anterior insula (aINS) and dorsal anterior cingulate cortex (dACC) reactivity and connectivity during stress anticipation following daily use of suvorexant.

Trial Locations

Locations (1)

The Ohio State University

🇺🇸

Columbus, Ohio, United States

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